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Bombesin Receptor

The bombesin receptors are a group of G-protein coupled receptors which bind bombesin.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T80148 GRP (14-27) (human, porcine, canine) 81608-29-9 98%
GRP (14-27) (human, porcine, canine)
GRP (14-27) (human, porcine, canine) functions as a ligand for bombesin receptors, with its specific binding being inhibited by GTP and GDP, while GMP does not a...
T80266 GB-6 2413262-74-3 98%
GB-6
GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), shows potential as a high-contrast imaging probe due to its...
TP1701 RC-3095 TFA 1217463-61-0 98%
RC-3095 TFA
RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity.
TP2239L [D-Phe12]-Bombesin acetate 98%
[D-Phe12]-Bombesin acetate
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.
TP1916L1 [D-Phe12,Leu14]-Bombesin acetate TP1916L1 99.14%
[D-Phe12,Leu14]-Bombesin acetate
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.
TP1281L1 Bombesin acetate(31362-50-2 free base) 1222319-87-0 98.44%
Bombesin acetate(31362-50-2 free base)
Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina). It has two known homologs in m...
T10722 CD80-IN-3 486449-65-4 98.08%
CD80-IN-3
CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).
T20604L Litorin acetate(55749-97-8 Free base) 97.64%
Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist. It stimulates the contraction of smooth muscle, stimulates gastrin, g...
TP1913L1 BA 1 acetate(183241-31-8 free base) TP1913L1 95.3%
BA 1 acetate(183241-31-8 free base)
BA 1 acetate is a potent bombesin receptor agonist (IC50 values are 0.26, 1.55 and 2.52 nM for BB1, BB2 and BB3 respectively). Enhances glucose transport in obes...
T4540 ML-18 1422269-30-4 100%
ML-18
ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.
T3S1612 Kuwanon G 75629-19-5 98%
kuwanon G
1. Kuwanon G (Moracenin B) as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective ...
T8691 PD 168368 204066-82-0 98%
PD 168368
PD 168368 is a novel, potent, competitive and selective nonpeptide neuromodulin B receptor (NMB-R) antagonist with inhibitory effects on the gastrin-releasing pe...
TN1849 Kuwanon H 76472-87-2 98%
Kuwanon H
Kuwanon H, and possibly kuwanon G also, are specific antagonists for the gastrin-releasing peptide (GRP) -preferring receptor and can be useful for studying the ...
T16449 PD176252 204067-01-6 98%
PD176252
PD176252 is a potent BB1 and BB2 antagonist with inhibitory effects on BB1 and BB2 receptors.PD176252 acts as a small molecule GRPR inhibitor and FPR1/FPR2 agoni...
T2126 MK-5046 1022152-70-0 98%
MK-5046
MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).
GRP (14-27) (human, porcine, canine)
T80148
GRP (14-27) (human, porcine, canine) functions as a ligand for bombesin receptors, with its specific binding being inhibited by GTP and GDP, while GMP does not a...
GB-6
T80266
GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), shows potential as a high-contrast imaging probe due to its...
RC-3095 TFA
TP1701
RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity.
[D-Phe12]-Bombesin acetate
TP2239L
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.
[D-Phe12,Leu14]-Bombesin acetate
TP1916L1
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.
Bombesin acetate(31362-50-2 free base)
TP1281L1
Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina). It has two known homologs in m...
CD80-IN-3
T10722
CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).
Litorin acetate(55749-97-8 Free base)
T20604L
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist. It stimulates the contraction of smooth muscle, stimulates gastrin, g...
BA 1 acetate(183241-31-8 free base)
TP1913L1
BA 1 acetate is a potent bombesin receptor agonist (IC50 values are 0.26, 1.55 and 2.52 nM for BB1, BB2 and BB3 respectively). Enhances glucose transport in obes...
ML-18
T4540
ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.
kuwanon G
T3S1612
1. Kuwanon G (Moracenin B) as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective ...
PD 168368
T8691
PD 168368 is a novel, potent, competitive and selective nonpeptide neuromodulin B receptor (NMB-R) antagonist with inhibitory effects on the gastrin-releasing pe...
Kuwanon H
TN1849
Kuwanon H, and possibly kuwanon G also, are specific antagonists for the gastrin-releasing peptide (GRP) -preferring receptor and can be useful for studying the ...
PD176252
T16449
PD176252 is a potent BB1 and BB2 antagonist with inhibitory effects on BB1 and BB2 receptors.PD176252 acts as a small molecule GRPR inhibitor and FPR1/FPR2 agoni...
MK-5046
T2126
MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).
TargetMol