α-adrenoceptor — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T5S2059	Glaucine		Calcium Channel , Dopamine Receptor , Influenza Virus , Adrenergic Receptor , PDE
	Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 production. Glaucine can inhibit the migration and invasion of h...
T0042	Xylometazoline hydrochloride	Xylometazoline HCl	Adrenergic Receptor
	Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.		Adrenergic Receptor
T30027	Amosulalol		Adrenergic Receptor
	Amosulalol is a combined alpha and beta adrenoceptor antagonist.		Adrenergic Receptor
T23397	ST 91		Others , Adrenergic Receptor
	ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.		Others , Adrenergic Receptor
T26923	Bunazosin Hydrochloride	E 1015,E643,E-1015,E-643,E 643	Adrenergic Receptor
	Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.		Adrenergic Receptor
T1247	Clonidine hydrochloride	Clonidine HCl,Catapres	Adrenergic Receptor
	Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.		Adrenergic Receptor
T10003	α1 adrenoceptor-MO-1		Others
	α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enantiomer.		Others
T35326	Labetalone hydrochloride	Labetalone hydrochloride,Benzoic amide	Others
	Labetalone hydrochloride (Benzoic amide) is an impurity of Labetalol. Labetalol is an orally active adrenoceptor blocking drug, Labetalol is a competitive antagonist at both alpha- and beta-adrenoceptor sites		Others
T7728	ACEPROMAZINE MALEATE		Dopamine Receptor
	ACEPROMAZINE MALEATE is a dopamine receptor antagonist		Dopamine Receptor
TN1922	Meranzin hydrate		ERK , Adrenergic Receptor
	Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptors; it produ...		ERK , Adrenergic Receptor
T10364	Arbutamine	GP 21213	Adrenergic Receptor
	Arbutamine (GP 21213) is a novel potent non-selective beta-adrenoceptor agonist with alpha-1-sympathomimetic activity.Arbutamine promotes cardiac stress and increases heart rate, cardiac contractility.Arbutamine can be u...		Adrenergic Receptor
T68138	Saterinone		Adrenergic Receptor , PDE
	Saterinone is a potent and selective phosphodiesterase III inhibitor and a potent antagonist of the vascular α-1-adrenoceptor. Saterinone has vasodilatory properties and can be used in the acute treatment of chronic hear...		Adrenergic Receptor , PDE
T0696	Naftopidil	KT-611,BM-15275	Adrenergic Receptor
	Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.		Adrenergic Receptor
T1158	Phenoxybenzamine hydrochloride	NCI-c01661,NSC 37448,Phenoxybenzamine HCl	CaMK , Adrenergic Receptor
	Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihypertensive and vasodilatory properties. Phenoxybenzamine non...		CaMK , Adrenergic Receptor
T1275	Phentolamine mesylate	Phentolamine methanesulfonate,Phentolamine mesilate	Adrenergic Receptor
	Phentolamine mesylate (Phentolamine methanesulfonate) is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma, vasospasm of RAYNAUD DISEAS...		Adrenergic Receptor
T2594	Dextromilnacipran	Levomilnacipran	Serotonin Transporter , Norepinephrine
	Dextromilnacipran (Levomilnacipran) is a selective serotonin and norepinephrine reuptake inhibitor.		Serotonin Transporter , Norepinephrine
T61165	Indoramin
	Indoramin, an orally active antihypertensive agent, exhibits selectivity for the α 1A -adrenoceptor [1].
T12815	(S)-Terazosin		Adrenergic Receptor
	(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with Ki values of 3.91 nM, 0.79 nM and 1.16 nM, respectively).		Adrenergic Receptor
TN1577	Dicentrine		Others
	Dicentrine, a selective α±(1)-adrenoceptor antagonist with potent antiarrhythmic and antihypertensive activities, it also has antinociception in different models of chemical pain.		Others
T64314	OxyMetazoline
	OxyMetazoline is an α-adrenoceptor agonist that acts on α1A (IC50: 0.02 μM), α1B (IC50: 0.25 μM), α2A (IC50: 0.58 μM) and α2C (IC50: 0.13 μM). OxyMetazoline can be used in studies to relieve nasal mucosal congestion.