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Search Result

Search Results for "infarction"

Libraries

Antioxidant Compound Library
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Compounds

Cat No. Product Name
T15108 DG-041 Prostaglandin Receptor
DG-041 是高亲和力，选择性的，有效的 EP3受体拮抗剂，在结合和 FLIPR 试验中，IC50分别为 4.6 nM 和 8.1 nM。DG-041通过抑制 PGE2促进血小板聚集。DG-041具有血脑屏障渗透性。
T2320 Indacaterol Adrenergic Receptor
Indacaterol 是一种超长效β-肾上腺素受体激动剂。
T4330 CaCCinh-A01 Chloride channel
CaCCinh-A01 是钙激活氯离子通道和TMEM16A 抑制剂，IC50值分别为 10 和 2.1 μM。
T3461 Losartan Carboxylic Acid E-3174,EXP-3174 RAAS
Losartan Carboxylic Acid 是 Losartan 的活性羧酸代谢产物，是血管紧张素Ⅱ受体 1 型(AT1)拮抗剂。它能够阻断血管紧张素 II 诱导的血管平滑肌细胞反应，可以提高血浆肾素活性，降低平均动脉压。
T67941 WAY-639921
WAY-639921对Phosphodiesterase PDE1c 具有抑制作用，可用来治疗高血压、心力衰竭、心肌梗塞、肾衰竭、哮喘、支气管炎和痴呆。
T15418 GS-6201 CVT-6883 Adenosine Receptor
GS-6201 是选择性腺苷 A2B 受体拮抗剂。它对人腺苷 A2B 受体具有高亲和力和选择性 (Ki=22 nM)。它降低了小鼠急性心肌梗死后心脏中 caspase-1 的活性，并减弱了心脏重塑。它减弱了致敏小鼠 NECA，AMP 或变应...
T3S0289 Araloside X Calcium Channel
Aralosides possess protective effect against experimental myocardial ischemia and infarction, the mechanism of myocardia...
T1479 Isosorbide dinitrate 硝酸异山梨酯,Isordil,Nitrosorbide,Sorbidnitrate,Sorbide nitrate Others , NO Synthase
Isosorbide dinitrate 是 NO 供体，可预防心肌梗死 (MI) 引起的左室重构及心功能退化。
T0407 Edaravone 依达拉奉,MCI-186 MMP , Apoptosis , Free radical scavengers
Edaravone 是一种新型自由基清除剂，能够抑制大鼠与 MMP-9有关的脑出血。
T77611 DAPK-IN-2 WAY-380496 DAPK
DAPK-IN-2 是一种 DAPK 抑制剂。 DAPK-IN-2 具有潜在的抗癌活性，可调节细胞发生自噬反应，可用于研究脑梗死和缺血性疾病。
TP2279L Obestatin (rat) acetate GHSR
Obestatin (rat) acetate 是 G 蛋白偶联受体 39 (GPR39) 的内源性配体。它具有抗炎、抗心肌梗塞和抗氧化特性。 它抑制食物摄入，抑制空肠收缩，并减少体重增加。
T0230 Prasugrel PCR 4099,LY640315,普拉格雷,CS-747 P2Y Receptor
Prasugrel 是一种噻吩吡啶和前药，是一种可口服的 P2Y12受体拮抗剂，抑制 ADP 诱导的血小板聚集，用于预防急性冠状动脉综合征患者的血栓形成、不稳定型心绞痛和心肌梗塞，以及接受经皮冠状动脉介入治疗的患者。
T0812 Propranolol hydrochloride 盐酸普萘洛尔,Propranolol HCl,NCS-91523,ICI-45520,AY-64043 Adrenergic Receptor
Propranolol hydrochloride 是非选择性的β-adrenergic receptor 拮抗剂，对 β1AR 和 β2AR 具有高亲和力。它能够抑制 [3H]-DHA 与大鼠脑膜制剂的结合。它可以用于研究高血压，嗜铬细胞...
T1239 Indacaterol maleate QAB149,马来酸茚达特罗 Adrenergic Receptor
Indacaterol maleate 是一种超长效的 β-肾上腺素受体激动剂。
T39115 ABR-238901 TLR
ABR-238901是一种可口服的、有作用的 S100A8/A9阻滞剂，对 S100A8/A9与其受体 RAGE(晚期糖基化终产物受体)和TLR4 (toll 样受体4)的相互作用具有抑制作用。ABR-238901具有作为治疗心肌梗死(MI...
T22323 Enoxaparin sodium Thrombin
Enoxaparin sodium 是一种低分子量肝素 (LMWH)，最近已获得美国 FDA 批准，可用于医疗管理的 ST 段心肌梗死 (STEMI) 或 STEMI 及随后的经皮冠状动脉介入治疗 (PCI) 患者。它与抗凝血酶结合并增强其...
T24873 TGX-115 TGX 115 PI3K
TGX-115是一种细胞渗透性和有效的PI 3-K 异构体p110β/p110δ抑制剂(对p110β IC50值为 0.13 μM, 对p110δ值为0.63 μM），是一种调节血小板粘附过程的酶，可抑制磷酸肌苷（PI）3-激酶，可用来治疗...
T0815L Warfarin sodium
Warfarin sodium 是一种抗凝血剂，通过抑制维生素 K 依赖性凝血因子的合成起作用。华法林适用于预防和/或治疗静脉血栓形成及其延伸、肺栓塞和房颤栓塞。它还用作预防心肌梗塞后全身性栓塞的辅助剂。华法林也用作杀鼠剂。
T36569 KR-32568 Sodium Channel
KR-32568是一种钠/氢交换器1（NHE-1）抑制剂（IC50：230 nM）。KR-32568具有强大的心脏保护作用。当使用浓度为10μM 时，它能在离体的缺血大鼠心脏模型中恢复心脏收缩功能。KR-32568（0.3mg/kg）在缺血...
T5329 Trandolapril Angiotensin-converting Enzyme (ACE)
Trandolapril 是 Trandolaprilat 的前体药物。Trandolapril 是一种口服血管紧张素转换酶抑制剂，在高血压和充血性心力衰竭及心肌梗死领域有研究价值。
DG-041
T15108
synonym:
Target:
Indacaterol
T2320
synonym:
Target:
CaCCinh-A01
T4330
synonym:
Target:
Losartan Carboxylic Acid
T3461
synonym: E-3174,EXP-3174
Target:
WAY-639921
T67941
synonym:
Target:
GS-6201
T15418
synonym: CVT-6883
Target:
Araloside X
T3S0289
synonym:
Target:
Isosorbide dinitrate
T1479
synonym: 硝酸异山梨酯,Isordil,Nitrosorbide,Sorbidnitrate,Sorbide nitrate
Target:
Edaravone
T0407
synonym: 依达拉奉,MCI-186
Target:
DAPK-IN-2
T77611
synonym: WAY-380496
Target:
Obestatin (rat) acetate
TP2279L
synonym:
Target:
Prasugrel
T0230
synonym: PCR 4099,LY640315,普拉格雷,CS-747
Target:
Propranolol hydrochloride
T0812
synonym: 盐酸普萘洛尔,Propranolol HCl,NCS-91523,ICI-45520,AY-64043
Target:
Indacaterol maleate
T1239
synonym: QAB149,马来酸茚达特罗
Target:
ABR-238901
T39115
synonym:
Target:
Enoxaparin sodium
T22323
synonym:
Target:
TGX-115
T24873
synonym: TGX 115
Target:
Warfarin sodium
T0815L
synonym:
Target:
KR-32568
T36569
synonym:
Target:
Trandolapril
T5329
synonym:
Target:
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