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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T21419 Diphenhydramine 58-73-1 99.49%
Diphenhydramine
Diphenhydramine (Syntedril), a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the...
T1097 Loratadine 79794-75-5 99.49%
Loratadine
Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical an...
T8439 Clobenpropit dihydrobromide 145231-35-2 99.48%
Clobenpropit dihydrobromide
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
T0263 Chloropyramine hydrochloride 6170-42-9 99.45%
Chloropyramine hydrochloride
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.
T2004 Ciproxifan maleate 184025-19-2 99.45%
Ciproxifan maleate
Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at...
T7564 Chlorphenoxamine 77-38-3 99.44%
Chlorphenoxamine
Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
T0236 Azatadine dimaleate 3978-86-7 99.4%
Azatadine dimaleate
Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).
T21428 Mianserin 24219-97-4 99.39%
Mianserin
Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, an...
T22746 Tesmilifene fumarate 1185241-83-1 99.38%
Tesmilifene fumarate
Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。
T68150 Talastine 16188-61-7 99.37%
Talastine
Talastine is an antihistamine compound that can induce an allergic rash.
T1266 Terfenadine 50679-08-8 99.36%
Terfenadine
Terfenadine ((±)-Terfenadine) is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist...
T0211 Azelastine 58581-89-8 99.35%
Azelastine
Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
T0031L Ziprasidone hydrochloride 122883-93-6 99.34%
Ziprasidone hydrochloride
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic acti...
T0137 Mirtazapine 85650-52-8 99.3%
Mirtazapine
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
T0205 Brompheniramine maleate 980-71-2 99.3%
Brompheniramine maleate
Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
T7176 Pitolisant hydrochloride 903576-44-3 99.26%
Pitolisant hydrochloride
Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).
T9084 Cetirizine Impurity B dihydrochloride 1000690-91-4 99.24%
Cetirizine Impurity B dihydrochloride
Cetirizine Impurity B dihydrochloride (De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride) is an impurity of Cetirizine dihydrochloride. Cetirizine is a s...
T0059 Diphenylpyraline hydrochloride 132-18-3 99.22%
Diphenylpyraline hydrochloride
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) is used in the treatment of Parkinsonism.It is a first-generation antihistami...
T0942 Quinacrine dihydrochloride 69-05-6 99.18%
Quinacrine dihydrochloride
Quinacrine dihydrochloride (Mepacrine dihydrochloride) is the dihydrochloride salt of the 9-aminoacridine derivative quinacrine with potential antineoplastic and...
T22501 2-Pyridylethylamine dihydrochloride 3343-39-3 99.17%
2-Pyridylethylamine dihydrochloride
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
Diphenhydramine
T21419
Diphenhydramine (Syntedril), a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the...
Loratadine
T1097
Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical an...
Clobenpropit dihydrobromide
T8439
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
Chloropyramine hydrochloride
T0263
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.
Ciproxifan maleate
T2004
Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at...
Chlorphenoxamine
T7564
Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
Azatadine dimaleate
T0236
Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).
Mianserin
T21428
Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, an...
Tesmilifene fumarate
T22746
Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。
Talastine
T68150
Talastine is an antihistamine compound that can induce an allergic rash.
Terfenadine
T1266
Terfenadine ((±)-Terfenadine) is a prodrug that is metabolized by intestinal CYP3A4 to the active form fexofenadine, a selective histamine H1-receptor antagonist...
Azelastine
T0211
Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
Ziprasidone hydrochloride
T0031L
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic acti...
Mirtazapine
T0137
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
Brompheniramine maleate
T0205
Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
Pitolisant hydrochloride
T7176
Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).
Cetirizine Impurity B dihydrochloride
T9084
Cetirizine Impurity B dihydrochloride (De(carboxymethoxy) Cetirizine Acetic Acid Dihydrochloride) is an impurity of Cetirizine dihydrochloride. Cetirizine is a s...
Diphenylpyraline hydrochloride
T0059
Diphenylpyraline hydrochloride (4-Diphenylmethoxy-1-methylpiperidine hydrochloride) is used in the treatment of Parkinsonism.It is a first-generation antihistami...
Quinacrine dihydrochloride
T0942
Quinacrine dihydrochloride (Mepacrine dihydrochloride) is the dihydrochloride salt of the 9-aminoacridine derivative quinacrine with potential antineoplastic and...
2-Pyridylethylamine dihydrochloride
T22501
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
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TargetMol