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Results for "

dopamine uptake

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    33
    TargetMol | Inhibitors_Agonists
  • Dye Reagents
    1
    TargetMol | Dye_Reagents
  • Recombinant Protein
    1
    TargetMol | Recombinant_Protein
Roxindole
EMD 49980
T26126112192-04-8In house
Roxindole (EMD 49980) is a selective dopamine autoreceptor and 5-HT1A dual agonist and inhibitor of 5-hydroxytryptamine (5-HT) uptake with antipsychotic and antidepressant activity.Roxindole can be used to study Parkinson's and neurodivergence.
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6-8 weeks
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AHN 1-055 hydrochloride
3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride
T39429202646-03-5In house
AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).
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Fezolamine
T6807080410-36-2In house
Fezolamine is a novel orally available non-tricyclic compound with antidepressant activity. It is three to two times more selective in blocking synaptosomal uptake of [3H]norepinephrine than uptake of [4H]3-hydroxytryptamine or [3H]dopamine in vitro. It blocked the inhibitory effects of rifampicin and tetraphenyl in classical behavioral tests using monoamine-depleted animals.
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Ziprasidone hydrochloride
Ziprasidone HCl, CP-88059 hydrochloride
T0031L122883-93-6
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
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Oxolinic acid
Emyrenil, Nidantin, NSC 110364, Dioxacin, Urinox
T123314698-29-4
Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY TRACT INFECTIONS.
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Benztropine mesylate
Benzotropine mesylate, Benzatropine mesylate, Benztropine methanesulfonate
T1336132-17-2
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON DISEASE. Benztropine also inhibits the uptake of dopamine.
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Amoxapine
CL-67772
T156814028-44-5
Amoxapine (CL-67772) exerts its antidepressant effect by inhibiting the re-uptake of norepinephrine and, to a lesser degree, of serotonin, at adrenergic nerve endings and blocks the response of dopamine receptors to dopamine. Amoxapine is a tricyclic antidepressant of the dibenzoxazepine class. This drug is used to treat symptoms of depression and may cause tardive dyskinesia. Amoxapine also binds to alpha-adrenergic, histaminergic, and cholinergic receptors which accounts for many of the side effects seen with this agent.
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Vanoxerine dihydrochloride
GBR-12909 dihydrochloride, I893 dihydrochloride
T715367469-78-7
Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor of dopamine uptake (IC50: 1-51 nM).
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3-CPMT
Chlortropbenzyl hydrochloride, 3-[(4-chlorophenyl)-phenylmethoxy]-8-methyl-8-azabicyclo[3.2.1]octane hydrochloride, SL6057, Wy 2149, FC-1
T2250814008-79-8
3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.
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TargetMol | Inhibitor Sale
GBR 12783
T1137167469-57-2
GBR 12783 can improve memory performance and increase hippocampal acetylcholine release in rats. GBR 12783 is a specific, potent and selective dopamine uptake inhibitor that inhibits the [3H]dopamine uptake by rat and mice striatal synaptosomes with IC50s of 1.8 nM and 1.2 nM, respectively.
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1-2 weeks
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GBR 12783 dihydrochloride
GBR12783 2HCl
T1933767469-75-4
GBR 12783 dihydrochloride (GBR12783 2HCl) is a specific, potent and selective dopamine uptake inhibitor. GBR 12783 dihydrochloride inhibits the [3H]dopamine uptake by rat and mice striatal synaptosomes with IC50s of 1.8 nM and 1.2 nM, respectively.GBR 12783 dihydrochloride can improve memory performance and increase hippocampal acetylcholine release in rats.
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6-8 weeks
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Mesocarb HCl
Mesocarb hydrochloride, 9TH184G0MY, 1,2,3-Oxadiazolium, 3-(1-methyl-2-phenylethyl)-5-(((phenylamino)carbonyl)amino)-, chloride (1:1)
T202074117015-72-2
Mesocarb HCl is a psychoactive stimulant with an N-alkylated amphetamine structure, known for its selective inhibition of dopamine uptake.
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MCN-5292
MCN5292, MCN 5292
T202835105234-89-7
MCN-5292 is a dopamine uptake inhibitor.
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Lu 19005
Lu19-005, Lu-19-005, Lu-19005, Lu19005, Lu 19-005
T20288597229-15-7
Lu 19005 is a potent inhibitor of dopamine, serotonin, and norepinephrine uptake.
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GBR 13069 dihydrochloride
T2279967469-45-8
GBR 13069 dihydrochloride is a dopamine uptake inhibitor.
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6-8 weeks
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JHW 007 hydrochloride
T22877202645-74-7
JHW 007 hydrochloride is a Dopamine uptake inhibitor.
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6-8 weeks
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Rimcazole dihydrochloride
T2323475859-03-9
Rimcazole dihydrochloride is the hydrochloride salt of Rimcazole, a σ receptor antagonist. Rimcazole dihydrochloride also binds to dopamine transporter proteins and inhibits dopamine uptake.
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Amfonelic Acid
T2371815180-02-6
Amfonelic Acid is a dopamine uptake blocker.
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6-8 weeks
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Benzatropine
NK 02, Cogentinol, Cogentine, Benztropine, Akitan
T2378186-13-5
Benzatropine is a centrally active muscarinic antagonist. It also inhibits the uptake of dopamine. It has been used in the symptomatic treatment of Parkinson's Disease.
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6-8 weeks
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Piroheptine HCl
Trimol, Piroheptine Hydrochloride
T2464516378-22-6
Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.
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6-8 weeks
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Rimcazole
T2471275859-04-0
Rimcazole is a sigma receptor antagonist. It also binds to the dopamine transporter and inhibiting dopamine uptake.
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1-2 weeks
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JNJ-7925476 HCl
JNJ-7925476,JNJ7925476,JNJ 7925476
T27689109085-56-5
JNJ-7925476 HCl is a triple monoamine uptake inhibitor. JNJ-7925476 Salt blocks the dopamine transporter (DAT), norepinephrine transporter (NET) and serotonin transporter (SERT) in the central nervous system. The ED(50) values for JNJ-7925476 occupancy of
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6-8 weeks
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PD-89211
PD89211
T28349444725-49-9
PD 89211 is a selective dopamine D4 receptor antagonist with high selectivity for the DA D4.2 receptor (> 800-fold) as compared to other hDA receptor subtypes, rat brain serotonin, and adrenergic receptors. In vitro, PD 89211 reverses quinpirole-induced [
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6-8 weeks
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Org 24598
T37699372198-97-5
Potent and selective inhibitor of the glial glycine transporter GlyT1b (IC50 = 6.9 nM). Displays negligible activity at GlyT-2, adrenoreceptors, dopamine, 5HT receptors and noradrenaline, dopamine, 5HT and GABA transporters (pIC50 in vivo. Chue et al (2013) Glycine reuptake inhibition as a new therapeutic approach in schizophrenia: focus on the glycine transporter 1 (GlyT1). Curr.Pharm.Des. 19 1311 PMID:23194655 |Brown et al (2001) Discovery and SAR of org 24598-a selective glycine uptake inhibitor. Bioorg.Med.Chem.Lett. 11 2007 PMID:11454468 |Williams et al (2003) Development of a scintillation proximity assay for analysis of Na+/Cl- -dependent neurotransmitter transporter activity. Anal. Biochem. 321 31 PMID:12963052
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6-8 weeks
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