T11798 |
L-692429
|
145455-23-8
|
99.9%
|
|
L-692429 (MK-0751) is a potent nonpeptidyl growth hormone secretagogue (GHS) agonist, a benzolactam derivative, which reverses the inhibition of GH secretion by ...
|
T80006 |
Emoghrelin
|
928262-58-2
|
98%
|
|
Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1].
|
T11560 |
HGPR91 antagonist 1
|
1314796-00-3
|
99.85%
|
|
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
|
T34281 |
Relamorelin
|
661472-41-9
|
99.85%
|
|
Relamorelin (RM-131), a selective and potent growth hormone-releasing peptide/growth hormone secretagogue receptor (GHSR) agonist, is a potent growth hormone-rel...
|
T16508 |
PF-5190457
|
1334782-79-4
|
99.34%
|
|
PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).
|
T23543 |
YIL 781
|
875258-85-8
|
99.3%
|
|
YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 μM). YIL 781 improves glucose hom...
|
TP1155L |
Human growth hormone-releasing factor acetate
|
|
99.26%
|
|
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on c...
|
T7225 |
AnaMorelin hydrochloride
|
861998-00-7
|
99.18%
|
|
AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
|
TP2279L |
Obestatin (rat) acetate
|
|
99.05%
|
|
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39). Obestatin (rat) acetate has anti-inflammatory, anti-myocardial infarcti...
|
TP2236L |
Cortistatin-8 acetate
|
TP2236L
|
99.01%
|
|
Cortistatin-8 acetate is a corticosteroid analog, a GHS-R antagonist with inhibitory effects on the growth hormone pro-secretin receptor.Cortistatin-8 acetate is...
|
T4648 |
TC-G-1008
|
1621175-65-2
|
99%
|
|
TC-G-1008 (GPR39-C3) is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat and human receptors respectively).
|
TQ0022 |
Capromorelin Tartrate
|
193273-69-7
|
98.98%
|
|
Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).
|
T11719 |
JMV 2959 hydrochloride (925238-89-7 free base)
|
2448414-54-6
|
98.09%
|
|
JMV 2959 hydrochloride (925238-89-7 free base) is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
|
TP2328L |
CJC-1295 acetate(863288-34-0 free base)
|
TP2328L
|
98%
|
|
CJC-1295 acetate(863288-34-0 free base) (DAC:GRF acetate) is a synthetic analogue of growth hormone-releasing hormone (GHRH) (also known as growth hormone-releas...
|
T7112 |
Ibutamoren Mesylate
|
159752-10-0
|
98%
|
|
Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
|
T12216L |
NF-56-EJ40 hydrochloride
|
2728500-80-7
|
97.02%
|
|
NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almo...
|
T17103 |
TM-N1324
|
1144477-35-9
|
90.39%
|
|
TM-N1324 is a GPR39 agonist. TM-N1324 activates human GPR39 with high efficacy and potencies of 280 nM and 9 nM in the absence and presence of Zn2+, respectively...
|
T10319 |
Anamorelin
|
249921-19-5
|
98%
|
|
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
|