Search Result

Search Results for " receptor "

Targets

Oxytocin Receptor Estrogen/progestogen Receptor Androgen Receptor Thyroid hormone receptor(THR) Estrogen Receptor/ERR Glucocorticoid Receptor Opioid Receptor Melanocortin Receptor Prostaglandin Receptor Histamine Receptor Adenosine Receptor Neuropeptide Y Receptor Melatonin Receptor Bombesin Receptor LPL Receptor RXFP receptor Amylin Receptor Endothelin Receptor TSH Receptor Protease-activated Receptor Neurokinin receptor OX Receptor Glucagon Receptor CGRP Receptor LPA Receptor Neurotensin Receptor Adrenergic Receptor 5-HT Receptor Adiponectin receptor Apelin receptor Motilin Receptor P2Y Receptor RXDP receptor Sigma receptor Cannabinoid Receptor Bradykinin Receptor Leukotriene Receptor Dopamine Receptor Vasopressin Receptor GNRH Receptor S1P Receptor Melanin-concentrating Hormone Receptor (MCHR) Thrombopoietin Receptor IL Receptor Aryl Hydrocarbon Receptor NOD-like Receptor (NLR) GABA Receptor P2X Receptor Liver X Receptor Taste receptor Retinoid Receptor MT Receptor Imidazoline Receptor TAM Receptor Discoidin Domain Receptor (DDR) Ephrin Receptor Trk receptor Progesterone Receptor S1P Receptor LPL Receptor

8380

Compounds

579

Natural Products

4866

Recombinant Proteins

Libraries

Cat No.	Product Name	Synonyms	Targets
T4031	S1p receptor agonist 1	S1p-receptor-agonist-1	S1P Receptor , LPL Receptor
	S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.		S1P Receptor , LPL Receptor
T38287	C3a Receptor Agonist	C3a receptor agonist 1,Complement 3a Receptor Agonist	Complement System
	C3a Receptor Agonist (C3a receptor agonist 1) binds the G protein-coupled C3a receptors (C3aRs) in the immune system complement pathway. Activation of C3aR prevents neutrophils from being mobilized in a model of intestin...		Complement System
T37792	A2A receptor antagonist 1	CPI-444 analog,A2A receptor antagonist 1	Adenosine Receptor
	A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.		Adenosine Receptor
T60075	Dopamine D2 receptor agonist-2	Dopamine D2 Receptor	Dopamine Receptor
	Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.		Dopamine Receptor
TP1422	Interleukin (IL)-6 Receptor		Others
	Interleukin (IL)-6 Receptor is a peptide.		Others
T5829	H4 Receptor antagonist 1		Histamine Receptor
	H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.		Histamine Receptor
T3177	Orexin 2 Receptor Agonist	OX2R	OX Receptor
	Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.		OX Receptor
T9244	σ1 Receptor antagonist-1		Sigma receptor
	σ1 Receptor antagonist-1 is a selective sigma 1 receptor antagonist.		Sigma receptor
T10058	A2B receptor antagonist 1		Adenosine Receptor
	A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.		Adenosine Receptor
T37734	AMPA receptor modulator-2		GluR
	AMPA receptor modulator-2 (Example 134) is a AMPA receptor modulator, with a pIC50 of 10.1 for TARPγ2 dependent AMPA receptor[1]. pIC50 = -lgIC50. [1]. BERRY CYNTHIA G B (US), et al. AZABENZIMIDAZOLES AND THEIR USE AS AM...		GluR
T13736	Interferon receptor inducer-1		IFNAR
	Interferon receptor inducer-1 Used in the treatment of a disorder in which the induction of interferon is involved. is an interferon (IFN) receptor inducer.		IFNAR
T11349	GABAA receptor agent 1		GABA Receptor
	GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.		GABA Receptor
T11211	EP4 receptor antagonist 1		Prostaglandin Receptor
	EP4 Receptor Antagonist 1 is a highly potent and selective competitive prostanoid EP4 receptor antagonist, effective for cancer immunotherapy. It inhibits both human and mouse EP4 receptors with IC50 values of 6.1 nM and...		Prostaglandin Receptor
T5586	CFMS Receptor Inhibitor II		c-Fms
	cFMS Receptor Inhibitor II is a CSF1R kinase inhibitor		c-Fms
T9247	Vanilloid receptor antagonist 1	4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile	TRP/TRPV Channel
	Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.		TRP/TRPV Channel
T9579L	GLP-1 receptor agonist 9 citrate	GLP-1 receptor agonist 9 citrate (2401892-71-3 Free base)	Glucagon Receptor
	GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.		Glucagon Receptor
T12910	Sigma-1 receptor antagonist 1		Sigma receptor
	Sigma-1 receptor antagonist 1 is an effective and selective antagonist of sigma-1 receptor. Sigma-1 receptor antagonist 1 exhibits antineuropathic pain activity and can be used in the treatment of neuropathic pain studie...		Sigma receptor
T7740	Protease-Activated Receptor-4 diTFA	Protease-Activated Receptor-4 diTFA(245443-52-1(free base))	Protease-activated Receptor
	Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist		Protease-activated Receptor
T12912	Sigma-1 receptor antagonist 3		Sigma receptor , HER
	Sigma-1 receptor antagonist 3 is a potent and selective antagonist of Sigma-1 (σ1) receptor(Ki : 1.14 nM), has the potential for the neuropathic pain.		Sigma receptor , HER
T1824	TGR5 Receptor Agonist		GPCR19
	TGR5 is a potent TGR5(GPCR19) agonist.		GPCR19
T12911	Sigma-1 receptor antagonist 2		Sigma receptor
	Sigma-1 receptor antagonist 2 is a potent and selective antagonist of sigma 1 receptor (σ1 R) (σ1 and σ2 receptor with Kis of 3.88 and 1288 nM , respectively).		Sigma receptor
T14127	Adenosine A1 receptor activator T62		Adenosine Receptor
	Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also reduces hypersensitivity in models of inflammatory and nerve...		Adenosine Receptor
T8848	GPR34 receptor antagonist 2	Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-,gpr34-receptor-antagonist-2	Others
	GPR34 receptor antagonist 2 (Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-) is an anti-inflammatory agent.		Others
TP1704	Galanin Receptor Ligand M35 TFA		Neuropeptide Y Receptor
	Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).		Neuropeptide Y Receptor
T37908	Glucocorticoid receptor agonist-1		Glucocorticoid Receptor
	Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].		Glucocorticoid Receptor
T15249	Estrogen receptor modulator 1		Estrogen Receptor/ERR
	Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.4...		Estrogen Receptor/ERR
T4521	Edg-2 receptor inhibitor 1	SAR-100842	LPA Receptor
	Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).		LPA Receptor
T10307	AMPA receptor modulator-1		iGluR
	AMPA receptor modulator-1 can be activated by glutamate, thereby modulating ion channels.		iGluR
T21620	Adenosine receptor antagonist 4		Adenosine Receptor
	Adenosine receptor antagonist 4 is an adenosine receptor antagonist.		Adenosine Receptor
T21723L	Epidermal Growth Factor Receptor Peptide Acetate	Epidermal Growth Factor Receptor Peptide Acetate(96249-43-3 Free base)	Others
	Epidermal Growth Factor Receptor Peptide Acetate (Epidermal Growth Factor Receptor Peptide Acetate(96249-43-3 Free base)) exists on the cell surface and is activated by the binding of its specific ligands.EGFR belongs t...		Others
T10499	H3 receptor-MO-1		Histamine Receptor
	H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.		Histamine Receptor
T22466	Adenosine receptor A1 antagonist 5		cAMP
	Adenosine receptor A1 antagonist 5 acts as an adenosine antagonist, is an oxypurine, acts as an insecticide and pest control agent, and has an inhibitory effect on elevated blood pressure.		cAMP
T15785	LPA1 receptor antagonist 1	LPA1 R antagonist 1	LPA Receptor
	LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a selective and potent lysophosphatidic acid (LPA1) receptor antagonist (IC50 : 25 nM) for the study of idiopathic pulmonary fibrosis.		LPA Receptor
T9157	GP130 receptor agonist-1	N-(4-Fluorophenyl)-4-phenyl-2-thiazolami	Interleukin
	GP130 receptor agonist-1 (N-(4-Fluorophenyl)-4-phenyl-2-thiazolami) is a potent, brain-penetrant and orally active GP130 receptor agonist.		Interleukin
T9579	GLP-1 receptor agonist 9		Glucagon Receptor
	1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.		Glucagon Receptor
T12404	CCK-A receptor inhibitor 1		cholecystokinin
	CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the study of diseases related to the digestive system.		cholecystokinin
T11137	(E)-GABAB receptor antagonist 1		GABA Receptor
	(E)-GABAB receptor antagonist 1 is a trans-GABAB receptor antagonist 1. (E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM. GABAB receptor antagonist 1 is ...		GABA Receptor
T7674	Thrombin Receptor Activator for Peptide		Protease-activated Receptor
	Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of coronary heart disease (CHD).		Protease-activated Receptor
T12247	NOT Receptor Modulator 1	2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol	Others
	NOT Receptor Modulator 1 (2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol) is a modulator of nuclear receptor NOT.		Others
T11077	Dopamine D2 receptor antagonist-1		Others
	Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.		Others
T60087	CFMS Receptor Inhibitor IV	5-cyano-N-(2,5-di(piperidin-1-yl)phenyl)furan-2-carboxamide	c-Fms
	cFMS Receptor Inhibitor IV is an inhibitor of c-Fms tyrosine kinase.		c-Fms
T67915	Succinate/succinate receptor antagonist 1		Others
	Succinate/succinate receptor antagonist 1 is a potent succinate receptor antagonist. Succinate/succinate receptor antagonist 1 interrupts succinate signals in gingival tissue and inhibits the activation of SucnRl Antagon...		Others
T77508	A2B receptor antagonist 2 hydrochloride
	A2B receptor antagonist 2 hydrochloride is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T7513	Protease-Activated Receptor-2, amide	SLIGKV-NH2	Protease-activated Receptor
	Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)		Protease-activated Receptor
T78646	Estrogen receptor antagonist 8		Estrogen Receptor/ERR
	Estrogen Receptor Antagonist 8 exhibits potent antagonistic activity against the estrogen receptor (ER), demonstrating effective anti-uterotrophic potential in vivo, with an EC50 value of 4.160 μM.		Estrogen Receptor/ERR
T22009	CB2 receptor agonist 2	ZINC72105556,4-Quinolone-3-Carboxamide Furan CB2 Agonist	Cannabinoid Receptor
	CB2 receptor agonist 2 (ZINC72105556) is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.		Cannabinoid Receptor
T38836L	Protease-Activated Receptor-1, PAR-1 Agonist acetate		Protease-activated Receptor
	Protease-Activated Receptor-1, PAR-1 Agonist acetate is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 Agonist acetate corresponds to PAR1 tethered ligand and whi...		Protease-activated Receptor
T4312	GPR120 Agonist 2	GPR120 receptor agonist	GPR
	GPR120 Agonist 2 is a potent and selective GPR120 receptor agonist.		GPR
T61068	AMPA receptor antagonist-2		iGluR
	AMPA receptor antagonist-2 is an AMPA receptor antagonist.		iGluR
T67946	EP2 receptor antagonist-2		Prostaglandin Receptor
	EP2 receptor antagonist-2 (CID891729) is a compound that not only serves as an antagonist to the EP2 receptor, blocking its activation by PGE2, but also reduces lactate dehydrogenase (LDH) release triggered by N-methyl-D...		Prostaglandin Receptor

Compounds

S1p receptor agonist 1

T4031

Synonym: S1p-receptor-agonist-1

Target: S1P Receptor, LPL Receptor

C3a Receptor Agonist

T38287

Synonym: C3a receptor agonist 1,Complement 3a Receptor Agonist

Target: Complement System

A2A receptor antagonist 1

T37792

Synonym: CPI-444 analog,A2A receptor antagonist 1

Target: Adenosine Receptor

Dopamine D2 receptor agonist-2

T60075

Synonym: Dopamine D2 Receptor

Target: Dopamine Receptor

Interleukin (IL)-6 Receptor

TP1422

Synonym:

Target: Others

H4 Receptor antagonist 1

T5829

Synonym:

Target: Histamine Receptor

Orexin 2 Receptor Agonist

T3177

Synonym: OX2R

Target: OX Receptor

σ1 Receptor antagonist-1

T9244

Synonym:

Target: Sigma receptor

A2B receptor antagonist 1

T10058

Synonym:

Target: Adenosine Receptor

AMPA receptor modulator-2

T37734

Synonym:

Target: GluR

Interferon receptor inducer-1

T13736

Synonym:

Target: IFNAR

GABAA receptor agent 1

T11349

Synonym:

Target: GABA Receptor

EP4 receptor antagonist 1

T11211

Synonym:

Target: Prostaglandin Receptor

cFMS Receptor Inhibitor II

T5586

Synonym:

Target: c-Fms

Vanilloid receptor antagonist 1

T9247

Synonym: 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile

Target: TRP/TRPV Channel

GLP-1 receptor agonist 9 citrate

T9579L

Synonym: GLP-1 receptor agonist 9 citrate (2401892-71-3 Free base)

Target: Glucagon Receptor

Sigma-1 receptor antagonist 1

T12910

Synonym:

Target: Sigma receptor

Protease-Activated Receptor-4 diTFA

T7740

Synonym: Protease-Activated Receptor-4 diTFA(245443-52-1(free base))

Target: Protease-activated Receptor

Sigma-1 receptor antagonist 3

T12912

Synonym:

Target: Sigma receptor, HER

TGR5 Receptor Agonist

T1824

Synonym:

Target: GPCR19

Sigma-1 receptor antagonist 2

T12911

Synonym:

Target: Sigma receptor

Adenosine A1 receptor activator T62

T14127

Synonym:

Target: Adenosine Receptor

GPR34 receptor antagonist 2

T8848

Synonym: Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-,gpr34-receptor-antagonist-2

Target: Others

Galanin Receptor Ligand M35 TFA

TP1704

Synonym:

Target: Neuropeptide Y Receptor

Glucocorticoid receptor agonist-1

T37908

Synonym:

Target: Glucocorticoid Receptor

Estrogen receptor modulator 1

T15249

Synonym:

Target: Estrogen Receptor/ERR

Edg-2 receptor inhibitor 1

T4521

Synonym: SAR-100842

Target: LPA Receptor

AMPA receptor modulator-1

T10307

Synonym:

Target: iGluR

Adenosine receptor antagonist 4

T21620

Synonym:

Target: Adenosine Receptor

Epidermal Growth Factor Receptor Peptide Acetate

T21723L

Synonym: Epidermal Growth Factor Receptor Peptide Acetate(96249-43-3 Free base)

Target: Histamine Receptor

Adenosine receptor A1 antagonist 5

T22466

Synonym:

Target: cAMP

LPA1 receptor antagonist 1

T15785

Synonym: LPA1 R antagonist 1

Target: LPA Receptor

GP130 receptor agonist-1

T9157

Synonym: N-(4-Fluorophenyl)-4-phenyl-2-thiazolami

Target: Interleukin

GLP-1 receptor agonist 9

T9579

Synonym:

Target: Glucagon Receptor

CCK-A receptor inhibitor 1

T12404

Synonym:

Target: cholecystokinin

(E)-GABAB receptor antagonist 1

T11137

Synonym:

Target: GABA Receptor

Thrombin Receptor Activator for Peptide

T7674

Synonym:

Target: Protease-activated Receptor

NOT Receptor Modulator 1

T12247

Synonym: 2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol

Target: Others

Dopamine D2 receptor antagonist-1

T11077

Synonym:

Target: Others

cFMS Receptor Inhibitor IV

T60087

Synonym: 5-cyano-N-(2,5-di(piperidin-1-yl)phenyl)furan-2-carboxamide

Target: c-Fms

Succinate/succinate receptor antagonist 1

T67915

Synonym:

Target: Others

A2B receptor antagonist 2 hydrochloride

T77508

Synonym:

Target:

Protease-Activated Receptor-2, amide

T7513

Synonym: SLIGKV-NH2

Target: Protease-activated Receptor

Estrogen receptor antagonist 8

T78646

Synonym:

Target: Estrogen Receptor/ERR

CB2 receptor agonist 2

T22009

Synonym: ZINC72105556,4-Quinolone-3-Carboxamide Furan CB2 Agonist

Target: Cannabinoid Receptor

Protease-Activated Receptor-1, PAR-1 Agonist acetate

T38836L

Synonym:

Target: Protease-activated Receptor

GPR120 Agonist 2

T4312

Synonym: GPR120 receptor agonist

Target: GPR

AMPA receptor antagonist-2

T61068

Synonym:

Target: iGluR

EP2 receptor antagonist-2

T67946

Synonym:

Target: Prostaglandin Receptor

Cat No.	Product Name	Synonyms	Targets
TN1217	2'-O-Methylisoliquiritigenin		Dopamine Receptor , 5-HT Receptor , GABA Receptor
	2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-regulates 5-HT, NE, DA and GABA pathways, but does not put a ...		Dopamine Receptor , 5-HT Receptor , GABA Receptor
TN1465	Cannabigerol		NOS , 5-HT Receptor , ROS
	Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also binds to the CB2 receptor; it can relieve interocular pressur...		NOS , 5-HT Receptor , ROS
T5754	Kavain		NF-κB , GABA Receptor
	Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of transcriptional factors such as NF-kB and LITAF.		NF-κB , GABA Receptor
TQ0119	Cirsimaritin		GABA Receptor
	Cirsimaritin exhibits antibacterial, anti-inflammation, anti-tumor, antioxidant properties and renal protection. Cirsimaritin binds weakly to the benzodiazepine site on GABAA receptors.		GABA Receptor
TN1015	Meranzin		Adrenergic Receptor , Immunology/Inflammation related
	Meranzin, a bioactive compound derived from the Traditional Chinese Medicine (TCM) Chaihu-Shugan-San (CSS) and isolated from Murraya exotica L. leaves, targets the alpha 2-adrenoceptor and engages the AMPA-ERK1/2–BDNF si...		Adrenergic Receptor , Immunology/Inflammation related
TN2247	Swertisin		Adenosine Receptor
	Swertisin, a novel herbal biomolecule, shows a strong antihyperglycemic action. Swertisin is an adenosine A1 receptor antagonist, is known to have antidiabetic, anti-inflammatory and antioxidant effects.		Adenosine Receptor
T3782	Jujuboside A		transporter , GABA Receptor
	Jujuboside A is a glycoside extracted from Semen Ziziphi Spinosae, having neurophysiological inhibitory effects, used as a potential therapeutic agent for the treatment of Alzheimer s disease.		transporter , GABA Receptor
T0076	Paliperidone	9-hydroxyrisperidone	Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
	Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the primary active metabolite of the older...
T7557	Guvacine hydrochloride		GABA Receptor
	Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)		GABA Receptor
T2815	Puerarin	Kakonein	5-HT Receptor
	Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.		5-HT Receptor
T8036	6-Methylflavone		GABA Receptor
	6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.		GABA Receptor
T6S2099	Geraniin		Antioxidant , TNF
	1. Geraniin has a protective effect against OVX-induced rat osteoporosis. 2. Geraniin has cytotoxic activity towards cancer cells in vitro and in vivo. 3. Geraniin exerts inhibitory effects on osteoclast differentiation ...		Antioxidant , TNF
TN1023	Miltirone		P450 , GABA Receptor
	Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.		P450 , GABA Receptor
T9113	Myristicin	Myristicine	IL Receptor , Anti-infection , BCL , P450 , PARP , 5-HT Receptor , Caspase , GABA Receptor , NO Synthase
	Myristicin (Myristicine) is a natural product found in spices and umbelliferous plants. Myristicin has anti-cholinergic, Antibacterial, and hepatoprotective effects, it also has anti-inflammatory properties related with ...
T6S0630	Hypaconitine		P450 , TNF
	Hypaconitine, an active and highly toxic constituent derived from Aconitum species, has anti-inflammatory activity, is widely used to treat rheumatism.		P450 , TNF
T0525	Flopropione	Phloropropiophenone	5-HT Receptor , Transferase
	Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.		5-HT Receptor , Transferase
T3S2100	(-)-Securinine	Securinine	GABA Receptor
	(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.		GABA Receptor
T6648	Rotundine	Gindarine,L-Tetrahydropalmatine,Caseanine,(-)-Tetrahydropalmatine	Dopamine Receptor , 5-HT Receptor
	Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.		Dopamine Receptor , 5-HT Receptor
T2720	Ginsenoside Rc	Panaxoside Rc	Others , TNF , GABA Receptor , Interleukin
	Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.		Others , TNF , GABA Receptor , Interleukin
T6S0654	Isocorynoxeine	7-Isocorynoxeine	5-HT Receptor
	1. Isocorynoxeine (7-Isocorynoxeine) shows the effects of lowering blood pressure, vasodilatation, and protection against ischemia-induced neuronal damage. 2. Isocorynoxeine exhibits a significant neuroprotective effect ...		5-HT Receptor
T3369	Nuciferine	(-)-Nuciferine,VLT 049,Sanjoinine E	Dopamine Receptor , 5-HT Receptor
	Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera. It has a profile of action associated with dopamine receptor blockade.		Dopamine Receptor , 5-HT Receptor
T5799	Arecaidine hydrochloride		Others
	Arecaidine hydrochloride may have carcinogenesis.		Others
T1681	Aminophylline	Phyllocontin	PDE , Adenosine Receptor
	Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.		PDE , Adenosine Receptor
T4S1637	Gamma-Mangostin	Normangostin	Others , 5-HT Receptor
	1. gamma-Mangostin (Normangostin) as a preventive agent of the metabolic syndrome. 2. Gamma-Mangostin has free radical scavenging activity, and antiproliferative and apoptotic activity in HepG2 cells. 3. Gamma-Mangostin ...		Others , 5-HT Receptor
TN2268	Tetrahydromagnolol		Cannabinoid Receptor , GPR , GABA Receptor
	Tetrahydromagnolol can activate cannabinoid (CB) receptors.		Cannabinoid Receptor , GPR , GABA Receptor
TN1032	Geissoschizine methyl ether		5-HT Receptor
	Geissoschizine methyl ether, a major indole alkaloid found in Uncaria hook, is a major active component of Yokukansan with psychotropic effects. Geissoschizine methyl ether is a potent serotonin A receptor agonist and ca...		5-HT Receptor
T6519	Gramine	NSC 16892,Donaxine	Adiponectin receptor , Reverse Transcriptase , Adrenergic Receptor
	Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4.2 μM for AdipoR2 and AdipoR1, respectively. Gramine is als...
T6662	Scopine	6,7-Epoxytropine	Adrenergic Receptor
	Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.		Adrenergic Receptor
T5S1882	Songorine	Napellonine,Zongorine,Bullatine G	Others , GABA Receptor
	Songorine (Napellonine) shows favorable anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.		Others , GABA Receptor
T4S0217	HOMOPLANTAGININ		TNF , NF-κB
	Homoplantaginin is a flavonoid from a traditional Chinese medicine Salvia plebeia,it has a protective and therapeutic effect on hepatocyte injury and shows potent inhibitory activities against influenza.		TNF , NF-κB
T8268	6,2'-Dihydroxyflavone		GABA Receptor
	6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.		GABA Receptor
TN1052	Lindleyin		Estrogen Receptor/ERR , Estrogen/progestogen Receptor
	Lindleyin is a novel phytoestrogen and might trigger many of the biological responses evoked by the physiological estrogens.		Estrogen Receptor/ERR , Estrogen/progestogen Receptor
T2850	Bicuculline	(+)-Bicuculline,d-Bicuculline	GABA Receptor
	Bicuculline ((+)-Bicuculline) is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and has been isolated from Dicentra cucullaria, Adlumia fungos...		GABA Receptor
T1711	Harmine	Telepathine	MAO , 5-HT Receptor , DYRK
	Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.		MAO , 5-HT Receptor , DYRK
T19931	Gentisein	NSC 329491,NSC329491,NSC-329491	Serotonin Transporter
	Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency with an IC50 value of 4.7 µM[1][2].		Serotonin Transporter
T2979	DL-Menthol	Hexahydrothymol,(±)-Menthol	GABA Receptor , AChE
	DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis. (–)-Menthol is more common than (+)-menthol in nature and exhibits analgesic, anti...		GABA Receptor , AChE
T0892	Diphylline	Dyphylline,Diprophylline	PDE , Adenosine Receptor
	Diphylline (Diprophylline) is a xanthine derivative. Diphylline exerts bronchodilator effects and to a lesser extent vasodilator and diuretic properties. Diphylline probably acts as a competitive inhibitor of phosphodies...		PDE , Adenosine Receptor
TN1849	Kuwanon H		GPR , Bombesin Receptor
	Kuwanon H, and possibly kuwanon G also, are specific antagonists for the gastrin-releasing peptide (GRP) -preferring receptor and can be useful for studying the physiological and pathological role of GRP.		GPR , Bombesin Receptor
T1396	Bemegride	Bemegrid,3-Ethyl-3-methylglutarimide,Agipnon	GABA Receptor
	Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.		GABA Receptor
T6S1256	Ruscogenin		NOS , NF-κB , NOD-like Receptor (NLR)
	1. Ruscogenin has anti-inflammatory activity, suppressed zymosan A-evoked peritoneal total leukocyte migration in mice in a dose-dependent manner, 2. Ruscogenin inhibited adhesion of leukocytes to a human umbilical vein ...		NOS , NF-κB , NOD-like Receptor (NLR)
T5S0543	Isocurcumenol		Apoptosis , Estrogen Receptor/ERR , Reductase
	1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).		Apoptosis , Estrogen Receptor/ERR , Reductase
T2749	Ginkgolide A	BN-52020	GABA Receptor , Endogenous Metabolite
	Ginkgolide A (BN-52020) is a highly active PAF antagonist cage molecule that is isolated from the leaves of the Ginkgo biloba tree. Shows potential in a wide variety of inflammatory and immunological disorders.		GABA Receptor , Endogenous Metabolite
T6S0627	Mesaconitine		TNF
	1. Mesaconitine has antiinflammatory activity. 2. Mesaconitine has antinociceptive activity through cyclic AMP and stimulation of the central β-adrenergic system.		TNF
T3698	Alpha-Asarone	α-Asarone,trans-Asarone	P450 , GABA Receptor , HMG-CoA Reductase
	alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.		P450 , GABA Receptor , HMG-CoA Reductase
TN2865	(E)-3,4,5-Trimethoxycinnamic acid	O-Methylsinapic acid,3,4,5-Trimethoxy-trans-cinnamic acid,3,4,5-Trimethoxyphenylacrylic acid	Others
	(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.		Others
T2879	Fisetin		TNF , Sirtuin , PPAR
	Fisetin is a natural flavonol extracted from Rhus succedanea L that is structurally and functionally related to kaempferol, can modulate sirtuins,with antioxidant, anticancer, neuroprotection effects.		TNF , Sirtuin , PPAR
T5940	Proxyphylline	7-(2-Hydroxypropyl)theophylline	PDE , Adenosine Receptor
	Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor. Proxyphylline acts as a cardiac stimulant, vasodilator and bronchodilator.		PDE , Adenosine Receptor
T13768	(+)-Medicarpin		Estrogen/progestogen Receptor
	(+)-Medicarpin, a pterocarpan, is an isoflavonoid compound derived from multiple medicinal plant species such as Sophora japonica, Zollernia paraensis, Platymiscium yucatamun, Machaerium aristulatum, and Platymiscium flo...		Estrogen/progestogen Receptor
T6S1597	Mulberroside A		TNF , Tyrosinase , Interleukin
	1. Mulberroside has nephroprotective, hypoglycemic, and antidiabetic effects. 2. Mulberroside A is a glycosylated stilbene of oxyresveratrol; thus, the deglycosylation of Mulberroside A resulted in enhanced inhibition of...		TNF , Tyrosinase , Interleukin
TN2437	Serotonin	5-hydroxytryptamine,5-HT	Others , 5-HT Receptor , Endogenous Metabolite , Transferase
	Serotonin (5-hydroxytryptamine) is a natural product from animals
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Natural Products

2'-O-Methylisoliquiritigenin

TN1217

Synonym:

Target: Dopamine Receptor, 5-HT Receptor, GABA Receptor

Cannabigerol

TN1465

Synonym:

Target: NOS, 5-HT Receptor, ROS

Kavain

T5754

Synonym:

Target: NF-κB, GABA Receptor

Cirsimaritin

TQ0119

Synonym:

Target: GABA Receptor

Meranzin

TN1015

Synonym:

Target: Adrenergic Receptor, Immunology/Inflammation related

Swertisin

TN2247

Synonym:

Target: Adenosine Receptor

Jujuboside A

T3782

Synonym:

Target: transporter, GABA Receptor

Paliperidone

T0076

Synonym: 9-hydroxyrisperidone

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor

Guvacine hydrochloride

T7557

Synonym:

Target: GABA Receptor

Puerarin

T2815

Synonym: Kakonein

Target: 5-HT Receptor

6-Methylflavone

T8036

Synonym:

Target: GABA Receptor

Geraniin

T6S2099

Synonym:

Target: Antioxidant, TNF

Miltirone

TN1023

Synonym:

Target: P450, GABA Receptor

Myristicin

T9113

Synonym: Myristicine

Target: IL Receptor, Anti-infection, BCL, P450, PARP, 5-HT Receptor, Caspase, GABA Receptor, NO Synthase

Synonym: Phloropropiophenone

Target: 5-HT Receptor, Transferase

(-)-Securinine

T3S2100

Synonym: Securinine

Target: GABA Receptor

Rotundine

T6648

Synonym: Gindarine,L-Tetrahydropalmatine,Caseanine,(-)-Tetrahydropalmatine

Target: Dopamine Receptor, 5-HT Receptor

Ginsenoside Rc

T2720

Synonym: Panaxoside Rc

Target: Others, TNF, GABA Receptor, Interleukin

Isocorynoxeine

T6S0654

Synonym: 7-Isocorynoxeine

Target: 5-HT Receptor

Nuciferine

T3369

Synonym: (-)-Nuciferine,VLT 049,Sanjoinine E

Target: Dopamine Receptor, 5-HT Receptor

Arecaidine hydrochloride

Synonym: Phyllocontin

Target: PDE, Adenosine Receptor

gamma-Mangostin

T4S1637

Synonym: Normangostin

Target: Others, 5-HT Receptor

Tetrahydromagnolol

TN2268

Synonym:

Target: Cannabinoid Receptor, GPR, GABA Receptor

Geissoschizine methyl ether

TN1032

Synonym:

Target: 5-HT Receptor

Gramine

T6519

Synonym: NSC 16892,Donaxine

Target: Adiponectin receptor, Reverse Transcriptase, Adrenergic Receptor

Scopine

T6662

Synonym: 6,7-Epoxytropine

Target: Adrenergic Receptor

Songorine

T5S1882

Synonym: Napellonine,Zongorine,Bullatine G

Target: Others, GABA Receptor

6,2'-Dihydroxyflavone

T8268

Synonym:

Target: GABA Receptor

Lindleyin

TN1052

Synonym:

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor

Bicuculline

T2850

Synonym: (+)-Bicuculline,d-Bicuculline

Target: GABA Receptor

Harmine

T1711

Synonym: Telepathine

Target: MAO, 5-HT Receptor, DYRK

Gentisein

T19931

Synonym: NSC 329491,NSC329491,NSC-329491

Target: Serotonin Transporter

DL-Menthol

T2979

Synonym: Hexahydrothymol,(±)-Menthol

Target: GABA Receptor, AChE

Diphylline

T0892

Synonym: Dyphylline,Diprophylline

Target: PDE, Adenosine Receptor

Kuwanon H

TN1849

Synonym:

Target: GPR, Bombesin Receptor

Bemegride

T1396

Synonym: Bemegrid,3-Ethyl-3-methylglutarimide,Agipnon

Target: GABA Receptor

Ruscogenin

T6S1256

Synonym:

Target: NOS, NF-κB, NOD-like Receptor (NLR)

Isocurcumenol

T5S0543

Synonym:

Target: Apoptosis, Estrogen Receptor/ERR, Reductase

Ginkgolide A

T2749

Synonym: BN-52020

Target: GABA Receptor, Endogenous Metabolite

Synonym: α-Asarone,trans-Asarone

Target: P450, GABA Receptor, HMG-CoA Reductase

(E)-3,4,5-Trimethoxycinnamic acid

TN2865

Synonym: O-Methylsinapic acid,3,4,5-Trimethoxy-trans-cinnamic acid,3,4,5-Trimethoxyphenylacrylic acid

Target: TNF, Sirtuin, PPAR

Proxyphylline

T5940

Synonym: 7-(2-Hydroxypropyl)theophylline

Target: PDE, Adenosine Receptor

(+)-Medicarpin

T13768

Synonym:

Target: Estrogen/progestogen Receptor

Mulberroside A

T6S1597

Synonym:

Target: TNF, Tyrosinase, Interleukin

Serotonin

TN2437

Synonym: 5-hydroxytryptamine,5-HT

Target: Others, 5-HT Receptor, Endogenous Metabolite, Transferase

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Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPY-03739	Transferrin Receptor/TFRC Protein, Cynomolgus, Rhesus, Recombinant (His)	Cynomolgus,Rhesus	HEK293
	Transferrin receptor protein 1, also known as transferrin receptor, Trfr, p9, CD71 and TFRC, is a single-pass type II membrane protein that belongs to the peptidase M28 family and M28B subfamily. TFRC / CD71 is a membran...
TMPY-01053	Prolactin Receptor Protein, Human, Recombinant (His)	Human	HEK293
	Prolactin receptor (PRLR) is a single-pass transmembrane receptor belonging to the type I cytokine receptor superfamily, and contains two fibronectin type-III domains. All class 1 ligands activate their respective recept...
TMPY-01146	Insulin Receptor Protein, Human, Recombinant (long isoform, His)	Human	HEK293
	INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to the protein kinase superfamily and exists as a tetramer consisting of two alpha subunits and two beta...
TMPY-01725	Leptin Receptor Protein, Human, Recombinant (His)	Human	HEK293
	Leptin Receptor or CD295 belongs to the gp130 family of cytokine receptors that are known to stimulate gene transcription via activation of cytosolic STAT proteins. This protein is a receptor for leptin (an adipocyte-spe...
TMPY-01873	Transferrin Receptor/TFRC Protein, Human, Recombinant (His)	Human	HEK293
	Transferrin receptor protein 1, also known as transferrin receptor, Trfr, p9, CD71 and TFRC, is a single-pass type II membrane protein that belongs to the peptidase M28 family and M28B subfamily. TFRC / CD71 is a membran...
TMPY-05096	Transferrin Receptor/TFRC Protein, Human, Recombinant (hFc)	Human	HEK293
	Transferrin receptor protein 1, also known as transferrin receptor, Trfr, p9, CD71 and TFRC, is a single-pass type II membrane protein that belongs to the peptidase M28 family and M28B subfamily. TFRC / CD71 is a membran...
TMPY-02294	Transferrin Receptor/TFRC Protein, Mouse, Recombinant (His)	Mouse	HEK293
	Transferrin receptor protein 1, also known as transferrin receptor, Trfr, p9, CD71 and TFRC, is a single-pass type II membrane protein that belongs to the peptidase M28 family and M28B subfamily. TFRC / CD71 is a membran...
TMPY-06661	Transferrin Receptor/TFRC Protein, Rat, Recombinant (His)	Rat	HEK293
	Transferrin receptor protein 1, also known as transferrin receptor, Trfr, p9, CD71 and TFRC, is a single-pass type II membrane protein that belongs to the peptidase M28 family and M28B subfamily. TFRC / CD71 is a membran...
TMPY-02434	Prolactin Receptor Protein, Rat, Recombinant (His)	Rat	HEK293
	Prolactin receptor (PRLR) is a single-pass transmembrane receptor belonging to the type I cytokine receptor superfamily, and contains two fibronectin type-III domains. All class 1 ligands activate their respective recept...
TMPK-01200	Nogo Receptor/RTN4R Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293
	NOGO Receptor 1 (RTN4R) regulates axonal growth, as well as axon regeneration after injury. The gene maps to the 22q11.2 schizophrenia susceptibility locus and is thus a strong functional and positional candidate gene.RT...
TMPY-03144	Nogo Receptor/RTN4R Protein, Human, Recombinant (His)	Human	HEK293
	Reticulon 4 receptor (RTN4R), also known as Nogo-66 Receptor (NgR), is a glycosylphosphoinositol (GPI)-anchored protein that belongs to the Nogo recptor family including three members. Mouse RTN4R cDNA contains 1 LRP (Le...
TMPY-04395	Insulin Receptor Protein, Human, Recombinant (His & GST)	Human	Baculovirus-Insect Cells
	INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to the protein kinase superfamily and exists as a tetramer consisting of two alpha subunits and two beta...
TMPY-01163	Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His)	Mouse	HEK293
	Reticulon 4 receptor (RTN4R), also known as Nogo-66 Receptor (NgR), is a glycosylphosphoinositol (GPI)-anchored protein that belongs to the Nogo recptor family including three members. Mouse RTN4R cDNA contains 1 LRP (Le...
TMPY-02984	Prolactin Receptor Protein, Mouse, Recombinant (His)	Mouse	HEK293
	Prolactin receptor (PRLR) is a single-pass transmembrane receptor belonging to the type I cytokine receptor superfamily, and contains two fibronectin type-III domains. All class 1 ligands activate their respective recept...
TMPY-01056	Nogo Receptor/RTN4R Protein, Human, Recombinant (His & hFc)	Human	HEK293
	Reticulon 4 receptor (RTN4R), also known as Nogo-66 Receptor (NgR), is a glycosylphosphoinositol (GPI)-anchored protein that belongs to the Nogo recptor family including three members. Mouse RTN4R cDNA contains 1 LRP (Le...
TMPY-01149	Insulin Receptor Protein, Human, Recombinant (short isoform, His)	Human	HEK293
	INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to the protein kinase superfamily and exists as a tetramer consisting of two alpha subunits and two beta...
TMPY-05025	Thrombin Receptor Protein, Human, Recombinant (His)	Human	HEK293

TMPH-00932	Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO)	Human	E. coli
	Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli.
TMPY-05283	Insulin Receptor Protein, Human, Recombinant (long isoform, His), Biotinylated	Human	HEK293
	INSR (Insulin receptor), also known as CD22, is a transmembrane receptor that is activated by insulin. INSR belongs to the protein kinase superfamily and exists as a tetramer consisting of two alpha subunits and two beta...
TMPY-02987	Vitamin D Receptor/VDR Protein, Mouse, Recombinant (His)	Mouse	Baculovirus-Insect Cells
	VDR (vitamin D (1,25- dihydroxyvitamin D3) receptor), also known as NR1I1, belongs to the NR1I family, NR1 subfamily. It is composed of three domains: a modulating N-terminal domain, a DNA-binding domain and a C-terminal...
TMPY-00874	Leptin Receptor Protein, Human, Recombinant (His & hFc)	Human	HEK293
	Leptin Receptor or CD295 belongs to the gp130 family of cytokine receptors that are known to stimulate gene transcription via activation of cytosolic STAT proteins. This protein is a receptor for leptin (an adipocyte-spe...
TMPY-01566	Prolactin Receptor Protein, Mouse, Recombinant (His & hFc)	Mouse	HEK293
	Prolactin receptor (PRLR) is a single-pass transmembrane receptor belonging to the type I cytokine receptor superfamily, and contains two fibronectin type-III domains. All class 1 ligands activate their respective recept...
TMPY-01221	Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His & hFc)	Mouse	HEK293
	Reticulon 4 receptor (RTN4R), also known as Nogo-66 Receptor (NgR), is a glycosylphosphoinositol (GPI)-anchored protein that belongs to the Nogo recptor family including three members. Mouse RTN4R cDNA contains 1 LRP (Le...
TMPY-02706	Vitamin D Receptor/VDR Protein, Human, Recombinant (His)	Human	Baculovirus-Insect Cells
	VDR (vitamin D (1,25- dihydroxyvitamin D3) receptor), also known as NR1I1, belongs to the NR1I family, NR1 subfamily. It is composed of three domains: a modulating N-terminal domain, a DNA-binding domain and a C-terminal...
TMPY-00317	Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc)	Human	HEK293

TMPY-00085	Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc)	Human	HEK293

TMPY-01612	CD155/PVR Protein, Rhesus, Recombinant (His)	Rhesus	HEK293
	CD155, commonly known as PVR (poliovirus receptor) and Necl-5 (nectin-like molecule-5), is a type I transmembrane single-span glycoprotein, and belongs to the nectins and nectin-like (Necl) subfamily. CD155 was originall...
TMPY-05617	Transferrin Receptor/TFRC Protein, Human, Recombinant (His), Biotinylated	Human	HEK293
	Transferrin receptor protein 1, also known as transferrin receptor, Trfr, p9, CD71 and TFRC, is a single-pass type II membrane protein that belongs to the peptidase M28 family and M28B subfamily. TFRC / CD71 is a membran...
TMPY-00181	Endothelin B Receptor Protein, Human, Recombinant (His)	Human	HEK293
	The hypermethylation of EDNRB gene was remarkably related to infiltration and metastasis of gastric cancer and may attribute to the tumor progression. EDNRB is a new candidate tumor suppressor gene which is often down-re...
TMPY-03860	Endothelin B Receptor Protein, Human, Recombinant (mFc)	Human	HEK293
	The hypermethylation of EDNRB gene was remarkably related to infiltration and metastasis of gastric cancer and may attribute to the tumor progression. EDNRB is a new candidate tumor suppressor gene which is often down-re...
TMPY-02648	PACAP receptor/ADCYAP1R1 Protein, Human, Recombinant (hFc)	Human	HEK293
	Pituitary adenylate cyclase activating polypeptide (PACAP, Adcyap1) activation of PAC1 receptors ( Adcyap1r1) significantly increases excitability of guinea pig cardiac neurons. This modulation of excitability is mediate...
TMPJ-00378	Transferrin Receptor/TFRC Protein, Human, Recombinant (aa 101-760, His)	Human	Human Cells
	Transferrin receptor protein 1 (TFRC) belongs to the peptidase M28 family that is synthesized as a 172 amino acid (aa). TFRC regulated by cellular iron levels through binding of the iron regulatory proteins, IRP1 and IRP...
TMPY-05274	IL-23R Protein, Human, Recombinant (His)	Human	HEK293
	IL23R, also known as the IL23 receptor, belongs to the type I cytokine receptor family, Type 2 subfamily. It contains 2 fibronectin type-III domains and is expressed by monocytes, Th1, Th0, NK, and dendritic cells. Isofo...
TMPY-05102	CD122/IL2RB Protein, Rat, Recombinant (His)	Rat	HEK293
	Interleukin-2 receptor (IL-2R) also known as High-affinity IL-2 receptor subunit beta, IL-2 receptor subunit beta, and IL-2RB, is involved in T cell-mediated immune responses. CD122/IL-2RB is present in 3 forms concernin...
TMPY-04717	CD122/IL2RB Protein, Rhesus, Recombinant (His)	Rhesus	HEK293
	Interleukin-2 receptor (IL-2R) also known as High-affinity IL-2 receptor subunit beta, IL-2 receptor subunit beta, and IL-2RB, is involved in T cell-mediated immune responses. CD122/IL-2RB is present in 3 forms concernin...
TMPY-02934	IL-2RG Protein, Rat, Recombinant (His)	Rat	HEK293
	The common gamma chain (γc) (or CD132), also known as interleukin-2 receptor subunit gamma or IL2RG, is a member of the type I cytokine receptor family expressed on most lymphocyte (white blood cell) populations, and its...
TMPY-04649	ROR1 Protein, Human, Recombinant (His)	Human	HEK293

TMPJ-00994	LTBR Protein, Mouse, Recombinant (hFc)	Mouse	Human Cells
	It is a single-pass type I membrane protein and contains 4 TNFR-Cys repeats. The protein is a member of the tumor necrosis factor (TNF) family of receptors. It is expressed on the surface of most cell types, including ce...
TMPY-00418	IL-21R Protein, Mouse, Recombinant (His)	Mouse	HEK293
	Interleukin-21 receptor, also known as IL-21 receptor, IL-21R, Novel interleukin receptor, IL21R, and NILR, is a single-pass type I membrane protein that belongs to the type I cytokine receptor family and Type 4 subfamil...
TMPY-02824	IL-18R alpha Protein, Rat, Recombinant (hFc)	Rat	HEK293
	Interleukin-18 receptor 1 (IL18R1) also known as CD218 antigen-like family member A, CDw218a, IL1 receptor-related protein, and CD218a, is an interleukin receptor of the immunoglobulin superfamily. IL18R1 is found expres...
TMPY-06022	FOLR1 Protein, Cynomolgus, Rhesus, Recombinant (His)	Cynomolgus,Rhesus	HEK293
	The protein encoded by FOLR1 gene is a member of the folate receptor family. Members of this gene family bind folic acid and its reduced derivatives, and transport 5-methyltetrahydrofolate into cells. This gene product i...
TMPJ-00154	IL-15RA Protein, Mouse, Recombinant (hFc)（Human Cells）	Mouse	Human Cells
	Mouse interleukin-15 receptor subunit alpha, also known as Il15ra, is a high-affinity receptor for interleukin-15. Il15ra associates as a heterotrimer with the IL-2 receptor beta and gamma subunits (Common gamma chain, o...
TMPY-02335	OSMR Protein, Mouse, Recombinant (His)	Mouse	HEK293
	Oncostatin-M specific receptor subunit beta also known as the oncostatin M receptor (OSMR) and Interleukin-31 receptor subunit beta (IL-31RB), is one of the receptor proteins for oncostatin M. OSMR is a member of the typ...
TMPY-04818	EGFR Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293
	As a member of the epidermal growth factor receptor (EGFR) family, EGFR protein is type I transmembrane glycoprotein that binds a subset of EGF family ligands including EGF, amphiregulin, TGF-α, betacellulin, etc. EGFR p...
TMPY-03951	IL-18R alpha Protein, Cynomolgus, Recombinant (hFc)	Cynomolgus	HEK293
	Interleukin-18 receptor 1 (IL18R1) also known as CD218 antigen-like family member A, CDw218a, IL1 receptor-related protein, and CD218a, is an interleukin receptor of the immunoglobulin superfamily. IL18R1 is found expres...
TMPY-01883	EPOR Protein, Human, Recombinant (His)	Human	HEK293
	Erythropoietin (EPO) is the major glycoprotein hormone regulator of mammalian erythropoiesis, and is produced by kidney and liver in an oxygen-dependent manner. The biological effects of EPO are mediated by the specific ...
TMPY-02286	Influenza A H1N1 (A/Puerto Rico/8/34/Mount Sinai) Matrix protein 1/M1 Protein (His)	H1N1	E. coli
	The Influenza virus matrix protein 1 (M1) is a matrix protein of the influenza virus. M1 protein has been shown to play a crucial role in virus replication, assembly, and budding. It forms a coat inside the viral envelop...
TMPY-05090	CD25/IL2R alpha Protein, Rat, Recombinant (His)	Rat	Baculovirus-Insect Cells
	CD25 (alpha-chain of the IL-2 receptor, or IL2RA), is a type I transmembrane glycoprotein with a signal peptide, an extracellular region, a transmembrane region, and a cytoplasmic domain. IL2RA is expressed on activated ...
TMPY-05644	CD25/IL2R alpha Protein, Rhesus, Recombinant (His & Avi), Biotinylated	Rhesus	HEK293
	CD25 (alpha-chain of the IL-2 receptor, or IL2RA), is a type I transmembrane glycoprotein with a signal peptide, an extracellular region, a transmembrane region, and a cytoplasmic domain. IL2RA is expressed on activated ...
TMPY-03644	CD25/IL2R alpha Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293
	CD25 (alpha-chain of the IL-2 receptor, or IL2RA), is a type I transmembrane glycoprotein with a signal peptide, an extracellular region, a transmembrane region, and a cytoplasmic domain. IL2RA is expressed on activated ...
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Transferrin Receptor/TFRC Protein, Cynomolgus, Rhesus, Recombinant (His)

TMPY-03739

Species: Cynomolgus,Rhesus

Expression System: HEK293

Prolactin Receptor Protein, Human, Recombinant (His)

TMPY-01053

Species: Human

Expression System: HEK293

Insulin Receptor Protein, Human, Recombinant (long isoform, His)

TMPY-01146

Species: Human

Expression System: HEK293

Leptin Receptor Protein, Human, Recombinant (His)

TMPY-01725

Species: Human

Expression System: HEK293

Transferrin Receptor/TFRC Protein, Human, Recombinant (His)

TMPY-01873

Species: Human

Expression System: HEK293

Transferrin Receptor/TFRC Protein, Human, Recombinant (hFc)

TMPY-05096

Species: Human

Expression System: HEK293

Transferrin Receptor/TFRC Protein, Mouse, Recombinant (His)

TMPY-02294

Species: Mouse

Expression System: HEK293

Transferrin Receptor/TFRC Protein, Rat, Recombinant (His)

TMPY-06661

Species: Rat

Expression System: HEK293

Prolactin Receptor Protein, Rat, Recombinant (His)

TMPY-02434

Species: Rat

Expression System: HEK293

Nogo Receptor/RTN4R Protein, Cynomolgus, Recombinant (His)

TMPK-01200

Species: Cynomolgus

Expression System: HEK293

Nogo Receptor/RTN4R Protein, Human, Recombinant (His)

TMPY-03144

Species: Human

Expression System: HEK293

Insulin Receptor Protein, Human, Recombinant (His & GST)

TMPY-04395

Species: Human

Expression System: Baculovirus-Insect Cells

Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His)

TMPY-01163

Species: Mouse

Expression System: HEK293

Prolactin Receptor Protein, Mouse, Recombinant (His)

TMPY-02984

Species: Mouse

Expression System: HEK293

Nogo Receptor/RTN4R Protein, Human, Recombinant (His & hFc)

TMPY-01056

Species: Human

Expression System: HEK293

Insulin Receptor Protein, Human, Recombinant (short isoform, His)

TMPY-01149

Species: Human

Expression System: HEK293

Thrombin Receptor Protein, Human, Recombinant (His)

TMPY-05025

Species: Human

Expression System: HEK293

Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO)

TMPH-00932

Species: Human

Expression System: E. coli

Insulin Receptor Protein, Human, Recombinant (long isoform, His), Biotinylated

TMPY-05283

Species: Human

Expression System: HEK293

Vitamin D Receptor/VDR Protein, Mouse, Recombinant (His)

TMPY-02987

Species: Mouse

Expression System: Baculovirus-Insect Cells

Leptin Receptor Protein, Human, Recombinant (His & hFc)

TMPY-00874

Species: Human

Expression System: HEK293

Prolactin Receptor Protein, Mouse, Recombinant (His & hFc)

TMPY-01566

Species: Mouse

Expression System: HEK293

Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His & hFc)

TMPY-01221

Species: Mouse

Expression System: HEK293

Vitamin D Receptor/VDR Protein, Human, Recombinant (His)

TMPY-02706

Species: Human

Expression System: Baculovirus-Insect Cells

Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc)

TMPY-00317

Species: Human

Expression System: HEK293

Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc)

TMPY-00085

Species: Human

Expression System: HEK293

CD155/PVR Protein, Rhesus, Recombinant (His)

TMPY-01612

Species: Rhesus

Expression System: HEK293

Transferrin Receptor/TFRC Protein, Human, Recombinant (His), Biotinylated

TMPY-05617

Species: Human

Expression System: HEK293

Endothelin B Receptor Protein, Human, Recombinant (His)

TMPY-00181

Species: Human

Expression System: HEK293

Endothelin B Receptor Protein, Human, Recombinant (mFc)

TMPY-03860

Species: Human

Expression System: HEK293

PACAP receptor/ADCYAP1R1 Protein, Human, Recombinant (hFc)

TMPY-02648

Species: Human

Expression System: HEK293

Transferrin Receptor/TFRC Protein, Human, Recombinant (aa 101-760, His)

TMPJ-00378

Species: Human

Expression System: Human Cells

IL-23R Protein, Human, Recombinant (His)

TMPY-05274

Species: Human

Expression System: HEK293

CD122/IL2RB Protein, Rat, Recombinant (His)

TMPY-05102

Species: Rat

Expression System: HEK293

CD122/IL2RB Protein, Rhesus, Recombinant (His)

TMPY-04717

Species: Rhesus

Expression System: HEK293

IL-2RG Protein, Rat, Recombinant (His)

TMPY-02934

Species: Rat

Expression System: HEK293

ROR1 Protein, Human, Recombinant (His)

TMPY-04649

Species: Human

Expression System: HEK293

LTBR Protein, Mouse, Recombinant (hFc)

TMPJ-00994

Species: Mouse

Expression System: Human Cells

IL-21R Protein, Mouse, Recombinant (His)

TMPY-00418

Species: Mouse

Expression System: HEK293

IL-18R alpha Protein, Rat, Recombinant (hFc)

TMPY-02824

Species: Rat

Expression System: HEK293

FOLR1 Protein, Cynomolgus, Rhesus, Recombinant (His)

TMPY-06022

Species: Cynomolgus,Rhesus

Expression System: HEK293

IL-15RA Protein, Mouse, Recombinant (hFc)（Human Cells）

TMPJ-00154

Species: Mouse

Expression System: Human Cells

OSMR Protein, Mouse, Recombinant (His)

TMPY-02335

Species: Mouse

Expression System: HEK293

EGFR Protein, Cynomolgus, Recombinant (His)

TMPY-04818

Species: Cynomolgus

Expression System: HEK293

IL-18R alpha Protein, Cynomolgus, Recombinant (hFc)

TMPY-03951

Species: Cynomolgus

Expression System: HEK293

EPOR Protein, Human, Recombinant (His)

TMPY-01883

Species: Human

Expression System: HEK293

Influenza A H1N1 (A/Puerto Rico/8/34/Mount Sinai) Matrix protein 1/M1 Protein (His)

TMPY-02286

Species: H1N1

Expression System: E. coli

CD25/IL2R alpha Protein, Rat, Recombinant (His)

TMPY-05090

Species: Rat

Expression System: Baculovirus-Insect Cells

CD25/IL2R alpha Protein, Rhesus, Recombinant (His & Avi), Biotinylated

TMPY-05644

Species: Rhesus

Expression System: HEK293

CD25/IL2R alpha Protein, Cynomolgus, Recombinant (His)

TMPY-03644

Species: Cynomolgus

Expression System: HEK293

--------- More ---------

Cat No.	Product Name
L1510	Nuclear Receptor Compound Library	546 compounds
	A unique collection of 546 nuclear receptor signaling targeted compounds for high throughput and high content screening;
L2610	Neurotransmitter Receptor Compound Library	1513 compounds
	A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
L2700	Adrenergic Receptor-Targeted Compound Library	219 compounds
	A unique collection of 219 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification;
L2800	Serotonin Receptor-Targeted Compound Library	275 compounds
	A unique collection of 275 compounds targeting serotonin receptors for high throughput screening and high content screening;
L3300	Histamine & Melatonin Receptor-Targeted Compound Library	155 compounds
	A unique collection of 155 compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS) for new drugs;
L7600	Chemokine Inhibitor Library	59 compounds
	A unique collection of 59 chemokines or chemokine receptors targeted compounds for high throughput and high content screening;
L2195	Anti-Prostate Cancer Compound Library	2096 compounds
	2096 compounds associated with prostate cancer that can be used for high-throughput and high-content screening.
L2191	Anti-Breast Cancer Compound Library	1965 compounds
	A unique collection of 1965 compounds with anti-breast cancer therapeutic activity or targeting breast cancer’s major signaling pathways, can be used for anti-breast cancer drug discovery and mechanism study；
L2193	Anti-Liver Cancer Compound Library	1816 compounds
	1816 species of compounds related to liver cancer that can be used in anti-liver cancer drug development and pharmacological studies.
L9830	Anti-Parkinson's Disease Compound Library	908 compounds
	A unique collection of 908 compounds with anti-PD activities or acting on main drug targets of PD can be used for HTS and HCS.
L1400	MAPK Inhibitor Library	367 compounds
	A unique collection of 367 compounds targeting MAPK signaling for drug discovery in MAPK related diseases;
L7110	Anti-Hypertension Compound Library	719 compounds
	719 hypertension-related small molecules for high-throughput and high-content screening.
L4100	TGF-beta/Smad Compound Library	185 compounds
	A unique collection of 185 TGF-beta/Smad signaling targeted compounds for high throughput and high content screening;
L9000	Apoptosis Compound Library	1796 compounds
	A unique collection of 1796 apoptosis-related compounds for apoptosis research, research in tumorigenesis, and anti-cancer drug screening;
L9840	Anti-Alzheimer's Disease Compound Library	1040 compounds
	A unique collection of 1040 compounds with anti-AD activities or acting on main drug targets of AD can be used for HTS and HCS.