Powder: -20°C for 3 years | In solvent: -80°C for 1 year
K41498 acetate, an analogues of antisauvagine-30 (aSvg-30), inhibits sauvagine-stimulated cAMP accumulation in hCRF2α- and hCRF2β-expressing cells. K41498 acetate is a potent and highly selective antagonist CRF2 receptor with Ki values of 0.66 nM, 0.62 nM and 425 nM for human CRF2α, CRF2β and CRF1 receptors respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 623.00 | |
5 mg | In stock | $ 1,330.00 | |
10 mg | In stock | $ 1,780.00 | |
25 mg | In stock | $ 2,680.00 | |
50 mg | In stock | $ 3,590.00 | |
100 mg | In stock | $ 4,880.00 |
Description | K41498 acetate, an analogues of antisauvagine-30 (aSvg-30), inhibits sauvagine-stimulated cAMP accumulation in hCRF2α- and hCRF2β-expressing cells. K41498 acetate is a potent and highly selective antagonist CRF2 receptor with Ki values of 0.66 nM, 0.62 nM and 425 nM for human CRF2α, CRF2β and CRF1 receptors respectively. |
Targets&IC50 | CRF1:425 nM(Ki), CRF2β:0.62 nM(Ki), CRF2α:0.66 nM(Ki) |
Molecular Weight | N/A |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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K 41498 aceate GPCR/G Protein CRFR inhibitor inhibit