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Search Results for "dynamin"

Targets

Compounds

Cat No. Product Name
T21798L Dynamin inhibitory peptide Acetate Dynamin inhibitory peptide Acetate(251634-21-6 Free base) GTPase
Dynamin inhibitory peptide Acetate 是一种具有序列 Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro 的肽,可抑制 GTPase dynamin
T64369 Dynamin IN-2 Dynamin
Dynamin IN-2是一种Wiskostatin 类似物。Dynamin IN-2有效抑制 dynamin ,对 dynamin I GTPase 的 IC50 为 1.0 μM。Dynamin IN-2 可阻断网格蛋白介导的内吞作用 ...
TP1907L1 Dynamin inhibitory peptide, myristoylated acetate Dynamin inhibitory peptide, myristoylated acetate(251634-22-7 free base) Dynamin
Dynamin inhibitory peptide, myristoylated acetate(251634-22-7 free base) 是一种 DynaMin 抑制剂,可干扰两性霉素与 dynamin 的结合。 DynaMin 抑...
T1848 Dynasore Dynamin Inhibitor I HSV , Dynamin , Virus Protease , Autophagy
Dynasore 是一种可渗透细胞的化学物质,可逆且非竞争性地抑制 dynamin 1/2 的 GTPase 活性。 它还抑制线粒体动力蛋白 Drp1,对其他小 GTPase 没有影响。
T72952 Dynamin IN-1
DynaminIN-1 是一种有效的dynamin 抑制剂,IC50值为 1.0 µM。
T75796 Dynamin inhibitory peptide TFA
Dynamininhibitory peptide TFA 竞争性地阻止了动力蛋白 (dynamin) 与两性纤维蛋白的结合,从而防止了内吞作用。Dynamininhibitory peptide TFA 阻断多巴胺 D3对 GABAA 受...
TP1907 DynaMin inhibitory peptide, myristoylated
Cell-permeable version of dynamin inhibitory peptide, an inhibitor of the GTPase dynamin that competitively blocks bindi...
TP2039 Dynamin inhibitory peptide, myristoylated (control)
Control peptide version of dynamin inhibitory peptide, myristoylated, an inhibitor of the GTPase dynamin that competitiv...
T6822 Hydroxy-Dynasore Dyngo-4a Dynamin
Hydroxy-Dynasore 是 Dynasore 结构模拟类似物,是一种改进的,低细胞毒性的 dynamin 通用抑制剂,抑制 dynamin 依赖性转铁蛋白的内吞作用的 IC50为 5.7 μM,对大脑重组 dynamin I 和重...
T1907 Mdivi-1 Mitochondrial division inhibitor 1 Autophagy , Dynamin , Mitophagy , Apoptosis
Mdivi-1 是选择性的发动蛋白相关蛋白 1 (Drp1) 抑制剂。Mdivi-1 是一种有效的线粒体分裂/线粒体自噬抑制剂。
T22445 Trimethyloctadecylammonium bromide Dynamin
Trimethyloctadecylammonium bromide 是 Dynamin I 的抑制剂 (IC50 : 1.9 μM),也抑制 Dynamin Ⅱ。
T3898 Schaftoside 夏佛塔苷,Shaftoside,APIGENIN-6-GLUCOSIDE-8-ARABINOSIDE Antioxidant , TLR , MyD88 , Autophagy , Dynamin , Mitochondrial Metabolism
Schaftoside 是在多种中草药中发现的一种黄酮类天然产物。它抑制 TLR4 和 Myd88 表达,还降低 Drp1 表达和磷酸化,并减少线粒体分裂,具有抗氧化和抗癌活性。
T30479 Bis-T-23 AG1717 HIV Protease
Bis-T-23是一种肌动蛋白依赖性达纳敏低聚物的促进剂,是一种 HIV-I 整合酶抑制剂,是泰尔普斯丁衍生物。Bis-T-23可以促进肌动蛋白依赖性的dynamin 寡聚化。Bis-T-23可用于HIV 和慢性肾脏疾病(CKD)的研究。
T22981 Tetradecyltrimethylammonium bromide Cetrimide,MitMAB,tetradecyl trimethyl ammonium bromide,十四烷基三甲基溴化铵 Dynamin
MitMAB 是一种具有不对称结构的阳离子表面活性剂,是一种有机结构单元。
TP1947L P110 TFA Others
P110 TFA 是一种 dynamin-related protein 1 (Drp1) 抑制剂,抑制 Drp1 GTPase 活性。
T35548 Dynapyrazole A Dynamin
Dynapyrazole A 是微管动力蛋白的特异性抑制剂,对动力蛋白 1 和动力蛋白 2 依赖性微管滑动的 IC50 分别为 2.3 和 2.6 μM。 Dynapyrazole A 抑制 Hedgehog 信号传导,IC50 为 1.9...
T22754 Dynole 34-2 Others
Dynamin I inhibitor
T38407 RTIL 13
RTIL 13 is a highly effective inhibitor of dynamin GTPase, exhibiting an IC50 value of 2.3 μM for dynamin I GTPase. Furt...
T37023 MB 0223
Dynamin-related GTPase DRP1 partial inhibitor (IC50 = 1.2 μM). Selective for DRP1 over other dynamin-related GTPases, OP...
TP1947 P110
Dynamin-related protein 1 (Drp1) inhibitor, inhibits Drp1 GTPase activity. Displays no effect on dynamin 1 or other mito...
Dynamin inhibitory peptide Acetate
T21798L
synonym: Dynamin inhibitory peptide Acetate(251634-21-6 Free base)
Target:
Dynamin IN-2
T64369
synonym:
Target:
Dynamin inhibitory peptide, myristoylated acetate
TP1907L1
synonym: Dynamin inhibitory peptide, myristoylated acetate(251634-22-7 free base)
Target:
Dynasore
T1848
synonym: Dynamin Inhibitor I
Target:
Dynamin IN-1
T72952
synonym:
Target:
Dynamin inhibitory peptide TFA
T75796
synonym:
Target:
DynaMin inhibitory peptide, myristoylated
TP1907
synonym:
Target:
Dynamin inhibitory peptide, myristoylated (control)
TP2039
synonym:
Target:
Hydroxy-Dynasore
T6822
synonym: Dyngo-4a
Target:
Mdivi-1
T1907
synonym: Mitochondrial division inhibitor 1
Target:
Trimethyloctadecylammonium bromide
T22445
synonym:
Target:
Schaftoside
T3898
synonym: 夏佛塔苷,Shaftoside,APIGENIN-6-GLUCOSIDE-8-ARABINOSIDE
Target:
Bis-T-23
T30479
synonym: AG1717
Target:
Tetradecyltrimethylammonium bromide
T22981
synonym: Cetrimide,MitMAB,tetradecyl trimethyl ammonium bromide,十四烷基三甲基溴化铵
Target:
P110 TFA
TP1947L
synonym:
Target:
Dynapyrazole A
T35548
synonym:
Target:
Dynole 34-2
T22754
synonym:
Target:
RTIL 13
T38407
synonym:
Target:
MB 0223
T37023
synonym:
Target:
P110
TP1947
synonym:
Target:
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