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GABA Receptor

The GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels (also known as ionotropic receptors); whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors.
Cat. No. Product name CAS No. Purity Chemical Structure
T11684 Isoguvacine hydrochloride 68547-97-7 98%
Isoguvacine hydrochloride is a GABA receptor agonist.
T6355 (R)-baclofen 69308-37-8 98%
(R)-baclofena, a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.
T14571 Bifenazate 149877-41-8 98%
Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.
T7822 Pagoclone 133737-32-3 98%
Pagoclone is a GABA receptor agonist and can be used for studies on the treatment of stuttering, panic disorder, and generalized anxiety. Pagoclone is a partial ...
T4688 Pipequaline hydrochloride 80221-58-5 98%
Pipequaline is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure t...
T6507 Gabapentin hydrochloride 60142-95-2 98%
Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain.
TN1325 (2S)-6-Prenylnaringenin 68236-13-5 98%
6-Prenylnaringenin is an isomer of the potent phytoestrogen, 8-prenylnaringenin.
T2749 Ginkgolide A 15291-75-5 98%
Ginkgolide A is a highly active PAF antagonist cage molecule that is isolated from the leaves of the Ginkgo biloba tree. Shows potential in a wide variety of inf...
T7064 Valproic Acid 99-66-1 98%
Valproic Acid is a branched chain fatty acid which potentially enhances central GABAergic neurotransmission and inhibits Na+ channels. Currently, the various mol...
T26600 Alpidem 82626-01-5 98%
Alpidem is an anxiolytic drug from the imidazopyridine family. Alpidem does not produce sedative effects at normal doses, and is instead used specifically for th...
T0024 Primidone 125-33-7 98%
Primidone is an anticonvulsant of the pyrimidinedione class.
TQ0023 Lorediplon 917393-39-6 98%
Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.
T2S1814 P-Hydroxybenzaldehyde 123-08-0 98%
1. 4-Hydroxybenzaldehyde shows an inhibitory effect on the GABA transaminase to contribute to an antiepileptic and anticonvulsive activity, and its inhibitory ac...
T4440 Saclofen 125464-42-8 98%
Saclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7....
TQ0040 ONO-8590580 1802661-73-9 98%
ONO-8590580 is a negative allosteric modulator of GABAA α5.
T12207 NEO 376 496921-73-4 98%
NEO 376 is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.
T36520 COR659 544450-68-2 98%
COR659 is a GABAB positive allosteric modulator (PAM) . COR659 suppresses alcohol and chocolate self-administration in rats[1]. COR659 apparently exerts its effe...
T16811 RWJ-51204 205701-85-5 98%
RWJ-51204 is A potent and selective adenosine A2A receptor antagonist. RWJ-51204 is a partial agonist of GABA(A) receptor (IC50: 0.2-2 nM), which has neuroprotec...
T3S2100 (-)-Securinine 5610-40-2 98%
(-)-Securinine is plant-derived alkaloid and also a GABAA receptor antagonist.
TQ0119 Cirsimaritin 6601-62-3 98%
Cirsimaritin exhibits antibacterial, anti-inflammation, anti-tumor, antioxidant properties and renal protection. Cirsimaritin binds weakly to the benzodiazepine ...
Isoguvacine hydrochloride
T11684
Isoguvacine hydrochloride is a GABA receptor agonist.
(R)-baclofen
T6355
(R)-baclofena, a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.
Bifenazate
T14571
Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.
Pagoclone
T7822
Pagoclone is a GABA receptor agonist and can be used for studies on the treatment of stuttering, panic disorder, and generalized anxiety. Pagoclone is a partial ...
Pipequaline hydrochloride
T4688
Pipequaline is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure t...
Gabapentin hydrochloride
T6507
Gabapentin HCl is a GABA analogue, used to treat seizures and neuropathic pain.
(2S)-6-Prenylnaringenin
TN1325
6-Prenylnaringenin is an isomer of the potent phytoestrogen, 8-prenylnaringenin.
Ginkgolide A
T2749
Ginkgolide A is a highly active PAF antagonist cage molecule that is isolated from the leaves of the Ginkgo biloba tree. Shows potential in a wide variety of inf...
Valproic Acid
T7064
Valproic Acid is a branched chain fatty acid which potentially enhances central GABAergic neurotransmission and inhibits Na+ channels. Currently, the various mol...
Alpidem
T26600
Alpidem is an anxiolytic drug from the imidazopyridine family. Alpidem does not produce sedative effects at normal doses, and is instead used specifically for th...
Primidone
T0024
Primidone is an anticonvulsant of the pyrimidinedione class.
Lorediplon
TQ0023
Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.
p-Hydroxybenzaldehyde
T2S1814
1. 4-Hydroxybenzaldehyde shows an inhibitory effect on the GABA transaminase to contribute to an antiepileptic and anticonvulsive activity, and its inhibitory ac...
Saclofen
T4440
Saclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7....
ONO-8590580
TQ0040
ONO-8590580 is a negative allosteric modulator of GABAA α5.
NEO 376
T12207
NEO 376 is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.
COR659
T36520
COR659 is a GABAB positive allosteric modulator (PAM) . COR659 suppresses alcohol and chocolate self-administration in rats[1]. COR659 apparently exerts its effe...
RWJ-51204
T16811
RWJ-51204 is A potent and selective adenosine A2A receptor antagonist. RWJ-51204 is a partial agonist of GABA(A) receptor (IC50: 0.2-2 nM), which has neuroprotec...
(-)-Securinine
T3S2100
(-)-Securinine is plant-derived alkaloid and also a GABAA receptor antagonist.
Cirsimaritin
TQ0119
Cirsimaritin exhibits antibacterial, anti-inflammation, anti-tumor, antioxidant properties and renal protection. Cirsimaritin binds weakly to the benzodiazepine ...
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