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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T1090 Perphenazine 58-39-9 99.63%
Perphenazine
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
T0157 Roxatidine Acetate hydrochloride 93793-83-0 99.61%
Roxatidine Acetate hydrochloride
Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. It inhibits gastric acid secretion and ulcer formation....
T4250 Bilastine 202189-78-4 99.61%
Bilastine
Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of ...
T15772 Lodoxamide tromethamine 63610-09-3 99.58%
Lodoxamide tromethamine
Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic conjunctivi...
T79500 KSK94 2566716-07-0 99.56%
KSK94
KSK94 is a specific H3 receptor antagonist that inhibits H3, sigma-1, and sigma-2 receptors , with Ki values of 7.9, 2958, and 75.2 nM, respectively, and can be ...
T6426 Buclizine dihydrochloride 129-74-8 99.56%
Buclizine dihydrochloride
Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and anti...
T25737 Linetastine 159776-68-8 99.55%
Linetastine
Linetastine (TMK-688) is a 5-lipoxygenase inhibitor (5-LOX) that inhibits leukotriene production and antagonizes the effects of histamine.Linetastine is used in ...
T1308 Orphenadrine hydrochloride 341-69-5 99.54%
Orphenadrine hydrochloride
Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.
T3429 Protopine 130-86-9 99.54%
Protopine
Protopine (Fumarine) is a benzylisoquinoline alkaloid. It has been found to inhibit histamine H1 receptors and platelet aggregation, and acts as an analgesic.
T0031L2 Ziprasidone 146939-27-7 99.53%
Ziprasidone
Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T3963 VUF10460 1028327-66-3 99.53%
VUF10460
VUF10460 is a non-imidazole histamine H4 receptor agonist.
T68921 Impromidine hydrochloride 65573-02-6 99.50%
Impromidine hydrochloride
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.
T9353 OXOMEMAZINE 3689-50-7 99.49%
OXOMEMAZINE
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M...
T21419 Diphenhydramine 58-73-1 99.49%
Diphenhydramine
Diphenhydramine (Syntedril), a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the...
T1097 Loratadine 79794-75-5 99.49%
Loratadine
Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical an...
T8439 Clobenpropit dihydrobromide 145231-35-2 99.48%
Clobenpropit dihydrobromide
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
T0263 Chloropyramine hydrochloride 6170-42-9 99.45%
Chloropyramine hydrochloride
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.
T2004 Ciproxifan maleate 184025-19-2 99.45%
Ciproxifan maleate
Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at...
T1393 Sodium butanoate 156-54-7 99.44%
Sodium butanoate
Sodium butanoate (Sodium Butyrate) is the sodium salt of butyrate with potential antineoplastic activity. Butyrate, a short chain fatty acid, competitively binds...
T7564 Chlorphenoxamine 77-38-3 99.44%
Chlorphenoxamine
Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
Perphenazine
T1090
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
Roxatidine Acetate hydrochloride
T0157
Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. It inhibits gastric acid secretion and ulcer formation....
Bilastine
T4250
Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of ...
Lodoxamide tromethamine
T15772
Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic conjunctivi...
KSK94
T79500
KSK94 is a specific H3 receptor antagonist that inhibits H3, sigma-1, and sigma-2 receptors , with Ki values of 7.9, 2958, and 75.2 nM, respectively, and can be ...
Buclizine dihydrochloride
T6426
Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and anti...
Linetastine
T25737
Linetastine (TMK-688) is a 5-lipoxygenase inhibitor (5-LOX) that inhibits leukotriene production and antagonizes the effects of histamine.Linetastine is used in ...
Orphenadrine hydrochloride
T1308
Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.
Protopine
T3429
Protopine (Fumarine) is a benzylisoquinoline alkaloid. It has been found to inhibit histamine H1 receptors and platelet aggregation, and acts as an analgesic.
Ziprasidone
T0031L2
Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
VUF10460
T3963
VUF10460 is a non-imidazole histamine H4 receptor agonist.
Impromidine hydrochloride
T68921
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.
OXOMEMAZINE
T9353
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M...
Diphenhydramine
T21419
Diphenhydramine (Syntedril), a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the...
Loratadine
T1097
Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical an...
Clobenpropit dihydrobromide
T8439
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
Chloropyramine hydrochloride
T0263
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.
Ciproxifan maleate
T2004
Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at...
Sodium butanoate
T1393
Sodium butanoate (Sodium Butyrate) is the sodium salt of butyrate with potential antineoplastic activity. Butyrate, a short chain fatty acid, competitively binds...
Chlorphenoxamine
T7564
Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
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TargetMol