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Search Result

Search Results for " neurotensin "

Targets

Neurotensin Receptor Neurotensin Receptor

46

Compounds

5

Recombinant Proteins

Cat No. Product Name Synonyms Targets
TP1310 Neurotensin Neurotensin Receptor
Neurotensin is a 13 amino acid neuropeptide that is implicated in the regulation of luteinizing hormone and prolactin release and has significant interaction with the dopaminergic system.
T7617 Neurotensin(8-13) Neurotensin(8-13)(3TFA) Neurotensin Receptor
Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.
T38807L [Lys8, Lys9]-Neurotensin (8-13) acetate Neurotensin Receptor
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2, with Ki values of 0.33 nM and 0.95 nM for hNTS1 and hNTS2 r...
T7617L Neurotensin(8-13) 3TFA(60482-95-3(free base)) Neurotensin Receptor
Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.
TP2309 NEUROTENSIN TFA (39379-15-2 free base) Pyr-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu-OH TFA（55508-42-4 free base),NEUROTENSIN TFA Others
Neurotensin TFA (39379-15-2 free base) is an endogenous 13 amino acid neuropeptide with profound opioid-independent analgesic effects. It behaves as a neurotransmitter in the brain, as a hormone in the gut, and also as a...
T40850 [D-Trp11]-Neurotensin [D-Trp11]-Neurotensin
[D-Trp11]-Neurotensin is a compound that functions as a selective antagonist of Neurotensin (NT) in perfused rat hearts, while exhibiting full agonist properties in guinea pig atria and rat stomach strips. Additionally, ...
T38807 [Lys8, Lys9]-Neurotensin (8-13) JMV438,[Lys8, Lys9]-Neurotensin (8-13)
[Lys8, Lys9]-Neurotensin (8-13) (JMV438) is a Neurotensin analog that elicits analgesic effects by activating the G protein-coupled receptors NTS1 and NTS2. The compound has K i values of 0.33 nM and 0.95 nM for hNTS1 an...
TP2393 Neurotensin-related hexapeptide Lant-6
Neurotensin-related hexapeptide exists in retinal ganglion cells and in their central projections in pigeons and may be utilized as a neuroactive substance by the central terminals of numerous retinal ganglion cells in b...
T33656 Neurotensin (1-6)
Neurotensin (1-6) affects dopamine release from striatum.
T76572 Acetyl neurotensin (8-13)
Acetyl neurotensin (8-13), the most concise analog of neurotensin, retains complete binding and pharmacological properties [1].
T16860 SBI-553 Neurotensin Receptor
SBI-553 is an effective and brain penetrant NTR1 allosteric modulator (EC50: 0.34 μM).
TQ0086 AF38469 AF-38469 Neurotensin Receptor
AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).
T9044 SORT-PGRN interaction inhibitor 1 Neurotensin Receptor
SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).
T8657 KYP-2047 Others
KYP-2047 is a very potent, selective Prolyl oligopeptidase (POP) inhibitor.
T23386 SR 142948 Neurotensin Receptor
SR 142948 is a neurotensin (NT) receptor antagonist.
T11861 LM11A-31 dihydrochloride Others
LM11A-31 dihydrochloride is a water-soluble, non-peptide with high blood-brain barrier permeability.LM11A-31 dihydrochloride, a p75NTR (neurotrophin receptor p75) Ligand, is a potent proNGF (nerve growth factor) antagoni...
T7615 Xenopsin Xenopsin(2TFA) Others
Xenopsin (Xenopsin(2TFA))(2TFA) is a neurotensin-like octapeptide previously isolated from amphibian skin.
T16034 Meclinertant SR 48692 Others
Meclinertant is an effective, selective, nonpeptide, and orally active neurotensin receptor 1 (NTS1) antagonist. Meclinertant competitively antagonizes neurotensin-induced intracellular Ca2+ mobilization (pA2 : 8.13), in...
T28217 NTRC-844 NTRC 844,NTRC844 Neurotensin Receptor
NTRC-844 is a selective rat neurotensin receptor type 2 (NTS2) antagonist that shows analgesic activity in animal models of pain.
T7615L Xenopsin 2TFA(51827-01-1(free base) Others
Xenopsin(2TFA) is a neurotensin-like octapeptide previously isolated from amphibian skin.
TP1116L Kinetensin acetate(103131-69-7 free base) Kinetensin (human) acetate Neurotensin Receptor
Kinetensin acetate(103131-69-7 free base) is isolated from pepsin-treated human plasma. Kinetensin acetate(103131-69-7 free base) is a neurotensin-like peptide.
TP2209L Xenin 8 acetate Xenin 8 acetate (117442-28-1 Free base) IGF-1R
Xenin 8 acetate is a biologically active fragment of Xenin in the neurotensin/xenopsin family. Xenin 8 acetate augments Arginine-induced insulin release (by 40%) and potentiates the glucagon responses to both Arginine (b...
TP1085L Neuromedin N acetate(92169-45-4 free base) Neuromedin N (rat, mouse, porcine, canine) acetate Dopamine Receptor
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.Neuromedin N is a potent modulator of d...
T37529 TC NTR1 17
Non-peptide neurotensin receptor 1 (NTS1) partial agonist (EC50 <15.6 nM and Emax = 63% of neurotensin response in Ca2+ mobilization assay). Exhibits over 50-fold selectivity for NTS1 over NTS2 and GPR35. Hershberger et ...
T16358 NTRC-824 Others
NTRC-824 is >150-fold selectivity for NTS2 over NTS1 (Ki >30 μM). NTRC-824 is an effective, selective, and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist (IC50: 38 nM and a Ki : 202 nM).
T32700 Levocabastine Livostin,Bilina
Levocarbastine is a second-generation H1 receptor antagonist for allergic conjunctivitis. It also acts as a potent selective antagonist for the neurotensin receptor NTS2 and is the first drug to be used to characterize d...
T75711 Contulakin G
Contulakin G, an O-glycosylated invertebrate neurotensin, serves as a weaker agonist for the neurotensin receptor. Additionally, it is recognized as a potent antinociceptive agent [1] [2].
T70271 PD-149163
PD-149163 is a selective, brain penetrating Neurotensin NTR1 receptor agonist. Neurotensin agonists block the pre-pulse inhibition deficits produced by a 5-HT2A and an α1 agonist. As a result, PD-149163 shows pro-cogniti...
TQ0075 ML314 Neurotensin Receptor
ML314 is a brain-permeable nonpeptide β-inhibin-biased neurotensin NTR1 receptor agonist (EC50: 1.9 μM), a biased neurotensin receptor ligand for methamphetamine abuse that inhibits NTR2 and GPR35.
T13530 AF40431 Others
AF40431 is the first reported small-molecule ligand of sortilin (IC50: 4.4 µM; Kd: 0.7 µM). AF40431 is bound in the neurotensin-binding site of sortilin.
TP2209 Xenin-8 Others
neurotensin-like peptide that modulate pancreatic insulin and glucagon secretion/effects
T24279 L 156903 L-156903,L156903
L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.
TP2462 Magaratensin Asp-lys-arg-pro-tyr-ile-leu-his-glu
Magaratensin is a neurotensin-related peptide related to the skin of Rana margarate.
T75868 JMV 449 acetate
JMV 449 acetate is a potent neurotensin receptor agonist. JMV 449 acetate shows an IC 50 of 0.15 nM for inhibition of 125 I-neurotensin binding to neonatal mouse brain and an EC 50 of 1.9 nM in contracting the guinea-pig...
T28845 SR142948A HCl SR142948A,SR 142948A,SR-142948A,SR142948A hydrochloride
SR 142948A is a non-peptide antagonist of neurotensin receptor. SR 142948A affects the expression of c-Fos and has properties of antipsychotic agent. SR 142948A blocks hypothermia and analgesia induced by neurotensin. It...
TP1116 Kinetensin Kinetensin (human)
Kinetensin is a neurotensin-like peptide.
TP1085 Neuromedin N Neuromedin N (rat, mouse, porcine, canine)
Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.
TP1482 Xenopsin TFA (51827-01-1 free base) Xenopsin TFA
Xenopsin TFA is a neurotensin-like octapeptide derived from the skin of xenopus xenopus.Xenopsin TFA is an inhibitor of tetrachloroside to stimulate gastric acid secretion.
T72410 Sortilin antagonist 1
Sortilin Antagonist 1, a potent sortilin antagonist, exhibits an inhibition constant (IC50) of 20 nM against Neurotensin (NTS) binding to sortilin. Neurotensin acts as a sortilin ligand. This compound is utilized in neur...
TP2012 JMV 449
Potent, metabolically stable neurotensin receptor agonist peptide (IC50 = 0.15 nM for inhibition of [125I]-NT binding to neonatal mouse brain; EC50 = 1.9 nM for contraction of guinea pig ileum). Produces long-lasting hyp...
T80765 Xenopsin TFA
Xenopsin TFA is a neurotensin-like octapeptide derived from the skin of Xenopus laevis [1] and serves as an inhibitor of Tetragastrin-induced gastric acid secretion [2].
T78954 HNTS1R agonist-1 Neurotensin Receptor
Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (BBB). It not only enhances motor function but also improves ...
T82647 Cyanine5 NHS ester bromide
Cyanine5 NHS ester bromide, a cyanine dye and active compound, is utilized for labeling amino groups in peptides, proteins, and oligonucleotides. It specifically labels fluorescence neurotensin (8-13) through arginine re...
T80766 Xenin-8 TFA
Xenin-8 TFA, a C-terminal octapeptide derived from the 25-amino acid peptide Xenin belonging to the neurotensin/xenopsin family, is biologically active. It enhances basal insulin secretion and amplifies glucose-stimulate...
T70039 BIM-46174
BIM-46174 is a New Inhibitor of the Heterotrimeric Gα/Gβγ Protein Complex. BIM-46174 acts as a selective inhibitor of heterotrimeric G-protein complex. BIM-46174 prevents the heterotrimeric G-protein signaling linked to...
T73677 SR 142948 dihydrochloride
SR 142948 dihydrochloride is a selective, orally active, non-peptide neurotensin receptor (NT) antagonist, featuring IC50 values of 1.19 nM, 0.32 nM, and 3.96 nM in h-NTR1-CHO cells, HT-29 cells, and adult rat brain, res...

Compounds

Neurotensin
TP1310
Synonym:
Target: Neurotensin Receptor
Neurotensin(8-13)
T7617
Synonym: Neurotensin(8-13)(3TFA)
Target: Neurotensin Receptor
[Lys8, Lys9]-Neurotensin (8-13) acetate
T38807L
Synonym:
Target: Neurotensin Receptor
Neurotensin(8-13) 3TFA(60482-95-3(free base))
T7617L
Synonym:
Target: Neurotensin Receptor
NEUROTENSIN TFA (39379-15-2 free base)
TP2309
Synonym: Pyr-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu-OH TFA（55508-42-4 free base),NEUROTENSIN TFA
Target: Others
[D-Trp11]-Neurotensin
T40850
Synonym: [D-Trp11]-Neurotensin
Target:
[Lys8, Lys9]-Neurotensin (8-13)
T38807
Synonym: JMV438,[Lys8, Lys9]-Neurotensin (8-13)
Target:
Neurotensin-related hexapeptide
TP2393
Synonym: Lant-6
Target:
Neurotensin (1-6)
T33656
Synonym:
Target:
Acetyl neurotensin (8-13)
T76572
Synonym:
Target:
SBI-553
T16860
Synonym:
Target: Neurotensin Receptor
AF38469
TQ0086
Synonym: AF-38469
Target: Neurotensin Receptor
SORT-PGRN interaction inhibitor 1
T9044
Synonym:
Target: Neurotensin Receptor
KYP-2047
T8657
Synonym:
Target: Others
SR 142948
T23386
Synonym:
Target: Neurotensin Receptor
LM11A-31 dihydrochloride
T11861
Synonym:
Target: Others
Xenopsin
T7615
Synonym: Xenopsin(2TFA)
Target: Others
Meclinertant
T16034
Synonym: SR 48692
Target: Others
NTRC-844
T28217
Synonym: NTRC 844,NTRC844
Target: Neurotensin Receptor
Xenopsin 2TFA(51827-01-1(free base)
T7615L
Synonym:
Target: Others
Kinetensin acetate(103131-69-7 free base)
TP1116L
Synonym: Kinetensin (human) acetate
Target: Neurotensin Receptor
Xenin 8 acetate
TP2209L
Synonym: Xenin 8 acetate (117442-28-1 Free base)
Target: IGF-1R
Neuromedin N acetate(92169-45-4 free base)
TP1085L
Synonym: Neuromedin N (rat, mouse, porcine, canine) acetate
Target: Dopamine Receptor
TC NTR1 17
T37529
Synonym:
Target:
NTRC-824
T16358
Synonym:
Target: Others
Levocabastine
T32700
Synonym: Livostin,Bilina
Target:
Contulakin G
T75711
Synonym:
Target:
PD-149163
T70271
Synonym:
Target:
ML314
TQ0075
Synonym:
Target: Neurotensin Receptor
AF40431
T13530
Synonym:
Target: Others
Xenin-8
TP2209
Synonym:
Target: Others
L 156903
T24279
Synonym: L-156903,L156903
Target:
Magaratensin
TP2462
Synonym: Asp-lys-arg-pro-tyr-ile-leu-his-glu
Target:
JMV 449 acetate
T75868
Synonym:
Target:
SR142948A HCl
T28845
Synonym: SR142948A,SR 142948A,SR-142948A,SR142948A hydrochloride
Target:
Kinetensin
TP1116
Synonym: Kinetensin (human)
Target:
Neuromedin N
TP1085
Synonym: Neuromedin N (rat, mouse, porcine, canine)
Target:
Xenopsin TFA (51827-01-1 free base)
TP1482
Synonym: Xenopsin TFA
Target:
Sortilin antagonist 1
T72410
Synonym:
Target:
JMV 449
TP2012
Synonym:
Target:
Xenopsin TFA
T80765
Synonym:
Target:
hNTS1R agonist-1
T78954
Synonym:
Target: Neurotensin Receptor
Cyanine5 NHS ester bromide
T82647
Synonym:
Target:
Xenin-8 TFA
T80766
Synonym:
Target:
BIM-46174
T70039
Synonym:
Target:
SR 142948 dihydrochloride
T73677
Synonym:
Target:

Recombinant Proteins

Species：
Human (2)
Mouse (2)
Cynomolgus (1)
Expression System：
HEK293 Cells (3)
Baculovirus Insect Cells (1)
E. coli (1)
Tag：
C-hFc (2)
C-His (1)
N-6xHis-SUMO (1)
N-His (1)
Cat No. Product Name Species Expression System
TMPY-00561 Neurotensin Protein, Human, Recombinant (hFc) Human HEK293 Cells
NTS (Neurotensin) is a Protein Coding gene. This gene encodes a common precursor for two peptides, neuromedin N and neurotensin. NTS is a neuropeptide distributed in the central nervous and digestive systems. It belongs ...
TMPK-00982 NTS1 Protein, Cynomolgus, Recombinant (His) Cynomolgus HEK293 Cells
Crystal structures of neurotensin receptor subtype 1 (NTS1) allowed us to visualize the binding mode of the endogenous peptide hormone neurotensin and its pharmacologically active C-terminal fragment NT(8-13) within the ...
TMPK-01162 NTS1 Protein, Mouse, Recombinant (hFc) Mouse HEK293 Cells
Crystal structures of neurotensin receptor subtype 1 (NTS1) allowed us to visualize the binding mode of the endogenous peptide hormone neurotensin and its pharmacologically active C-terminal fragment NT(8-13) within the ...
TMPH-01041 Carboxypeptidase A6 Protein, Human, Recombinant (His & SUMO) Human E. coli
May be involved in the proteolytic inactivation of enkephalins and neurotensin in some brain areas. May convert inactive angiotensin I into the biologically active angiotensin II. Releases a C-terminal amino acid, with p...
TMPY-03269 Prolyl Endopeptidase Protein, Mouse, Recombinant (His) Mouse Baculovirus Insect Cells
Prolyl endopeptidase, also known as PREP, belongs to a distinct class of serine peptidases. It is a large cytosolic enzyme which was first described in the cytosol of rabbit brain as an oligopeptidase. Prolyl endopeptida...
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