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Search Result

Search Results for "threonine proteases"

Compounds

Cat No. Product Name
T7017 WNK463 Serine/threonin kinase
WNK463 是口服有活性的 WNK 激酶抑制剂，能够抑制 WNK1 (IC50:5 nM)、WNK2 (IC50:1 nM)、WNK3 (IC50:6 nM)及 WNK4 (IC50:9 nM)。
T11666 IPR-803 Serine/threonin kinase
IPR-803 是一种有效的 uPAR·uPA 蛋白-蛋白相互作用抑制剂，具有抗肿瘤活性。 IPR-803 直接与 uPAR 结合，Ki 为 0.2 μM。
T11885 LSP-249 Others
LSP-249是血浆 kallikrein 的抑制剂，用于血管性水肿的研究，EC50值小于 100 nM。摘自专利 WO2016011209A1。
T10547 BioE-1115 Serine/threonin kinase , Casein Kinase
BioE-1115 是一种特异性和有效的丝氨酸-苏氨酸蛋白激酶抑制剂 (PASK, IC50 = 4 nM)。 BioE-1115 是一种有效的酪蛋白激酶 2α 抑制剂 (IC50 = 10 μM)。
T5456 WNK-IN-11 Allosteric WNK Kinase Inhibitor Serine/threonin kinase
Allosteric WNK Kinase Inhibitor 是(WNK)激酶的变构抑制剂，能够抑制 WNK1 (IC50:4 nM) 。
TP1277 Bradykinin 缓激肽 Bradykinin Receptor , Endogenous Metabolite
Bradykinin 是由激肽释放酶-激肽系统产生的活性肽。 它是炎症调节因子和神经调节因子，对几种血管和肾功能也有调节作用。
T4524 SBC-110736 SBC110736 Serine/threonin kinase , Others
SBC110736 是一种蛋白转化酶枯草杆菌蛋白酶 9 型 (PCSK9) 抑制剂，提取于专利 WO2014150395A1（图例1）。
T6370 AEBSF hydrochloride Pefabloc SC,AEBSF HCl Influenza Virus , Serine Protease , Thrombin
AEBSF hydrochloride 是一种丝氨酸蛋白酶的不可逆抑制剂。
TN2082 Pinostrobin Beta Amyloid , IL Receptor , Serine/threonin kinase , TNF
Pinostrobin 是一种 PCSK9抑制剂，可抑制 PCSK9 的催化活性。它是能够在多种植物中发现的黄酮类化合物，并具有抗氧化，抗炎，抗癌和神经保护作用。它是有前景的胆固醇调节和脂质管理剂。
T14358 Avoralstat BCX4161 Others
Avoralstat 是血浆激肽释放酶(PKK)抑制剂，具有口服活性，可用于遗传性血管性水肿的研究。
T4058 R-IMPP Others , Serine/threonin kinase
R-IMPP 是抗 PCSK9分泌的药物 (IC50=4.8 μM)，靶向作用于 80S 核糖体，抑制 PCSK9 蛋白的翻译。
T2626 SBC-115076 SBC115076 Serine/threonin kinase , Others
SBC115076 是前蛋白转化酶枯草杆菌蛋白酶/ kexin 9型(PCSK9)抑制剂。其中PCSK9 是一种前蛋白转化酶，在 LDL 受体代谢中的重要物质。
T8645 PF-06446846 Others
PF-06446846 是口服有活性的 PCSK9抑制剂。它能够在密码子区域附近阻断 80S ribosome，选择性地直接抑制 PCSK9 的翻译。
T9920 Evolocumab Others
Evolocumab 是人源化单克隆抗体PCSK9的抑制剂。它与循环的 PCSK9 蛋白结合，使得PCSK9与 LDLR 结合受到抑制。它可用研究于高胆固醇血症以及动脉粥样硬化性心血管疾病的研究。
T13257 Upamostat Serine/threonin kinase , Serine Protease , PAI-1
Upamostat 是一种丝氨酸蛋白酶抑制剂，也是一种具有口服活性的 WX-UK1 前药，是一种尿激酶型纤溶酶原激活剂 (uPA) 抑制剂。
T9276 SBC-115337 Others , Serine/threonin kinase
SBC-115337 是苯并呋喃化合物，也是 PCSK9抑制剂 (IC50:0.5 μM) 。
T8676 FOY 251 Others , Serine/threonin kinase , SARS-CoV
FOY 251 是一种蛋白酶抑制剂，是具有抗蛋白水解活性的 Camostate 代谢物，能抑制 SARS-CoV-2 的感染。
T8350 TPCK Proteasome
TPCK 是丝氨酸蛋白酶抑制剂，通过与 HPV-18 E7 蛋白的视网膜母细胞瘤蛋白 (RB) 结合核心发生反应，并能够消除其 RB 结合能力。将它添加到培养基内，可修饰活角质形成细胞中的 E7 蛋白。
T3359 Aprotinin Antilysin,Traskolan,Bovine Pancreatic Trypsin Inhibitor,抑肽酶,抑酶肽 Serine Protease , Proteasome , Others , Influenza Virus
Aprotinin 是分离自牛肺的一种广谱丝氨酸蛋白酶抑制剂，可抑制多种不同酯酶和蛋白酶的活性。
T8362 Benzamidine hydrochloride 苄脒盐酸盐,Benzamidine HCl Serine Protease , Serine/threonin kinase
Benzamidine HCl 是可逆的胰蛋白酶样丝氨酸蛋白酶 (trypsin-like serine proteases) 竞争性抑制剂，对 uPA、类胰蛋白酶、胰蛋白酶和 Xa 因子作用的Ki 分别为 97 µM、20 µM、21 µ...
WNK463
T7017
synonym:
Target:
IPR-803
T11666
synonym:
Target:
LSP-249
T11885
synonym:
Target:
BioE-1115
T10547
synonym:
Target:
WNK-IN-11
T5456
synonym: Allosteric WNK Kinase Inhibitor
Target:
Bradykinin
TP1277
synonym: 缓激肽
Target:
SBC-110736
T4524
synonym: SBC110736
Target:
AEBSF hydrochloride
T6370
synonym: Pefabloc SC,AEBSF HCl
Target:
Pinostrobin
TN2082
synonym:
Target:
Avoralstat
T14358
synonym: BCX4161
Target:
R-IMPP
T4058
synonym:
Target:
SBC-115076
T2626
synonym: SBC115076
Target:
PF-06446846
T8645
synonym:
Target:
Evolocumab
T9920
synonym:
Target:
Upamostat
T13257
synonym:
Target:
SBC-115337
T9276
synonym:
Target:
FOY 251
T8676
synonym:
Target:
TPCK
T8350
synonym:
Target:
Aprotinin
T3359
synonym: Antilysin,Traskolan,Bovine Pancreatic Trypsin Inhibitor,抑肽酶,抑酶肽
Target:
Benzamidine hydrochloride
T8362
synonym: 苄脒盐酸盐,Benzamidine HCl
Target:
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