Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
Applied FilterClear all
TargetMol | Tags By Target
  • Glucocorticoid Receptor
    (2)
  • Others
    (3)
Filter
Search Result
Results for "

glucocorticoid receptor modulator 1

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    6
    TargetMol | Inhibitors_Agonists
  • Natural Products
    1
    TargetMol | Natural_Products
Glucocorticoid receptor modulator 1
T721022868357-11-1
Glucocorticoid receptor modulator 1 is a potent, orally active, non-steroidal selective glucocorticoid receptor modulator, exhibiting IC50 values of 9 nM and 130 nM against NF-κB and AP-1, respectively. It effectively reduces the expression of inflammatory factors such as IL-6, IL-1β, and TNF-α, and alleviates dermatitis in mice.
  • Inquiry Price
6-8 weeks
Size
QTY
EX-A5386
Glucocorticoid receptor modulator-1
T677422452396-89-1
EX-A5386 (Glucocorticoid receptor modulator-1) is a potent glucocorticoid receptor modulator, IC50 EC50<100nM.
  • Inquiry Price
Size
QTY
Dazucorilant
CORT113176
T389831496508-34-9
Dazucorilant (CORT113176) is a non-steroidal glucocorticoid receptor (GR) modulator characterized by its high affinity and selectivity. With an impressive K i value of <1 nM in vitro, Dazucorilant proves to be an exceptional compound for investigating neurological disorders.
  • Inquiry Price
10-14 weeks
Size
QTY
pparγ/gr modulator 1
T75009
PPARγ GR Modulator 1, an orally active dual agonist for the Peroxisome Proliferator-Activated Receptor Gamma (PPARγ) and Glucocorticoid Receptor (GR), exhibits Ki values of 3.3 and 33.6 μM, respectively. This compound is utilized in metabolic disease research, including diabetes [1].
  • Inquiry Price
Size
QTY
HP210
T78073728039-52-9
HP210, a selective glucocorticoid receptor modulator (SGRM), can suppress IL-1β and IL-6 mRNA expression, suggesting its utility in investigating inflammation-related diseases [1].
  • Inquiry Price
8-10 weeks
Size
QTY
2-O-trans-p-Coumaroylalphitolic acid
TN760067911-63-1
2-O-trans-p-Coumaroylalphitolic acid (Zj7), a triterpene sourced from jujube plants, functions as a selective modulator of the glucocorticoid receptor (GR). This compound holds potential for use in obesity research [1].
  • Inquiry Price
Inquiry
Size
QTY