TN1370 |
Allura Red AC
|
25956-17-6
|
98%
|
|
Allura Red AC and amaranth are very important food azo dyes used in food, drug, paper, cosmetic and textile industries.
|
TN2245 |
Sunset Yellow FCF
|
2783-94-0
|
98%
|
|
Sunset yellow FCF and Brilliant Blue FCF are used as colorant food additives in many food products, they can have cytotoxic and genotoxic potential, it care must...
|
T15749 |
LGD-2226
|
328947-93-9
|
98%
|
|
LGD-2226 is a selective and orally active androgen receptor modulator (EC50: 0.2 nM, Ki: 1.5 nM for the human androgen receptor). LGD-2226 can be used for muscle...
|
T19449 |
N-desmethyl Enzalutamide D6
|
T19449
|
98%
|
|
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
|
TN1061 |
Ganoderol B
|
104700-96-1
|
98%
|
|
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate ...
|
T14675 |
BMS-564929
|
627530-84-1
|
98%
|
|
BMS-564929 is an agonist of androgen receptor (AR, Ki of 2.11±0.16 nM).
|
T15816 |
LY341495
|
201943-63-7
|
98%
|
|
LY341495 is an antagonist of metabotropic glutamate receptor (IC50s: 2.9 nM, 10 nM, 170 nM for mGluR-2, mGluR-3, mGluR-8, respectively).
|
TN4774 |
Physalin A
|
23027-91-0
|
98%
|
|
Physalin A exerts anti-tumor activity in non-small cell lung cancer cell lines by suppressing JAK/STAT3 signaling, it inhibits androgen-independent prostate canc...
|
T10946 |
D4-abiraterone
|
154229-21-7
|
98%
|
|
D4-Abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid 5a-reductase (SRD5A), the main metabolite of abiraterone. D4-Abira...
|
TN1663 |
Ganoderic acid DM
|
173075-45-1
|
98%
|
|
Ganoderic acid DM is an antiandrogenic osteoclastogenesis inhibitor, it especially suppresses the expression of c-Fos and nuclear factor of activated T cells c1 ...
|
TMA1012 |
Ganoderiol F
|
114567-47-4
|
98%
|
|
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
|
T14843 |
Bifluranol
|
34633-34-6
|
98%
|
|
Bifluranol is an anti-androgen.
|
T12928 |
SK33
|
1928724-23-5
|
98%
|
|
SK33 is a potent and tissue selective anti-androgen,and is a trifluoromethylated enobosarm analog, SK33 reduces androgen receptor (AR) transcriptional activity.
|
T10896L |
CSRM617 hydrochloride
|
1353749-74-2
|
98%
|
|
CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 ( OC2, a master regulator of androgen receptor) with a K d of 7...
|
T39695 |
ARD-2128
|
2222111-87-5
|
98%
|
|
ARD-2128 is a highly potent, orally bioavailable PROTAC degrader of androgen receptor (AR). ARD-2128 effectively reduces AR protein, suppresses AR-regulated gene...
|
T20625 |
Prochloraz
|
67747-09-5
|
98%
|
|
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
|
T11410L |
GLPG0492
|
1215085-92-9
|
98%
|
|
GLPG0492 is a novel selective androgen receptor modulator. After oral dosing, it showed anabolic activity on muscle, strongly dissociated from the androgenic act...
|
TN1067 |
Galloylpaeoniflorin
|
122965-41-7
|
98%
|
|
6'-O-Galloylpaeoniflorin (GPF) may be developed as a cytoprotector against ROS-mediated oxidative stress
|
T20761 |
RU 59063
|
155180-53-3
|
98%
|
|
RU 59063 is a prototype of high-affinity nonsteroidal androgen receptor (AR) ligands.
|
T8860 |
DSRM-3716
|
58142-99-7
|
98%
|
|
Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of a...
|