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Compounds

Cat No. Product Name
T8630 Baclofen hydrochloride 4-amino-3-(4-chlorophenyl)butanoic acid hydron chloride GABA Receptor
Baclofen hydrochloride 是一种 GAMMA-AMINOBUTYRIC ACID 衍生物,是一种特异性 GABA-B 受体激动剂。它用于治疗肌肉痉挛,尤其是由于脊髓损伤引起的肌肉痉挛。其治疗效果来自于脊髓和脊髓上部位的作...
T6355 (R)-baclofen STX209,(R)-巴氯芬,Arbaclofen GABA Receptor
(R)-Baclofen 是一种选择性GABAB 受体激动剂。
T11986L Mebeverine acid hydrochloride
Mebeverine acid hydrochloride 是一种有效的、可口服的、可直接作用于胃肠道平滑肌解除痉挛症状的化合物。
T8452 Dantrolene Others
Dantrolene 是一种肌肉松弛剂,是人红细胞谷胱甘肽还原酶的非竞争性抑制剂,其Ki 和IC50值分别为 111.6 μM 和 52.3 μM。它是兰尼碱受体拮抗剂及Ca2+信号稳定剂。它可用于研究恶性高热、亨廷顿病、肌肉痉挛和其他神经...
T72023 JB002 Myosin
JB002 是一种肌球蛋白 II 抑制剂,IC50值 ≤10 μM。JB002 可用于肌肉痉挛、慢性肌肉骨骼疼痛、肥厚型心肌病的研究。
T0077 Dantrolene sodium 丹曲林钠,Lapatinib ditosylate monohydrate,Dantrolene sodium salt Others , Calcium Channel
Dantrolene sodium salt 是一种骨骼肌松弛药,是一种钙通道蛋白抑制剂,可抑制钙离子从肌浆释放。
T5295 1-Hydroxyoctadecane Octadecanol,1-Octadecanol,Stearyl alcohol,硬脂醇 Endogenous Metabolite , Others
1-Octadecanol 是内源性代谢产物的一种。
T1308 Orphenadrine hydrochloride Mephenamin,盐酸邻甲苯海拉明,Mebedrol Sodium Channel , NMDAR , Norepinephrine , iGluR , Histamine Receptor
Orphenadrine hydrochloride 是一种非竞争性的NMDA 受体拮抗剂, Ki=6.0 ± 0.7 μM。
T1065 Baclofen Lioresal,巴氯芬 GABA Receptor
Baclofen 是 γ-氨基丁酸 (GABA) 的亲脂性衍生物,是可口服的选择性代谢型 GABA-B 受体激动剂,具有高血脑屏障渗透率,用于治疗因脊髓损伤和多发性硬化引起的痉挛。
T6618 Orphenadrine Citrate 枸酸芬那君,奥芬那君,Flexoject,Flexon,Banflex iGluR , AChR
Orphenadrine Citrate 是NMDA 受体拮抗剂,Ki 为6.0μM,还是HERG 钾离子通道阻断剂。它是一种骨骼肌松弛剂,它作用于中枢神经系统以产生肌肉松弛作用。
T1092 Zolmitriptan 311C90,BW-311C90,佐米曲普坦 5-HT Receptor
Zolmitriptan 是一种5-HT1B/1D 受体部分激动剂,可用于偏头痛的研究,对 5-HT1B、5-HT1D、5-HT1F 受体的Ki 分别为 5.01、0.63 和 63.09 nM。
T67952 JB062 Myosin
JB062 是一种非肌肉肌球蛋白 (nonmusclemyosin) 抑制剂,对骨骼肌肌球蛋白、心肌肌球蛋白和平滑肌肌球蛋白 II 的IC50值分别为分别为 1.6、5.4 和 >100 μM。JB062 对人类癌细胞具有细胞毒性,但对正常...
T28657 SAD-448
SAD-448 is a cannabinoid receptor type 1 (CB1) agonist. SAD-448 controls spasticity via action on the peripheral nerve C...
T21077 Tolperisone free base Menopatol,Atmosgen free base,Mideton,Mydocalm,Mydeton,Besnoline free base
Tolperisone free base, a centrally acting muscle relaxant, has been used for the symptomatic treatment of spasticity and...
T29117 VSN-16 VSN16R,VSN 16R,VSN-16R
VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.
T17306 (R)-Baclofen hydrochloride Arbaclofen hydrochloride,(R)-巴氯芬盐酸盐 GABA Receptor
Arbaclofen hydrochloride, a Gamma-Aminobutyric Acid derivative, is a specific agonist of GABA-B receptors, it is used to...
T73439 MPH-220
MPH-220 是一种选择性的、具有口服活性的骨骼肌myosin-2抑制剂。MPH-220 可使肌肉放松。MPH-220 是一种抗痉挛剂,可用于痉挛和肌肉僵硬的研究。
TMPY-03282 FUCA1 Protein, Human, Recombinant (His Tag)
FUCA1 is a lysosomal enzyme involved in the degradation of fucose-containing glycoproteins and glycolipids. Mutations in...
TMPY-01876 HSP60 Protein, Human, Recombinant (His & GST Tag)
HSPD1, also known as HSP60, is a member of the chaperonin family. HSPD1 may function as a signaling molecule in the inna...
TMPY-01057 SPG21 Protein, Human, Recombinant (GST Tag)
Spastic paraplegia 21 (SPG21), also known as acid Cluster Protein 33 (ACP33) and Mast syndrome protein, is a member of t...
Baclofen hydrochloride
T8630
synonym: 4-amino-3-(4-chlorophenyl)butanoic acid hydron chloride
Target:
(R)-baclofen
T6355
synonym: STX209,(R)-巴氯芬,Arbaclofen
Target:
Mebeverine acid hydrochloride
T11986L
synonym:
Target:
Dantrolene
T8452
synonym:
Target:
JB002
T72023
synonym:
Target:
Dantrolene sodium
T0077
synonym: 丹曲林钠,Lapatinib ditosylate monohydrate,Dantrolene sodium salt
Target:
1-Hydroxyoctadecane
T5295
synonym: Octadecanol,1-Octadecanol,Stearyl alcohol,硬脂醇
Target:
Orphenadrine hydrochloride
T1308
synonym: Mephenamin,盐酸邻甲苯海拉明,Mebedrol
Target:
Baclofen
T1065
synonym: Lioresal,巴氯芬
Target:
Orphenadrine Citrate
T6618
synonym: 枸酸芬那君,奥芬那君,Flexoject,Flexon,Banflex
Target:
Zolmitriptan
T1092
synonym: 311C90,BW-311C90,佐米曲普坦
Target:
JB062
T67952
synonym:
Target:
SAD-448
T28657
synonym:
Target:
Tolperisone free base
T21077
synonym: Menopatol,Atmosgen free base,Mideton,Mydocalm,Mydeton,Besnoline free base
Target:
VSN-16
T29117
synonym: VSN16R,VSN 16R,VSN-16R
Target:
(R)-Baclofen hydrochloride
T17306
synonym: Arbaclofen hydrochloride,(R)-巴氯芬盐酸盐
Target:
MPH-220
T73439
synonym:
Target:
FUCA1 Protein, Human, Recombinant (His Tag)
TMPY-03282
synonym:
Target:
HSP60 Protein, Human, Recombinant (His & GST Tag)
TMPY-01876
synonym:
Target:
SPG21 Protein, Human, Recombinant (GST Tag)
TMPY-01057
synonym:
Target:
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