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Search Results for "ligands for target protein for protac"

Compounds

Cat No. Product Name
T2110 (+)-JQ-1 JQ1 Epigenetic Reader Domain , Autophagy
(+)-JQ-1 是一种有效特异性的可逆 BET 溴结构域抑制剂,可激活自噬,抑制BRD4(1/2)的IC50分别为 77 nM 和 33 nM。
T10359 AR antagonist 1 Androgen Receptor
AR antagonist 1 是 AR 拮抗剂,能够与 E3 连接酶配体结合,与 VHL 蛋白结合亲和力较弱,用于 PROTACARD-266 合成。
T5480 BI-4464 FAK
BI-4464 是一种高选择性的 ATP 竞争性 PTK2/FAK 抑制剂,IC50=17 nM。它可用于PROTAC 降解剂的 PTK2 配体。
T12186 Navitoclax-piperazine ABT-263-piperazine BCL
Navitoclax-piperazine 是一种特大型 B 细胞淋巴瘤(BCL-XL)抑制剂。它和 E3 泛素连接酶的 VHL 配体可用来合成 PROTAC DT2216。
T19301 DUPA N,N''-Carbonylbis[L-glutamic acid],(2S,2'S)-2,2'-Carbonylbis(Azanediyl)Dipentanedioic Acid Others
DUPA 是谷氨酸脲,在药物偶联中作为靶向部分,可选择靶向性地将细胞毒性药物递送到前列腺癌细胞。
T1835 Ibrutinib 依鲁替尼,伊布替尼,PCI-32765 Src , BTK , Tyrosine Kinases
Ibrutinib 是一种不可逆的、选择性的 Btk 抑制剂,IC50=0.5 nM,它是一种 Btk 配体,用于合成一系列 PROTAC 分子,如 P13I。P13I 作用于人 Burkitt’s 淋巴瘤 RAMOS 细胞,浓度为 10 ...
T39910 Desmorpholinyl Navitoclax-NH-Me Desmorpholinyl ABT-263-NH-Me,Desmorpholinyl Navitoclax-NH-Me BCL
Desmorpholinyl Navitoclax-NH-Me is a Bcl-xL inhibitor, which can be employed alongside a CRBN ligand to synthesize XZ739...
T2066 Quizartinib 奎扎替尼,AC220 Apoptosis , FLT , Autophagy
Quizartinib 是一种具有口服活性的高选择性Ⅱ 型 FLT3酪氨酸激酶抑制剂,可诱导细胞凋亡。它抑制 Wt FLT3 和 突变型 FLT3-ITD 自磷酸化,IC50分别为 4.1 nM 和 1.1 nM。它可通过优化的 linke...
T15125 Diethylene Glycol Monobenzyl Ether Others
Diethylene Glycol Monobenzyl Ether is a PEG-based linker, specifically designed for the synthesis of PROTACs[1]. It serv...
T17345 7-Octynoic acid Others
7-Octynoic acid (compound 42) serves as a PROTAC linker for synthesizing various PROTACs, which are composed of two dist...
T18542 Phthalimide-PEG3-C2-OTs Others
Phthalimide-PEG3-C2-OTs (Compound 5) is a PROTAC linker composed of PEGs. It is utilized in the synthesis of various PRO...
(+)-JQ-1
T2110
synonym: JQ1
Target:
AR antagonist 1
T10359
synonym:
Target:
BI-4464
T5480
synonym:
Target:
Navitoclax-piperazine
T12186
synonym: ABT-263-piperazine
Target:
DUPA
T19301
synonym: N,N''-Carbonylbis[L-glutamic acid],(2S,2'S)-2,2'-Carbonylbis(Azanediyl)Dipentanedioic Acid
Target:
Ibrutinib
T1835
synonym: 依鲁替尼,伊布替尼,PCI-32765
Target:
Desmorpholinyl Navitoclax-NH-Me
T39910
synonym: Desmorpholinyl ABT-263-NH-Me,Desmorpholinyl Navitoclax-NH-Me
Target:
Quizartinib
T2066
synonym: 奎扎替尼,AC220
Target:
Diethylene Glycol Monobenzyl Ether
T15125
synonym:
Target:
7-Octynoic acid
T17345
synonym:
Target:
Phthalimide-PEG3-C2-OTs
T18542
synonym:
Target: