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Targets

Compounds

Cat No. Product Name
T14349 Auristatin F Microtubule Associated
Auristatin F 是一种有效的微管抑制剂和血管损伤剂。 Auristatin F 可用于抗体-药物偶联物。
T13278 Valecobulin hydrochloride CKD-516 hydrochloride Microtubule Associated
Valecobulin hydrochloride 是 S516 的缬氨酸前体药和血管阻断剂。Valecobulin hydrochloride 对β-微管蛋白聚合有强效的抑制作用,对小鼠和人类的实体肿瘤具有显著的抗肿瘤活性。
T37024 Mca-DEVDAPK(Dnp)-OH
T2511 Plinabulin 普那布林,NPI-2358 Microtubule Associated
Plinabulin 是一种抗微管蛋白解聚肿瘤细胞的血管破坏剂,选择性地靶向并结合到微管蛋白的秋水仙碱结合位点,从而中断微管动力学的平衡。它对人肿瘤细胞系具有抑制作用,对 HT-29 细胞系的IC50值为 9.8 nM。
T68273 BNC105P
BNC105P is a benzofuran-based vascular disrupting agent (VDA) prodrug with potential anti-vascular and antineoplastic ac...
Auristatin F
T14349
synonym:
Target:
Valecobulin hydrochloride
T13278
synonym: CKD-516 hydrochloride
Target:
Mca-DEVDAPK(Dnp)-OH
T37024
synonym:
Target:
Plinabulin
T2511
synonym: 普那布林,NPI-2358
Target:
BNC105P
T68273
synonym:
Target: