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Search Result

Search Results for "cb-1-in-1"

Compounds

Cat No. Product Name
T5996 CB1-IN-1 DBPR211,1-(2,4-二氯苯基)-N-1-哌啶基-4-[[(1-吡咯烷基磺酰基)氨基]甲基]-5-[5-[2-[4-(三氟甲基)苯基]乙炔基]-2-噻吩基]-1H-吡唑-3-甲酰胺 Cannabinoid Receptor
CB1-IN-1 是新型的外周大麻素-1受体 (CB1R) 拮抗剂，作用于CB1R (EC50 = 3 nM) 和 CB2R 的Ki 分别为0.3 nM 和 21 nM。
T30252 AZD1940 AZD 1940,UNII-0J0035E9FT,AZD-1940 Cannabinoid Receptor
AZD1940是一种高亲和力的大麻素CB(1)/CB(2)受体激动剂，具有口服活性，应用于口面疼痛的研究。
T10697 CB2R-IN-1 Others
CB2R-IN-1 is a potent inverse agonist of the cannabinoid CB2 receptor (Ki: 0.9 nM).
T5S1897 Linderalactone JAK , Apoptosis , Others
Linderalactone 是从乌药中分离出来的一种倍半萜烯内酯，通过调节凋亡相关蛋白的表达和抑制 JAK/STAT 信号通路来抑制癌细胞生长。它以 IC50值为 15 µM 来抑制肺癌 A-549 细胞的增殖。
T8425 Linoleoyl Ethanolamide TRP/TRPV Channel
Linoleoyl ethanolamide 是脂肪酸乙醇酰胺。它可弱结合 CB1 和 CB2 受体，并分别抑制[3H]CP-55,940的结合，Ki 分别为 10 和 25μM。它在引起小鼠过氧化氢酶方面的效力是 anandamide 的...
T4654 (±)-Ibipinabant (±)-SLV319,SLV319,(±)-BMS6462 Cannabinoid Receptor
SLV319 是一种有效选择性的大麻素-1 (CB-1) 受体拮抗剂，IC50=22 nM。(±)-SLV319 是 SLV319的消旋体。
T36520 COR659 Cannabinoid Receptor , GABA Receptor
COR659 是一种有效的 GABAB 的阳性变构调节剂。COR659具有缓解大鼠对酒精和巧克力成瘾的作用。
T23099 O-2050 Others
O-2050 是一种高亲和力的大麻素CB1受体拮抗剂，Ki 为 2.5 nM。O-2050 抑制大麻素 CB2受体，Ki 为 0.2 nM。O-2050 减少了小鼠的食物摄入量，并且引起小鼠运动。
T28235 OMDM169 OMDM-169,OMDM 169
OMDM169 is a potent and selective MAGL inhibitor. OMDM169 could enhances 2-AG levels and of exerts analgesic activity vi...
T61336 Numidargistat dihydrochloride
Numidargistat dihydrochloride (CB-1158) is a highly potent and orally active chemical compound that effectively inhibits...
T38028 (R)-(+)-Docosahexaenyl-1'-Hydroxy-2'-Propylamide
N-Acyl ethanolamines (NAEs) have diverse biological actions that are strongly affected by the associated acyl group. Doc...
T39309 Telaglenastat hydrochloride CB-839 hydrochloride
Telaglenastat (CB-839) hydrochloride is a first-in-class, reversible, and orally active inhibitor of glutaminase 1 (GLS1...
T38029 (R)-(+)-Linoleyl-1'-Hydroxy-2'-Propylamide
N-Acyl ethanolamines have diverse biological actions that are strongly affected by the associated acyl group. Linoleoyl ...
T38138 Arachidonoyl 2'-Chloroethylamide Arachidonoyl 2'-Chloroethylamide,2'-chloro-AEA,ACEA
Arachidonoyl 2-chloroethylamide (ACEA) is a potent and selective cannabinoid (CB) receptor 1 agonist with Ki values of 1...
T38204 GAT229
GAT229 is a positive allosteric modulator of cannabinoid receptor 1 (CB1) and the S-(-) enantiomer of the CB1 modulator ...
CB1-IN-1
T5996
synonym: DBPR211,1-(2,4-二氯苯基)-N-1-哌啶基-4-[[(1-吡咯烷基磺酰基)氨基]甲基]-5-[5-[2-[4-(三氟甲基)苯基]乙炔基]-2-噻吩基]-1H-吡唑-3-甲酰胺
Target:
AZD1940
T30252
synonym: AZD 1940,UNII-0J0035E9FT,AZD-1940
Target:
CB2R-IN-1
T10697
synonym:
Target:
Linderalactone
T5S1897
synonym:
Target:
Linoleoyl Ethanolamide
T8425
synonym:
Target:
(±)-Ibipinabant
T4654
synonym: (±)-SLV319,SLV319,(±)-BMS6462
Target:
COR659
T36520
synonym:
Target:
O-2050
T23099
synonym:
Target:
OMDM169
T28235
synonym: OMDM-169,OMDM 169
Target:
Numidargistat dihydrochloride
T61336
synonym:
Target:
(R)-(+)-Docosahexaenyl-1'-Hydroxy-2'-Propylamide
T38028
synonym:
Target:
Telaglenastat hydrochloride
T39309
synonym: CB-839 hydrochloride
Target:
(R)-(+)-Linoleyl-1'-Hydroxy-2'-Propylamide
T38029
synonym:
Target:
Arachidonoyl 2'-Chloroethylamide
T38138
synonym: Arachidonoyl 2'-Chloroethylamide,2'-chloro-AEA,ACEA
Target:
GAT229
T38204
synonym:
Target:
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