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Compounds

Cat No. Product Name
T5996 CB1-IN-1 DBPR211,1-(2,4-二氯苯基)-N-1-哌啶基-4-[[(1-吡咯烷基磺酰基)氨基]甲基]-5-[5-[2-[4-(三氟甲基)苯基]乙炔基]-2-噻吩基]-1H-吡唑-3-甲酰胺 Cannabinoid Receptor
CB1-IN-1 是新型的外周大麻素-1受体 (CB1R) 拮抗剂,作用于CB1R (EC50 = 3 nM) 和 CB2R 的Ki 分别为0.3 nM 和 21 nM。
T14881 CB1 antagonist 2 AM4113 Cannabinoid Receptor
CB1 antagonist 2 是一种 caimabinoid 1 拮抗剂,在体内抑制 CB1 的IC50值为 25.5 nM。摘自 WO2016184310A1 中获得,化合物 3。
T28468 PSNCBAM-1 PSNCBAM 1 Cannabinoid Receptor
PSNCBAM-1 是一种 CB1 受体负变构调节剂 (EC50 = 0.1 μM),在体内具有吞噬作用。 PSNCBAM-1 可用于肥胖研究。
TN5131 Tetrahydrocannabivarin delta9-Tetrahydrocannabivarin,THCV,Tetrahydrocannavarin,CRM Cannabinoid Receptor
Tetrahydrocannabivarin 是 cannabinoid type 1 receptor 的中性拮抗剂,对 2 型糖尿病有潜在治疗价值。
T36520 COR659 Cannabinoid Receptor , GABA Receptor
COR659 是一种有效的 GABAB 的阳性变构调节剂。COR659具有缓解大鼠对酒精和巧克力成瘾的作用。
T9466 RTICBM-189 Others
RTICBM-189 是可透过血脑屏障的大麻素 1 型受体变构调节剂,在 Ca2+动员试验中pIC50为 7.54,对 hCB1和 mCB1的 pIC50分别为 5.29 和 6.25。
T8425 Linoleoyl Ethanolamide TRP/TRPV Channel
Linoleoyl ethanolamide 是脂肪酸乙醇酰胺。它可弱结合 CB1CB2 受体,并分别抑制[3H]CP-55,940的结合,Ki 分别为 10 和 25μM。它在引起小鼠过氧化氢酶方面的效力是 anandamide 的...
T10510 CB1 antagonist 1 Cannabinoid Receptor
CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and metabolic syndrome, neuroinflammatory...
T61849 AM8936
AM8936 is a well-balanced and highly potent agonist for the cannabinoid receptor type-1 (CB1) in functional assays, with...
T62180 CB1/2 agonist 2
CB1/2 agonist 2 (compound 23) 是一种有效的非选择性大麻素 (cannabinoid) 配体,其Ki 分别为 3.5 nM 和 1.2 nM。CB1/2 agonist 2 是一种 CB1 的完全激动剂,也是 C...
T61609 CB1-IN-2
CB1-IN-2 (Compound 4g) is a potent and selective inhibitor of the CB1 receptor, exhibiting an IC50 value of 0.644 μM. Th...
T38204 GAT229
GAT229 is a positive allosteric modulator of cannabinoid receptor 1 (CB1) and the S-(-) enantiomer of the CB1 modulator ...
T72395 CB1 inverse agonist 2
CB1inverse agonist 2 是一种口服有效的大麻素受体 CB1反向激动剂。CB1inverse agonist 2 在小鼠模型中,能有效抑制 CP55940 导致的体温失温和厌食情况。
T69740 AMG-315
AMG-315 is a Potent Endocannabinoid Ligand with Stability to Metabolizing Enzymes. AMG-315 is a chiral arachidonoyl eth...
T38138 Arachidonoyl 2'-Chloroethylamide Arachidonoyl 2'-Chloroethylamide,2'-chloro-AEA,ACEA
Arachidonoyl 2-chloroethylamide (ACEA) is a potent and selective cannabinoid (CB) receptor 1 agonist with Ki values of 1...
T38049 Glycerophospho-N-Palmitoyl Ethanolamine
N-Acylated ethanolamines (NAE) are naturally-occurring lipids that have diverse bioactivities. For example, arachidonoyl...
T21811 LH 21
LH-21 是一种有效的体内中性大麻素 CB1受体拮抗剂。LH-21 会导致剂量依赖性进食抑制,减少肥胖 Zucker 大鼠的食物摄入和体重增加。
T22146 S-1 Methanandamide
S-1 Methanandamide ((S)-Methanandamide) 是 Anandamide 的类似物,是一种 CB1受体配体,Ki 值为 173 nM。S-1 Methanandamide 抑制小鼠输精管中电诱发的抽搐反应,I...
T75798 Hemopressin(rat) TFA
Hemopressin(rat) TFA 是一种源自血红蛋白 α1 链的九肽,最初是从大鼠脑匀浆中分离出来的。Hemopressin(rat) TFA 是口服有效的,选择性的CB1大麻素受体的反向激动剂。Hemopressin(rat) T...
T11834 Leelamine hydrochloride Others
Leelamine hydrochloride suppresses transcriptional activity of androgen receptor, which is known to regulate fatty acid ...
CB1-IN-1
T5996
synonym: DBPR211,1-(2,4-二氯苯基)-N-1-哌啶基-4-[[(1-吡咯烷基磺酰基)氨基]甲基]-5-[5-[2-[4-(三氟甲基)苯基]乙炔基]-2-噻吩基]-1H-吡唑-3-甲酰胺
Target:
CB1 antagonist 2
T14881
synonym: AM4113
Target:
PSNCBAM-1
T28468
synonym: PSNCBAM 1
Target:
Tetrahydrocannabivarin
TN5131
synonym: delta9-Tetrahydrocannabivarin,THCV,Tetrahydrocannavarin,CRM
Target:
COR659
T36520
synonym:
Target:
RTICBM-189
T9466
synonym:
Target:
Linoleoyl Ethanolamide
T8425
synonym:
Target:
CB1 antagonist 1
T10510
synonym:
Target:
AM8936
T61849
synonym:
Target:
CB1/2 agonist 2
T62180
synonym:
Target:
CB1-IN-2
T61609
synonym:
Target:
GAT229
T38204
synonym:
Target:
CB1 inverse agonist 2
T72395
synonym:
Target:
AMG-315
T69740
synonym:
Target:
Arachidonoyl 2'-Chloroethylamide
T38138
synonym: Arachidonoyl 2'-Chloroethylamide,2'-chloro-AEA,ACEA
Target:
Glycerophospho-N-Palmitoyl Ethanolamine
T38049
synonym:
Target:
LH 21
T21811
synonym:
Target:
S-1 Methanandamide
T22146
synonym:
Target:
Hemopressin(rat) TFA
T75798
synonym:
Target:
Leelamine hydrochloride
T11834
synonym:
Target:
1 2