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Androgen Receptor

The androgen receptor (AR), also known as NR3C4 (nuclear receptor subfamily 3, group C, member 4), is a type of nuclear receptor that is activated by binding any of the androgenic hormones, including testosterone and dihydrotestosterone in the cytoplasm and then translocating into the nucleus.
Cat. No. Product name CAS No. Purity Chemical Structure
TN1370 Allura Red AC 25956-17-6 98%
Allura Red AC and amaranth are very important food azo dyes used in food, drug, paper, cosmetic and textile industries.
TN2245 Sunset Yellow FCF 2783-94-0 98%
Sunset yellow FCF and Brilliant Blue FCF are used as colorant food additives in many food products, they can have cytotoxic and genotoxic potential, it care must...
T15749 LGD-2226 328947-93-9 98%
LGD-2226 is a selective and orally active androgen receptor modulator (EC50: 0.2 nM, Ki: 1.5 nM for the human androgen receptor). LGD-2226 can be used for muscle...
T19449 N-desmethyl Enzalutamide D6 T19449 98%
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
TN1061 Ganoderol B 104700-96-1 98%
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate ...
T14675 BMS-564929 627530-84-1 98%
BMS-564929 is an agonist of androgen receptor (AR, Ki of 2.11±0.16 nM).
T15816 LY341495 201943-63-7 98%
LY341495 is an antagonist of metabotropic glutamate receptor (IC50s: 2.9 nM, 10 nM, 170 nM for mGluR-2, mGluR-3, mGluR-8, respectively).
TN4774 Physalin A 23027-91-0 98%
Physalin A exerts anti-tumor activity in non-small cell lung cancer cell lines by suppressing JAK/STAT3 signaling, it inhibits androgen-independent prostate canc...
T10946 D4-abiraterone 154229-21-7 98%
D4-Abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid 5a-reductase (SRD5A), the main metabolite of abiraterone. D4-Abira...
TN1663 Ganoderic acid DM 173075-45-1 98%
Ganoderic acid DM is an antiandrogenic osteoclastogenesis inhibitor, it especially suppresses the expression of c-Fos and nuclear factor of activated T cells c1 ...
TMA1012 Ganoderiol F 114567-47-4 98%
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
T14843 Bifluranol 34633-34-6 98%
Bifluranol is an anti-androgen.
T12928 SK33 1928724-23-5 98%
SK33 is a potent and tissue selective anti-androgen,and is a trifluoromethylated enobosarm analog, SK33 reduces androgen receptor (AR) transcriptional activity.
T10896L CSRM617 hydrochloride 1353749-74-2 98%
CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 ( OC2, a master regulator of androgen receptor) with a K d of 7...
T39695 ARD-2128 2222111-87-5 98%
ARD-2128 is a highly potent, orally bioavailable PROTAC degrader of androgen receptor (AR). ARD-2128 effectively reduces AR protein, suppresses AR-regulated gene...
T20625 Prochloraz 67747-09-5 98%
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
T11410L GLPG0492 1215085-92-9 98%
GLPG0492 is a novel selective androgen receptor modulator. After oral dosing, it showed anabolic activity on muscle, strongly dissociated from the androgenic act...
TN1067 Galloylpaeoniflorin 122965-41-7 98%
6'-O-Galloylpaeoniflorin (GPF) may be developed as a cytoprotector against ROS-mediated oxidative stress
T20761 RU 59063 155180-53-3 98%
RU 59063 is a prototype of high-affinity nonsteroidal androgen receptor (AR) ligands.
T8860 DSRM-3716 58142-99-7 98%
Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of a...
Allura Red AC
TN1370
Allura Red AC and amaranth are very important food azo dyes used in food, drug, paper, cosmetic and textile industries.
Sunset Yellow FCF
TN2245
Sunset yellow FCF and Brilliant Blue FCF are used as colorant food additives in many food products, they can have cytotoxic and genotoxic potential, it care must...
LGD-2226
T15749
LGD-2226 is a selective and orally active androgen receptor modulator (EC50: 0.2 nM, Ki: 1.5 nM for the human androgen receptor). LGD-2226 can be used for muscle...
N-desmethyl Enzalutamide D6
T19449
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
Ganoderol B
TN1061
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate ...
BMS-564929
T14675
BMS-564929 is an agonist of androgen receptor (AR, Ki of 2.11±0.16 nM).
LY341495
T15816
LY341495 is an antagonist of metabotropic glutamate receptor (IC50s: 2.9 nM, 10 nM, 170 nM for mGluR-2, mGluR-3, mGluR-8, respectively).
Physalin A
TN4774
Physalin A exerts anti-tumor activity in non-small cell lung cancer cell lines by suppressing JAK/STAT3 signaling, it inhibits androgen-independent prostate canc...
D4-abiraterone
T10946
D4-Abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid 5a-reductase (SRD5A), the main metabolite of abiraterone. D4-Abira...
Ganoderic acid DM
TN1663
Ganoderic acid DM is an antiandrogenic osteoclastogenesis inhibitor, it especially suppresses the expression of c-Fos and nuclear factor of activated T cells c1 ...
Ganoderiol F
TMA1012
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
Bifluranol
T14843
Bifluranol is an anti-androgen.
SK33
T12928
SK33 is a potent and tissue selective anti-androgen,and is a trifluoromethylated enobosarm analog, SK33 reduces androgen receptor (AR) transcriptional activity.
CSRM617 hydrochloride
T10896L
CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 ( OC2, a master regulator of androgen receptor) with a K d of 7...
ARD-2128
T39695
ARD-2128 is a highly potent, orally bioavailable PROTAC degrader of androgen receptor (AR). ARD-2128 effectively reduces AR protein, suppresses AR-regulated gene...
Prochloraz
T20625
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
GLPG0492
T11410L
GLPG0492 is a novel selective androgen receptor modulator. After oral dosing, it showed anabolic activity on muscle, strongly dissociated from the androgenic act...
Galloylpaeoniflorin
TN1067
6'-O-Galloylpaeoniflorin (GPF) may be developed as a cytoprotector against ROS-mediated oxidative stress
RU 59063
T20761
RU 59063 is a prototype of high-affinity nonsteroidal androgen receptor (AR) ligands.
DSRM-3716
T8860
Isoquinoline, 5-iodo- (9CI) is a potent and selective inhibitor of SARM1(IC50 = 75 nM) by preventing axonal degeneration and by allowing functional recovery of a...
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