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Adenosine Receptor

T0070 Pentoxifylline Pentoxifylline modulates immunologic activity by stimulating cytokine production. Pentoxifylline is a methylxanthine derivative that inhibits phosphodiesterase ...
T1368 Methyl protocatechuate Thermographic recording material with improved image tone.
T1825 Reversine Reversine, a small synthetic purine analogue (2,6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).
T2205 Theophylline-7-acetic acid Theophylline-7-acetic acid, a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist. It is combined with diphenhydramine in th...
T2373 Vipadenant Vipadenant(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).
T2671 Regadenoson Regadenoson is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadenoson select...
T6115 Fostamatinib Fostamatinib(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.
T6441 CGS 21680 HCl CGS 21680 HCl( IC50=22 nM),an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.
T6552 Istradefylline Istradefylline(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails. It has been used in trials s...
T6979 SCH58261 SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.
T7021 ZM241385 ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.
T4265 AZD4635 AZD4635 is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).
T4290 Preladenant Preladenant is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine receptors.
T6884 2-Cl-IB-MECA 2-Cl-IB-MECA is an adenosine A3 receptor agonist.
T7183 CPI-444 CPI-444 is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.
T7188 Piclidenoson Piclidenoson, a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.
T7320 Tozadenant Tozadenant is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)
T7509 PD 117519 PD 117519 is an agonist of adenosine receptor
T7683 Adenosine amine congener Adenosine amine congener (ADAC) is an agonist of selective A1 adenosine receptor,.
TQ0125 Capadenoson Capadenoson is a selective adenosine-A1 receptor agonist.
TQ0136 GR 79236 GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
T8312 Derenofylline Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)
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