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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12928 | SK33 | Androgen Receptor | |
SK33 is a potent and tissue selective anti-androgen agent. SK33 reduces androgen receptor (AR) transcriptional activity. | |||
T64372 | DB722 | Others | |
DB722 is a furamidine analogues with DNA binding activity. DB722 shows antiproliferative activity. | |||
TWP2911 | Thymidine | 5-Methyldeoxyuridine,Deoxyribothymidine,DThyd,NSC 21548,Thymidin | Others , DNA/RNA Synthesis , Endogenous Metabolite |
1. Thymidine (DThyd) overload due to Thymidine phosphorylase deficiency, and mitochondrial toxicity caused by antiviral Thymidine analogues. | |||
T67792 | BTA-188 | Antiviral | |
BTA-188 is one of the most potent analogues of novel and orally active synthetic benzoxazole and benzothiazole derivatives with significant anti-rhinovirus activity. | |||
T0028 | Gamibetal | 3-Hydroxy-GABA,4-Amino-3-hydroxybutyric Acid | HIV Protease |
Gamibetal (4-Amino-3-hydroxybutyric Acid) is used as a chiral reagent in the synthesis of antiepileptic and hypotensive drug GABOB and analogues. Also used in the preparation of HIV-1 inhibitors derived from Betulinic Ac... | |||
T4735 | 2'-Deoxyuridine 5'-monophosphate disodium | 2'-dUMP⋅2Na,2'-Deoxyuridine 5'-monophosphate disodium salt | Others , Endogenous Metabolite |
2'-Deoxyuridine 5'-monophosphate disodium (2'-dUMP⋅2Na) salt is used by the enzyme thymidylate synthetase (TS) for the de novo production of dTMP. dUMP is used as the reference substrate in studies of dUMP analogues in p... | |||
T38271 | TH1217 | TH 1217 | Others |
TH1217, a potent and selective inhibitor of dCTPase pyrophosphatase 1 (dCTPase), demonstrates an IC50 value of 47 nM. It amplifies the cytotoxic impact of cytidine analogues on leukemia cells and exhibits potential again... | |||
TP2009L | K 41498 aceate | CRFR | |
K41498 acetate, an analogues of antisauvagine-30 (aSvg-30), inhibits sauvagine-stimulated cAMP accumulation in hCRF2α- and hCRF2β-expressing cells. K41498 acetate is a potent and highly selective antagonist CRF2 receptor... | |||
T1349 | 5-Fluorouridine | Others , DNA/RNA Synthesis | |
5-fluorouridine is also known as FUrd, 5-Fluorouracil 1-beta-D-ribofuranoside, 5-Fur, or 5-Fluoro-uridine. 5-fluorouridine is a solid. This compound belongs to the pyrimidine nucleosides and analogues. These are compound... | |||
T35449 | α-(difluoromethyl)-DL-Arginine | DFMA,RMI 71897,α-(difluoromethyl)-DL-Arginine | Others |
α-(difluoromethyl)-DL-Arginine (RMI 71897) is an enzyma-activated, irreversible inhibitor of arginine decarboxylase for E. coli (Ki = 800 μM), Pseudomonas aeruginosa, and Klebsiella pneumoniae. At 0.01 mM, it has been sh... | |||
T36520 | COR659 | Cannabinoid Receptor , GABA Receptor | |
COR659 is a GABAB positive allosteric modulator (PAM) . COR659 suppresses alcohol and chocolate self-administration in rats[1]. COR659 apparently exerts its effects via a composite mechanism, including positive allosteri... | |||
T19100 | 2-(Dimethylamino)acetaldehyde | Others | |
2-(Dimethylamino)acetaldehyde can be used to synthesis Muscarine analogues. | |||
T19099 | 2-(Dimethylamino)acetaldehyde hydrochloride | Others | |
2-(Dimethylamino)acetaldehyde hydrochloride can be used to synthesis Muscarine analogues. | |||
T27264 | Endochin | ||
Endochin is an experimental antimalarial. Endochin and analogues thereof are causal prophylactic and potent erythrocytic stage agents in avian models. | |||
T69565 | Hadacidin sodium | ||
Hadacidin sodium is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase. | |||
T15059 | DBCO-C6-acid | Others | |
DBCO-C6-acid is a non-cleavable linker utilized for the synthesis of antibody-drug conjugates (ADCs) and carmaphycin analogues[1]. | |||
TP1455 | Cardiotoxin Analog (CTX) IV (6-12) | Cardiotoxin Analog (CTX) IV 6-12 | |
Cardiotoxin Analog (CTX) IV (6-12) is a part peptide of Cardiotoxin Analog (CTX) IV. Cardiotoxin analogues IV isolated from the venom of Taiwan Cobra. | |||
T68868 | Hadacidin | ||
Hadacidin is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase. | |||
T26469 | A-176120 | ||
A-176120 is a potent farnesyl pyrophosphate (FPP) analogues, it selectively inhibits farnesyltransferase. It has anti-angiogenic potential and may reduce H-ras NIH3T3 tumour growth. | |||
T76575 | Arg-Trp | ||
Arg-Trp, a dipeptide consisting of arginine and tryptophan, and its analogues, specifically the octyl ester, exhibit antibacterial activity [1]. |