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GPCR/G Protein GHSR

GHSR

Growth hormone secretagogue receptor(GHS-R), also known as ghrelin receptor, is a G protein-coupled receptor that binds growth hormone secretagogues (GHSs), such as ghrelin, the "hunger hormone". The role of GHS-R is thought to be in regulating energy homeostasis and body weight. In the brain, they are most highly expressed in the hypothalamus, specifically the ventromedial nucleus and arcuate nucleus. GSH-Rs are also expressed in other areas of the brain, including the ventral tegmental area, hippocampus, and substantia nigra. Outside the central nervous system, too, GSH-Rs are also found in the liver, in skeletal muscle, and even in the heart.
Cat No. product name
T10319 Anamorelin Anamorelin is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
T11719 JMV 2959 hydrochloride (925238-89-7 free base) JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
T4648 TC-G-1008 TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).
T5025 Pralmorelin Pralmorelin is an oral active synthetic peptide analogue of MEK. Pralmorelin is an auxin releasing peptide/growth hormone secretory receptor agonist, can selec...
T5025L Pralmorelin acetate 158861-67-7(free base) Pralmorelin acetate stimulates growth hormone secretion.Pralmorelin acetate is an oral active synthetic peptide analogue of MEK. Pralmorelin acetate, an auxi...
T7112 Ibutamoren Mesylate Ibutamoren Mesylate is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
T7225 AnaMorelin hydrochloride Anamorelin hydrochloride is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
T7325 GHRP-6 acetate GHRP-6 acetate is a synthetic growth hormone (GH) secretagogue and an agonist of the GH secretagogue receptor (GHS-R), which is also known as the ghrelin recept...
T7398 ONC212 ONC212, a fluorinated-ONC201 analogue, is a selective agonist of GPR132.
TP2328L CJC-1295 acetate(863288-34-0 free base) CJC-1295 acetate is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releasing factor (GRF)) and a growth hormone s...
TP2328L CJC-1295 acetate(863288-34-0 free base) CJC-1295 acetate is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releasing factor (GRF)) and a growth hormone s...
TQ0022 Capromorelin Tartrate Capromorelin Tartrate is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).
Anamorelin
T10319CAS 249921-19-5
Anamorelin is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
JMV 2959 hydrochloride (925238-89-7 free base)
T11719CAS T11719
JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
TC-G-1008
T4648CAS 1621175-65-2
TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).
Pralmorelin
T5025CAS 158861-67-7
Pralmorelin is an oral active synthetic peptide analogue of MEK. Pralmorelin is an auxin releasing peptide/growth hormone secretory receptor agonist, can selec...
Pralmorelin acetate 158861-67-7(free base)
T5025LCAS T5025L
Pralmorelin acetate stimulates growth hormone secretion.Pralmorelin acetate is an oral active synthetic peptide analogue of MEK. Pralmorelin acetate, an auxi...
Ibutamoren Mesylate
T7112CAS 159752-10-0
Ibutamoren Mesylate is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
AnaMorelin hydrochloride
T7225CAS 861998-00-7
Anamorelin hydrochloride is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
GHRP-6 acetate
T7325CAS 145177-42-0
GHRP-6 acetate is a synthetic growth hormone (GH) secretagogue and an agonist of the GH secretagogue receptor (GHS-R), which is also known as the ghrelin recept...
ONC212
T7398CAS 1807861-48-8
ONC212, a fluorinated-ONC201 analogue, is a selective agonist of GPR132.
CJC-1295 acetate(863288-34-0 free base)
TP2328LCAS TP2328L
CJC-1295 acetate is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releasing factor (GRF)) and a growth hormone s...
CJC-1295 acetate(863288-34-0 free base)
TP2328LCAS TP2328L
CJC-1295 acetate is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releasing factor (GRF)) and a growth hormone s...
Capromorelin Tartrate
TQ0022CAS 193273-69-7
Capromorelin Tartrate is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).