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Search Result

Search Results for " gep "

Targets

CGRP Receptor

22

Compounds

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T4610 Rimegepant BMS 927711,BMS-927711,BMS927711,BHV-3000 CGRP Receptor
Rimegepant (BMS 927711) is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.
T19917 Gepirone 5-HT Receptor
Gepirone is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone HCl possesses greater selectivity for the 5-HT1A receptor than SSRIs.
T12293L Olcegepant BIBN-4096,BIBN 4096BS CGRP Receptor
Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP).
T8682 Vazegepant hydrochloride Vazegepant HCl CGRP Receptor
Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.
T12375 Fezagepras sodium Setogepram sodium salt,PBI-4050 sodium salt GPR
Fezagepras sodium (Setogepram sodium salt) is an orally active GPR40 agonist and is an antagonist or inverse agonist for GPR84, with anti-fibrotic, anti-inflammatory and anti-proliferative actions.
T17194 Ubrogepant MK-1602 CGRP Receptor
Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.
T12883 Fezagepras PBI-4050,Setogepram GPR
Fezagepras (Setogepram) is an orally active GPR40 agonist and is an antagonist or inverse agonist of GPR84 with anti-inflammatory, anti-fibrotic, and anti-proliferative actions.
T11314 Fosmanogepix APX001,E1211 Others
Fosmanogepix (APX001) is a first-in-class, orally available broad-spectrum antifungal agent. It acts as an N-phosphonooxymethyl prodrug that undergoes rapid and complete metabolism by systemic alkaline phosphatases. This...
T73703 (3R,5R,6S)-Atogepant
Atogepant ((3R,5R,6S)-MK-8031) is the enantiomer of itself and serves as a calcitonin gene-related peptide (CGRP) receptor antagonist, primarily utilized in migraine research.
T73216 Gepefrine
Gepefrine, an orally active pressor and sympathomimetic agent, enhances the initial orthostatic regulation of arterial pressure.
T38734 Vazegepant Zavegepant,BHV-3500
Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.
T26682 Atogepant MK 8031,MK8031. Atogepant,MK-8031
Atogepant is an antagonist of calcitonin gene-related peptide receptor.
T12293 Olcegepant hydrochloride BIBN-4096 hydrochloride,BIBN4096BS hydrochloride Others
Olcegepant hydrochloride is a potent and selective non-peptidethe calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (with IC50 of 0.03 nM for human CGRP).
T79049 Tegeprotafib PTPN2/1-IN-1 Phosphatase
Tegeprotafib (PTPN2/1-IN-1) (Compound 124) is an orally active inhibitor targeting both PTPN2 and PTPN1B, displaying potent IC50 values at 4.4 nM for PTPN2 and 1-10 nM for PTPN1B, respectively [1].
T70358 Gepotidacin mesylate dihydrate
Gepotidacin mesylate dihydrate, also known as GSK-2140944 mesylate dihydrate, is a potent Type II DNA topoisomerase inhibitor. Gepotidacin mesylate dihydrate is a novel antibacterial drug candidate. Gepotidacin mesylate ...
T70837 Rimegepant sulfate hydrate
Rimegepant, also known as BMS-927711 and BHV-3000, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist in clinical trials for treating migraines. Rimegepant has shown ...
T11391L Gepotidacin GSK2140944 Others
Gepotidacin is a novel triazaacenaphthylene inhibitor of bacterial type II topoisomerase.
T16093 Telcagepant MK-0974 Others
Telcagepant is an orally active antagonist of calcitonin gene-related peptide (CGRP) receptor (Kis: 0.77 nM and 1.2 nM for human and rhesus CGRP receptors, respectively).
T77023 Geptanolimab
Geptanolimab (CBT-501), a humanized IgG4κ monoclonal antibody targeting PD-1 (Programmed Death-1), functions by competitively inhibiting the interaction between PD-L1/L2 and PD-1, thereby possessing potential use in canc...
T31922 Gepefrine, (+/-)-
Gepefrine, (+/-)- is a bioactive chemical.
T11391 Gepotidacin S enantiomer GSK2140944 S enantiomer Others
Gepotidacin S enantiomer is an S enantionmer of gepotidacin.
T71490 Gepotidacin hydrochloride
Gepotidacin hydrochloride, also known as GSK-2140944 hydrochloride, is a potent Type II DNA topoisomerase inhibitor. Gepotidacin hydrochloride is a novel antibacterial drug candidate. Gepotidacin hydrochloride Demonstrat...

Recombinant Proteins

Species：
Human (1)
Expression System：
HEK293 (1)
Tag：
His (1)
Cat No. Product Name Species Expression System
TMPY-00978 Progranulin Protein, Human, Recombinant (His) Human HEK293
Granulins are a family of secreted, glycosylated peptides that are cleaved from a single precursor protein with 7.5 repeats of a highly conserved 12-cysteine granulin/epithelin motif. The precursor protein, progranulin, ...
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