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Search Result

Search Results for " faah "

Targets

FAAH Cannabinoid Receptor FAAH

70

Compounds

6

Natural Products

1

Recombinant Proteins

1

Libraries

Cat No. Product Name Synonyms Targets
T67745 CB2R/FAAH modulator-2 Cannabinoid Receptor , FAAH
CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-2 acts as a CB2R agonist and FAAH inhibitor, the Ki values are 10.8 and 152.9 nM for CB2R and CB1R, respectively, an...
T11256 FAAH inhibitor 1 Benzothiazole analog 3 FAAH
FAAH inhibitor 1 (Benzothiazole analog 3) is an effective FAAH inhibitor with an IC50 of 18 nM.
T67896 CB2R/FAAH modulator-1 Cannabinoid Receptor , FAAH
CB2R/FAAH modulator-1, a cannabinoid type 2 receptor (CB2R) agonist, is also a fatty acid amide hydrolase (FAAH) inhibitor (IC50=4 μM) that reduces the production of pro-inflammatory and anti-inflammatory cytokines and i...
T15268 FAAH-IN-2 O-Desmorpholinopropyl Gefitinib FAAH , Autophagy
FAAH-IN-2 (O-Desmorpholinopropyl Gefitinib) is a potent inhibitor of FAAH(fatty acid amide hydrolase).
T67747 CB2R/FAAH modulator-3 Cannabinoid Receptor , FAAH
CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-3 acts as a CB2R agonist and FAAH inhibitor, the Ki values are 20.1 and 67.6 nM for CB2R and CB1R, respectively, and the ...
T63536 Dual FAAH/sEH-IN-1 FAAH , Epoxide Hydrolase
Dual FAAH/sEH-IN-1 is a dual inhibitor of sEH (soluble epoxide hydrolase) (IC50: 9.6 nM) and FAAH (fatty acid amide hydrolase) (IC50: 7 nM) with high affinity and anti-inflammatory activity.
T6714 URB-597 KDS-4103,FAAH Inhibitor II Mitophagy , FAAH , Autophagy
URB-597 (FAAH Inhibitor II) is an effective, orally bioavailable FAAH inhibitor (IC50: 4.6 nM), and no effect on other cannabinoid-related targets.
T11255 FAAH-IN-1 FAAH
FAAH-IN-1 is a fatty acid amide hydrolase (FAAH) inhibitor, with IC50s of 145 nM and 650 nM for rat and human FAAH, respectively.
T82421 FAAH/cPLA2α-IN-1 Phospholipase
FAAH/cPLA2α-IN-1 is a compound that simultaneously inhibits both FAAH and cPLA2α, demonstrating potent activity with half-maximal inhibitory concentrations (IC50s) of 32 nM for FAAH and 47 nM for cPLA2α [1].
T62558 FAAH-IN-5
FAAH-IN-5 (Compound 7) is a relatively selective, irreversible inhibitor of fatty acid amide hydrolase (FAAH) (IC50: 10.5 nM). FAAH-IN-5 has low PAMPA (parallel artificial membrane permeability assay) permeability.
T73302 FAAH-IN-7
FAAH-IN-7, a potent and reversible inhibitor of fatty acid amide hydrolase (FAAH), demonstrates significant neuroprotective effects, particularly by mitigating oxidative stress in 1321N1 astrocytes. With an IC50 value of...
T62671 FAAH/MAGL-IN-3
FAAH/MAGL-IN-3 (Compound 10) is an irreversible dual inhibitor of fatty acid amide hydrolase (FAAH) and monoacylglycerol lipase (MAGL) that acts on FAAH (IC50: 179 nM) and MAGL (IC50: 759 nM). FAAH/MAGL-IN-3 showed littl...
T61198 FAAH/MAGL-IN-1
FAAH/MAGL-IN-1, also known as compound SIH 3, is a highly effective inhibitor of FAAH (fatty acid amide hydrolase) and MAGL (monoacylglycerol lipase). It exhibits IC50 values of 31 nM and 29 nM against FAAH and MAGL, res...
T26311 URB532 URB-532,FAAH Inhibitor I,FAAH Inhibitor-I,URB 532
URB532 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor.
T61707 FAAH/MAGL-IN-2
FAAH/MAGL-IN-2, a potent and reversible inhibitor of FAAH and MAGL, demonstrates oral activity and the ability to cross the blood-brain barrier. It exhibits IC50 values of 11 nM for FAAH and 36 nM for MAGL (Ki values of ...
T8927 WWL 154 WWL-154 FAAH
WWL 154 is an serine hydrolase (SH) and fatty acid amide hydrolase FAAH-4 inhibitor.
T28353 PDP-EA FAAH
PDP-EA is an activator of fatty acid amide hydrolase(FAAH) and enhances the amidohydrolase activity of FAAH.
T9967 MAGL-IN-5 Lipid
MAGL-IN-5 is a non-selective lipase inhibitor.
T3215 JNJ-42165279 JNJ42165279 FAAH , Autophagy
JNJ-42165279 covalently inactivates the FAAH enzyme but is highly selective with regard to other enzymes, ion channels, transporters, and receptors. JNJ-42165279 (10 μM) exhibits high selectivity against a panel of 50 re...
T8646 URB937 FAAH
URB937 is an inhibitor of FAAH and increases anandamide levels(IC50 : 26.8 nM).
T4323 PF-04457845 PF04457845,PF 04457845 FAAH , Autophagy
PF-04457845 is a greatly and effctive FAAH inhibitor, and for hFAAH(IC50=7.2±0.63 nM) and rFAAH(IC50=7.4±0.62 nM).
T7688 4-Nonylphenylboronic acid FAAH
4-Nonylphenylboronic acid is a inhibitor of FAAH.
T15802 LY2183240 FAAH , Autophagy
LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM).
T2338 JZL195 FAAH , Lipase , Autophagy
JZL195 is a selective and efficacious dual FAAH/MAGL inhibitor.
T3354 BIA 10-2474 BIA10-2474 FAAH , Autophagy
BIA 10-2474 is a long-acting reversible inhibitor of fatty acid amide hydrolase (FAAH) that increases levels of the neurotransmitter anandamide in the central nervous system and in peripheral tissues (that is, the rest o...
T6043 PF-3845 FAAH , Autophagy
PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.
T1325 Carprofen Ridamyl,Imadyl,Rimadyl FAAH , COX , Autophagy
Carprofen (Ridamyl) is a propionic acid derivate and nonsteroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic, and antipyretic activities.
T9687 MAGL-IN-4 His121 ARG57 Lipase
MAGL-IN-4 (His121 ARG57) is one of the monoacylglycerol lipase (MAGL) inhibitors in central nervous system-related diseases.
T12306 OMDM-5 Cannabinoid Receptor , Endogenous Metabolite , TRP/TRPV Channel
OMDM-5 is a selective anandamide cellular uptake (ACU)inhibitor(Ki of 4.8 μM).
T2684 JNJ-1661010 JNJ1661010,Takeda-25,JNJ 1661010 FAAH
JNJ-1661010 (Takeda-25) is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows >100-fold selectivity for FAAH-1 than FAAH-2.
T9374 AA38-3 1-Piperidinecarboxylic acid, 4-nitrophenyl ester FAAH , Lipase , MAGL
AA38-3 (1-Piperidinecarboxylic acid, 4-nitrophenyl ester) inhibites three SHs (ABHD6, ABHD11, and FAAH)
T12302 OMDM-1 (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide Endogenous Metabolite
OMDM-1 ((Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide) is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor with a Ki of 2.4 μM.
T16515 PF 750 PF-750,UNII-7756CPP14K,ZINC27647189 FAAH
PF 750 (ZINC27647189) is a selective and covalent inhibitor of FAAH. PF 750 shows IC50s varying from 16.2 to 595 nM in different incubation times.
T27703 JZP-361 JZP361,JZP 361 Lipase
JZP-361 is a specific MAGL inhibitor with IC50s of 46 nM, 7.24 μM, and 1.79 μM for human recombinant MAGL, human recombinant FAAH, and human hABHD6. JZP-361 displays anti-histaminergic activities. JZP-361 can be used in ...
T23119 Palmitoylisopropylamide FAAH
Palmitoylisopropylamide is a selective FAAH inhibitor that inhibits [H]-AEA uptake and cell proliferation at low concentrations.
T77594 VU534 FAAH , Phospholipase , Epoxide Hydrolase
VU534 is a NAPE-PLD agonist with an EC50 of 0.30 μM.VU534 is a dual inhibitor of FAAH and sEH, with an IC50 of 1.2 μM for sEH.VU534 is used in diseases related to cardiometabolism.
T28076 MM-433593 FAAH
MM-433593 is a selective fatty acid amide hydrolase (FAAH-1) inhibitor for the treatment of pain, inflammation, and other disorders.
T68492 AM 374 HDSF,Hexadecanesulfonyl fluoride FAAH
AM 374 (HDSF), a fatty acid amide hydrolase (FAAH) inhibitor, demonstrates the capacity to inhibit amidase activity, boasting an IC50 value of 13 nM. This compound is potentially applicable in neurological disease resear...
T5357 ARN272 ARN 272 FAAH
ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).
T6554 JZL 184 JZL184 Lipase
JZL 184 is a potent and selective inhibitor of MAGL with IC50 of 8 nM and 4 μM for inhibition of MAGL and FAAH in mouse brain membranes respectively.
T15635 JZP-430 Lipase , MAGL
JZP-430 is an effective, highly selective, irreversible inhibitor of α/β-hydrolase domain 6 (ABHD6) (IC50: 44 nM). It also shows ~230-fold selectivity over fatty acid amide hydrolase (FAAH) and lysosomal acid lipase (LAL...
T4052 KML29 Lipase
KML29 is highly selective and effective monoacylglycerol lipase (MAGL) inhibitor. It has effective inhibition of human/mouse/rat MAGL (IC50: 5.9/15/43 nM). It has not inhibitory for FAAH (IC50 > 50 μM). It also effective...
T12826 SA57 FAAH
SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).
T23432 TC-F 2 Others
TC-F 2 is a FAAH inhibitor.
T12827 SA72 Others
SA72 is a highly selective inhibitor of fatty acid amide hydrolase (FAAH).
T68407 URB-694
URB-694 is a fatty acid amide hydrolase (FAAH) inhibitor.
T33953 PF3845yne PF-3845yne,PF 3845yne
PF3845yne is an alkyne analogue of PF-3845 maintaining high potency for FAAH.
T23415 TAK 21d Others
Potent FAAH inhibitor
T29045 UCM710
UCM710 is a dual inhibitor of α/β hydrolase domain 6 (ABHD6) and fatty acid amide hydrolase (FAAH).
T22582 Arachidonyl serotonin Others
Dual FAAH inhibitor/TRPV1 antagonist

Compounds

CB2R/FAAH modulator-2
T67745
Synonym:
Target: Cannabinoid Receptor, FAAH
FAAH inhibitor 1
T11256
Synonym: Benzothiazole analog 3
Target: FAAH
CB2R/FAAH modulator-1
T67896
Synonym:
Target: Cannabinoid Receptor, FAAH
FAAH-IN-2
T15268
Synonym: O-Desmorpholinopropyl Gefitinib
Target: FAAH, Autophagy
CB2R/FAAH modulator-3
T67747
Synonym:
Target: Cannabinoid Receptor, FAAH
Dual FAAH/sEH-IN-1
T63536
Synonym:
Target: FAAH, Epoxide Hydrolase
URB-597
T6714
Synonym: KDS-4103,FAAH Inhibitor II
Target: Mitophagy, FAAH, Autophagy
FAAH-IN-1
T11255
Synonym:
Target: FAAH
FAAH/cPLA2α-IN-1
T82421
Synonym:
Target: Phospholipase
FAAH-IN-5
T62558
Synonym:
Target:
FAAH-IN-7
T73302
Synonym:
Target:
FAAH/MAGL-IN-3
T62671
Synonym:
Target:
FAAH/MAGL-IN-1
T61198
Synonym:
Target:
URB532
T26311
Synonym: URB-532,FAAH Inhibitor I,FAAH Inhibitor-I,URB 532
Target:
FAAH/MAGL-IN-2
T61707
Synonym:
Target:
WWL 154
T8927
Synonym: WWL-154
Target: FAAH
PDP-EA
T28353
Synonym:
Target: FAAH
MAGL-IN-5
T9967
Synonym:
Target: Lipid
JNJ-42165279
T3215
Synonym: JNJ42165279
Target: FAAH, Autophagy
URB937
T8646
Synonym:
Target: FAAH
PF-04457845
T4323
Synonym: PF04457845,PF 04457845
Target: FAAH, Autophagy
4-Nonylphenylboronic acid
T7688
Synonym:
Target: FAAH
LY2183240
T15802
Synonym:
Target: FAAH, Autophagy
JZL195
T2338
Synonym:
Target: FAAH, Lipase, Autophagy
BIA 10-2474
T3354
Synonym: BIA10-2474
Target: FAAH, Autophagy
PF-3845
T6043
Synonym:
Target: FAAH, Autophagy
Carprofen
T1325
Synonym: Ridamyl,Imadyl,Rimadyl
Target: FAAH, COX, Autophagy
MAGL-IN-4
T9687
Synonym: His121 ARG57
Target: Lipase
OMDM-5
T12306
Synonym:
Target: Cannabinoid Receptor, Endogenous Metabolite, TRP/TRPV Channel
JNJ-1661010
T2684
Synonym: JNJ1661010,Takeda-25,JNJ 1661010
Target: FAAH
AA38-3
T9374
Synonym: 1-Piperidinecarboxylic acid, 4-nitrophenyl ester
Target: FAAH, Lipase, MAGL
OMDM-1
T12302
Synonym: (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide
Target: Endogenous Metabolite
PF 750
T16515
Synonym: PF-750,UNII-7756CPP14K,ZINC27647189
Target: FAAH
JZP-361
T27703
Synonym: JZP361,JZP 361
Target: Lipase
Palmitoylisopropylamide
T23119
Synonym:
Target: FAAH
VU534
T77594
Synonym:
Target: FAAH, Phospholipase, Epoxide Hydrolase
MM-433593
T28076
Synonym:
Target: FAAH
AM 374
T68492
Synonym: HDSF,Hexadecanesulfonyl fluoride
Target: FAAH
ARN272
T5357
Synonym: ARN 272
Target: FAAH
JZL 184
T6554
Synonym: JZL184
Target: Lipase
JZP-430
T15635
Synonym:
Target: Lipase, MAGL
KML29
T4052
Synonym:
Target: Lipase
SA57
T12826
Synonym:
Target: FAAH
TC-F 2
T23432
Synonym:
Target: Others
SA72
T12827
Synonym:
Target: Others
URB-694
T68407
Synonym:
Target:
PF3845yne
T33953
Synonym: PF-3845yne,PF 3845yne
Target:
TAK 21d
T23415
Synonym:
Target: Others
UCM710
T29045
Synonym:
Target:
Arachidonyl serotonin
T22582
Synonym:
Target: Others
1 2
Cat No. Product Name Synonyms Targets
T2859 Biochanin A 4-Methylgenistein,Olmelin EGFR , FAAH , Autophagy
Biochanin A (4-Methylgenistein) is an isoflavone derivative isolated from red clover Trifolium pratense with anticarcinogenic properties. Biochanin A is a naturally occurring fatty acid amide hydrolase (FAAH) inhibitor.
TN1965 N-​Benzyllinolenamide N-Benzyllinolenamide FAAH , Autophagy
N-Benzyllinolenamide is a natural product. It is an inhibitor of fatty acid amide hydrolase (FAAH, IC50 of 41.8 μM).
T12139 N-(3-Methoxybenzyl)Palmitamide FAAH
N-(3-Methoxybenzyl)Palmitamide is a promising FAAH inhibitor, treatment of pain, inflammation and CNS degenerative disorders.
T3S2105 N-Benzylpalmitamide Macamide 1,N-Benzylhexadecanamide Others , FAAH , Autophagy
N-Benzylpalmitamide (Macamide 1) inhibits fatty acid amide hydrolase (FAAH) in a time-dependent manner and could potentially offer a good alternative for the treatment of pain, inflammation and CNS degenerative disorders...
T4859 1-Monomyristin rac-Glycerol 1-myristate,Glyceryl myristate,Monomyristin,2,3-Dihydroxypropyl tetradecanoate Others , FAAH , Endogenous Metabolite , Antibacterial , Autophagy , Antifungal
1-Monomyristin (2,3-Dihydroxypropyl tetradecanoate) , a 1-monoglyceride of myristic acid, has antibacterial activity against several Gram-positive bacterial strains. 1-Myristoyl-rac-glycerol is used in colloidal chemistr...
TMA1122 N-Feruloylserotonin (E/Z)-Moschamine,Moschamine Antioxidant
N-Feruloylserotonin ((E/Z)-Moschamine) is a selective FAAH inhibitor that inhibits [H]-AEA uptake and cell proliferation at low concentrations.

Natural Products

Biochanin A
T2859
Synonym: 4-Methylgenistein,Olmelin
Target: EGFR, FAAH, Autophagy
N-​Benzyllinolenamide
TN1965
Synonym: N-Benzyllinolenamide
Target: FAAH, Autophagy
N-(3-Methoxybenzyl)Palmitamide
T12139
Synonym:
Target: FAAH
N-Benzylpalmitamide
T3S2105
Synonym: Macamide 1,N-Benzylhexadecanamide
Target: Others, FAAH, Autophagy
1-Monomyristin
T4859
Synonym: rac-Glycerol 1-myristate,Glyceryl myristate,Monomyristin,2,3-Dihydroxypropyl tetradecanoate
Target: Others, FAAH, Endogenous Metabolite, Antibacterial, Autophagy, Antifungal
N-Feruloylserotonin
TMA1122
Synonym: (E/Z)-Moschamine,Moschamine
Target: Antioxidant

Recombinant Proteins

Species：
Human (1)
Expression System：
in vitro E. coli expression system (1)
Tag：
N-terminal 10xHis-tagged (1)
Cat No. Product Name Species Expression System
TMPH-01325 FAAH2 Protein, Human, Recombinant (His) Human in vitro E. coli expression system
Catalyzes the hydrolysis of endogenous amidated lipids like the sleep-inducing lipid oleamide ((9Z)-octadecenamide), the endocannabinoid anandamide (N-(5Z,8Z,11Z,14Z-eicosatetraenoyl)-ethanolamine), as well as other fatt...
Cat No. Product Name
L2510 Lipid Metabolism Compound Library

496 compounds
A unique collection of 496 compounds targeting lipid metabolism, can be used for high-throughput screening (HTS) and high-content screening (HCS).

Libraries

Lipid Metabolism Compound Library
L2510
Compounds: 496
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