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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5751 | Tigogenin | Others | |
Tigogenin is one of steroidal sapogenins which is widely used for synthesizing steroid drugs. It might have protective effect on bone and be helpful in preventing the development of osteoporosis. | |||
T3672 | Nomilin | MAPK | |
Nomilin is naturally occurring triterpenoids, have immunomodulatory activity. | |||
T3836 | Eudesmin | MAPK , S6 Kinase | |
Eudesmin shows antiinflammatory, neuritogenic, anticonvulsant and sedative effects, the mechanism of eudesmin may be related to up-regulation of GABAA and GAD65 expressions, and anti-apoptosis of neuron the in brain.50 m... | |||
TN6772 | Malabaricone C | Others | |
Malabaricone C is a bioactive chemical. | |||
T12580 | PTUPB | COX , Epoxide Hydrolase | |
PTUPB is a potent and dual inhibitor of sEH and COX-2 enzymes(IC50 of 0.9 nM and 1.26 μM, respectively). | |||
T9491 | Pyraclostrobin | Antibacterial , Antifungal | |
Pyraclostrobin is one of the most heavily used fungicides that inhibits mitochondrial complex III of fungal and mammalian cells. | |||
T5583 | Turanose | D-(+)-Turanose | Endogenous Metabolite |
D(+)-Turanose (D-(+)-Turanose) is a naturally occuring compound. It is a reducing disaccharide. | |||
T5778 | 5,7-DIMETHOXYFLAVONE | Anti-infection , P450 | |
5,7-DIMETHOXYFLAVONE possessed remarkable leishmanicidal potential. | |||
T22447 | Tri-Salicylic Acid | Others | |
Tri-Salicylic Acid, a product of the thermal decomposition of aspirin, is a compound for proteomics research. | |||
T7482 | 3-chloro-5-hydroxybenzoic Acid | GPR | |
3-chloro-5-hydroxy Benzoic Acid (3-chloro-5-hydroxy BA) is an agonist of GPR81 (EC50 : 16 μM) | |||
T9089 | FTO-IN-1 | UUN44923 | Others |
UUN44923 is a FTO inhibitor. It may be useful for treating diseases assocd. with FTO targets, obesity, metabolic syndrome (MS) , type 2 diabetes (T2D) , Alzheimer's diseases, breast cancers, small- cell lung cancers, a h... | |||
T2057 | BVT 2733 | Dehydrogenase | |
BVT 2733 is a new, non-steroidal, isoform-specific inhibitor of 11β-HSD1. | |||
T7704 | KY-226 | Phosphatase | |
KY-226 is a potent inhibitor of protein tyrosine phosphatase 1B (PTP1B)(IC50: 0.25 μM,) | |||
T4733 | Sucrose | D(+)-Sucrose,D-(+)-Saccharose | Others , Endogenous Metabolite |
Sucrose (D-(+)-Saccharose) is a nonreducing disaccharide composed of glucose and fructose linked via their anomeric carbons. | |||
T11590 | (-)-Hydroxycitric acid | Garcinia acid | ATP Citrate Lyase |
(-)-Hydroxycitric acid (Garcinia acid) (Garcinia acid) is the principal acid of fruit rinds of Garcinia cambogia. It is a potent and competitive inhibitor of ATP citrate lyase. (-)-Hydroxycitric acid suppresses fatty aci... | |||
T15017 | CU-T12-9 | TLR | |
CU-T12-9 is a potent TLR1/2 agonist(EC50 of 52.9 nM in HEK-Blue hTLR2 SEAP assay). It acts by activating the NFkB pathway, upregulating proinflammatory cytokines, and enhancing TLR1 and TLR2 dimerization.CU-T12-9 activat... | |||
T3283 | Cetilistat | ATL-962 | Lipid |
Cetilistat (ATL-962) is a novel inhibitor of pancreatic lipase being developed by Alizyme for the treatment of obesity and associated co-morbidities, including type 2 diabetes. | |||
T7832 | Ibrolipim | NO-1886 | LPL Receptor |
Ibrolipim (NO-1886) attenuates high glucose-induced endothelial dysfunction in cultured human umbilical vein endothelial cells via PI3K/Akt pathway. | |||
T2626 | SBC-115076 | SBC115076 | Others , Serine/threonin kinase |
SBC-115076 is a potent extracellular proprotein convertase subtilisin kexin type 9 (PCSK9) antagonist. | |||
T16074 | Mifobate | SR-202 | PPAR |
Mifobate (SR-202) is a potent and specific antagonist of PPARγ. Mifobate shows antiobesity, antidiabetic and antiatherosclerotic effects[1]. |