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Results for "

125i-cgtyr

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    99
    TargetMol | Inhibitors_Agonists
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    TargetMol | Inhibitors_Agonists
Cholylglycyltyrosine
I-Cholylglycyltyrosine, Cholyl-glycyl-tyrosine, Chol-gly-tyr, 125I-Cgtyr
T3090667319-56-6
Cholylglycyltyrosine is a hepatobiliary imaging agent.
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Dexamethasone
Prednisolone F, NSC 34521, MK 125, Hexadecadrol
T107650-02-2
Dexamethasone (Hexadecadrol) is a glucocorticoid receptor agonist and IL receptor modulator with anti-inflammatory and immunosuppressive properties that induces autophagy and inhibits LPS-induced inflammatory responses in macrophages.
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TargetMol | Inhibitor Hot
PSI-697
WAY-197697, WAY197697, PSI697, P-Selectin Inhibitor
T16676851546-61-7In house
PSI-697 (P-Selectin Inhibitor) is an orally active P-selectin inhibitor with anti-inflammatory and anti-thrombotic effects, useful for studying cardiovascular diseases such as atherosclerosis.
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6-8 weeks
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TargetMol
Laromustine
VNP 40101M, VNP40101M
T70229173424-77-6In house
Laromustine (VNP40101M) is a sulfonyl hydrolytic alkylating prodrug used in cancer therapy with significant anticancer activity. Inhibiting thioredoxin reductase can be used to study acute myeloid leukemia.
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6-8 weeks
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Tigecycline
GAR-936
T1569220620-09-7
Tigecycline (GAR-936) is a broad-spectrum glycylcycline antibiotic derived from tetracycline that binds to the 30S ribosomal subunit, disrupting the binding of aminoacyl-tRNA to the mRNA-ribosome complex.
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Nystatin
Stamycin, Nystavescent, Fungicidin
T16781400-61-9
Nystatin (Fungicidin) is a topical and oral antifungal agent with activity against many species of yeast and candida albicans, which is used largely to treat skin and oropharyngeal candidiasis.
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Etravirine
TMC125, R165335
T2551269055-15-4
Etravirine (R165335) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor. Etravirine is designed to be active against HIV isolates with mutations that confer resistance to the two most commonly prescribed first-generation NNRTIs. It can bind the enzyme reverse transcriptase (RT) in multiple conformations, both for native and mutant RT, thereby blocking the enzymatic activity of RT.
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Octyl gallate
Gallic acid octyl ester, n-Octylgallate, Octyl 3,4,5-trihydroxybenzoate, Progallin O, Stabilizer GA-8
T2S18651034-01-1
1. Octyl Gallate is an antioxidant approved by the US Food and Drug Administration (FDA) as a food additive. 2. Octyl Gallate has antimetastatic activity. 3. Octyl Gallate shows antimicrobial activity against H. pylori, with a minimum inhibitory concentration (MIC) value of 125 ug mL. 4. Combination therapy with octyl gallate and ferulic acid improves cognition and neurodegeneration in a transgenic mouse model of Alzheimer's disease.5. Octyl Gallate is a potential anticancer agent, it exhibited decreased MCF-7 & MDA-MB-231 survival and induced apoptosis, with IC50 value of 40 uM. 6. Octyl gallate (Octyl 3,4,5-trihydroxybenzoate) has antiviral activity, it shows an inhibitory effect on the growth of herpes simplex virus type 1 (HSV-1) in HEp-2 or Vero cells. 7. Octyl gallate shows antifungal activity against Saccharomyces cerevisiae ATCC7754 and Zygosaccharomyces bailii ATCC 60483.
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KRN-633
KRN633
T6137286370-15-8
KRN-633 is an effective VEGFR inhibitor. The IC50s of KRN-633(KRN633) for VEGFR1, VEGFR2, and VEGFR3 is 170, 160 and 125 nM, respectively.
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TargetMol | Inhibitor Sale
PI4KIIIbeta-IN-9
T124691429624-84-9
PI4KIIIbeta-IN-9 is a potent inhibitor of PI4KIIIβ [IC50 of 7 nM].
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TargetMol | Inhibitor Sale
PF-CBP1
T39731962928-21-7
PF-CBP1 HCl is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP). It inhibits CREBBP (IC50: 125 nM) and p300 bromodomains (IC50: 363 nM).
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TargetMol | Inhibitor Sale
Simufilam dihydrochloride
PTI-125 dihydrochloride
T91722480226-06-8
Simufilam dihydrochloride (PTI-125 dihydrochloride) is a low toxicity, orally active filamin A (FLNA) activator, which can be used for the research of Alzheimer's disease. Simufilam dihydrochloride preferentially binds altered FLNA and restores its native conformation, restoring receptor and synaptic activities and reducing its α7nAChR TLR4 associations and downstream pathologies.
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CD80-IN-3
T10722486449-65-4
CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80 CD28 interaction (Kd: 125 nM; EC50: 630 nM).
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Etravirine D4
R-165335 D4,TMC-125 D4
T112471142095-93-9
Etravirine is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used for the treatment of HIV. Etravirine D4 is the deuterium labeled Etravirine.
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7-10 days
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JBJ-04-125-02
T117142060610-53-7
JBJ-04-125-02 can inhibit cancer cell proliferation and EGFRL858R T790M C797S signaling. JBJ-04-125-02 has anti-tumor activities. JBJ-04-125-02 is a potent, mutant-selective, allosteric and orally active EGFR inhibitor with an IC50 of 0.26 nM for EGFRL858
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6-8 weeks
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Lesopitron dihydrochloride
E4424
T11839132449-89-9
Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.
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1-2 weeks
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MOZ-IN-2
T120982055397-88-9
MOZ-IN-2 is an protein MOZ inhibitor(IC50 of 125 μM).
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XPC-6444
T133592230144-21-3
XPC-6444 is a isoform-selective, and CNS-penetrant inhibitor of NaV1.6 with IC50 of41 nM for hNaV1.6,with anticonvulsant activity.
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6-8 weeks
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Acivicin
U-42126, U42126, U 42126, AT-125, AT125, AT 125
T1411442228-92-2
Acivicin (AT-125), a chlorinated amino acid antibiotic produced by Streptomyces porcineus, is a γ-glutamyl transpeptidase (GGT) inhibitor that crosses the blood-brain barrier, exhibits anticancer and antiparasitic activity, and is used in the study of visceral leishmaniasis.
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AM679
T142051206880-66-1
AM679 is a potent and selective FLAP inhibitor with IC50s of 2.2 nM/0.6 nM/154 nM for FLAP binding/hLA/hWB respectively. IC50 value: 2.2 nM/0.6 nM/154 nM(FLAP binding/hLA/hWB) [1] AM679 showed an improved CYP inhibition profile (IC50 3A4 = 16.7 lM, 2C9 =
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10-14 weeks
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M443
T159431820684-31-8
M443 is a potent small molecule inhibitor of MRK that inhibits radiation-induced activation of p38 and Chk2 and can be used in cancer research.
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6-8 weeks
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MSN-125
T161551592908-16-1
MSN-125 effectively inhibits Bax Bak-mediated apoptosis in HCT-116, BMK Cells, and primary cortical neurons protect primary neurons against glutamate excitotoxicity. MSN-125 is an effective Bax and Bak oligomerization inhibitor. MSN-125 prevents mitochond
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6-8 weeks
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PRN694
T165781575818-46-0
PRN694 shows extended target residence time on ITK and RLK, enabling durable attenuation of effector cells in vitro and in vivo. PRN694 is an irreversible, highly selective, and effective covalent interleukin-2-inducible T-cell kinase (ITK) and resting ly
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3-6 months
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Dot1L-IN-9
T200597
Dot1L-IN-9 (Compound 12) is a DOT1L inhibitor with an IC50 of 125 nM. It effectively reduces H3K79 dimethylation and is utilized in leukemia research.
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