T1090 |
Perphenazine
|
58-39-9
|
99.63%
|
|
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
|
T0157 |
Roxatidine Acetate hydrochloride
|
93793-83-0
|
99.61%
|
|
Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. It inhibits gastric acid secretion and ulcer formation....
|
T4250 |
Bilastine
|
202189-78-4
|
99.61%
|
|
Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of ...
|
T15772 |
Lodoxamide tromethamine
|
63610-09-3
|
99.58%
|
|
Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic conjunctivi...
|
T79500 |
KSK94
|
2566716-07-0
|
99.56%
|
|
KSK94 is a specific H3 receptor antagonist that inhibits H3, sigma-1, and sigma-2 receptors , with Ki values of 7.9, 2958, and 75.2 nM, respectively, and can be ...
|
T6426 |
Buclizine dihydrochloride
|
129-74-8
|
99.56%
|
|
Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and anti...
|
T25737 |
Linetastine
|
159776-68-8
|
99.55%
|
|
Linetastine (TMK-688) is a 5-lipoxygenase inhibitor (5-LOX) that inhibits leukotriene production and antagonizes the effects of histamine.Linetastine is used in ...
|
T1308 |
Orphenadrine hydrochloride
|
341-69-5
|
99.54%
|
|
Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.
|
T3429 |
Protopine
|
130-86-9
|
99.54%
|
|
Protopine (Fumarine) is a benzylisoquinoline alkaloid. It has been found to inhibit histamine H1 receptors and platelet aggregation, and acts as an analgesic.
|
T0031L2 |
Ziprasidone
|
146939-27-7
|
99.53%
|
|
Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
|
T3963 |
VUF10460
|
1028327-66-3
|
99.53%
|
|
VUF10460 is a non-imidazole histamine H4 receptor agonist.
|
T68921 |
Impromidine hydrochloride
|
65573-02-6
|
99.50%
|
|
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.
|
T9353 |
OXOMEMAZINE
|
3689-50-7
|
99.49%
|
|
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M...
|
T21419 |
Diphenhydramine
|
58-73-1
|
99.49%
|
|
Diphenhydramine (Syntedril), a first-generation antihistamine possessing antiemetic, antitussive, anticholinergic, and sedative properties, is mainly used in the...
|
T1097 |
Loratadine
|
79794-75-5
|
99.49%
|
|
Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria. Unlike most classical an...
|
T8439 |
Clobenpropit dihydrobromide
|
145231-35-2
|
99.48%
|
|
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)
|
T0263 |
Chloropyramine hydrochloride
|
6170-42-9
|
99.45%
|
|
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.
|
T2004 |
Ciproxifan maleate
|
184025-19-2
|
99.45%
|
|
Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at...
|
T1393 |
Sodium butanoate
|
156-54-7
|
99.44%
|
|
Sodium butanoate (Sodium Butyrate) is the sodium salt of butyrate with potential antineoplastic activity. Butyrate, a short chain fatty acid, competitively binds...
|
T7564 |
Chlorphenoxamine
|
77-38-3
|
99.44%
|
|
Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
|