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Urantide acetate(669089-53-6 free base)

🥰Excellent
Catalog No. TP2106L

Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors).

Urantide acetate(669089-53-6 free base)
Other Forms of Urantide acetate(669089-53-6 free base):
UrantideTP2106669089-53-6
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Urantide acetate(669089-53-6 free base)

🥰Excellent
Purity: 99.22%
Catalog No. TP2106L
Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors).
Pack SizePriceAvailabilityQuantity
1 mg$115In Stock
5 mg$233In Stock
10 mg$335In Stock
25 mg$565In Stock
50 mg$812In Stock
100 mg$1,130In Stock
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Purity:99.22%
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COA HPLC MS

Product Introduction

Bioactivity
Description
Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acetylcholine-induced relaxation. Behaves as a partial agonist in a calcium mobilization assay (in CHO cells expressing hUT receptors).
Chemical Properties
Molecular Weight1135.31
FormulaC53H70N10O14S2
SmilesCC([C@@H](C(O)=O)NC([C@@H]1CSSC(C)([C@H](C(N[C@H](C(N[C@@H](C(N[C@H](C(N[C@H](C(N1)=O)Cc2ccc(O)cc2)=O)CCCN)=O)Cc(c[nH]3)c4c3cccc4)=O)Cc5ccccc5)=O)NC([C@H](CC(O)=O)N)=O)C)=O)C.CC(O)=O
Relative Density.no data available
ColorWhite
AppearanceSolid
SequenceH-Asp-D-Pen(1)-DL-Phe-D-Trp-Orn-DL-Tyr-DL-Cys(1)-Val-OH
Sequence ShortDXFWXYCV
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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Keywords

urotensin-II (UT)Urantide acetate(669089-53-6 free base)Urantide acetate(669089536 free base)Urantide acetate(669089 53 6 free base)NeurotensinReceptorNeurotensin Receptor
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