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Search Results for " congener "

18

Compounds

Cat No. Product Name Synonyms Targets
T23535L Xanthine amine congener trihydrochloride Xanthine amine congener trihydrochloride (96865-92-8 Free base) Adenosine Receptor
Xanthine amine congener trihydrochloride is a potent adenosine antagonist that reverses the reduction in urine flow, sodium excretion and heart rate produced by the adenosine agonist, N6-cyclohexyladenosine.
T7683 Adenosine amine congener ADAC Adenosine Receptor
Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.
T39387 Xanthine amine congener dihydrochloride XAC dihydrochloride,Xanthine amine congener dihydrochloride
Xanthine amine congener dihydrochloride (XAC dihydrochloride), a potent antagonist for both Adenosine A1 and A2 receptors, exhibits IC50 values of 1.8 nM for A1 and 114 nM for A2 receptors. Additionally, it functions as ...
T23535 Xanthine amine congener Adenosine Receptor
Xanthine amine congener is an Adenosine receptor antagonist.
T62963 Xanthine amine congener hydrochloride
Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice.
T3421 Nordihydrocapsaicin Others
Nordihydrocapsaicin is an analog and congener of capsaicin, belonging to the capsaicinoid class of compounds found in Capsicum chili peppers.
T0797 Cimetidine SKF-92334 Histamine Receptor
Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological actions. It inhibits GASTRIC ACID secretion, as well as PEP...
T1378 Tegafur Fluorafur,FT-207,NSC 148958,FT 207 Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis
Tegafur (FT 207) is a congener of the antimetabolite fluorouracil with antineoplastic activity. Tegafur is a prodrug that is gradually converted to fluorouracil in the liver by the cytochrome P-450 enzyme.
T1591 Ancitabine hydrochloride NSC 145668 HCl,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C Others , DNA/RNA Synthesis , Autophagy
Ancitabine hydrochloride (NSC 145668 HCl) is the hydrochloride salt of a cytarabine congener prodrug with antineoplastic activity. Upon administration, ancitabine is slowly hydrolyzed into cytarabine. Subsequently, cytar...
T21161 Ancitabine
Ancitabine, a congener of cyterabine, is metabolized to cytarabine, thereby maintains a more constant antineoplastic action.
T61409 CXCR4 antagonist 3
CXCR4 antagonist 3 (compound 12a), an effective antagonist of CXCR4, exhibits an IC50 of 11 nM. It is a congener of TIQ15, showcasing exceptional properties such as CXCR4 antagonism, CYP 2D6 inhibition, metabolic stabili...
T72682 Lankacyclinone C
Lankacyclinone C, a congener of lankacidin C devoid of the δ-lactone moiety, exhibits antitumor activity.
T74722 Demethyl bleomycin A2
Demethyl bleomycin A2 is a Bleomycin congener. The DNA cleavage of demethyl bleomycin A2 is insensitive to the presence of 5-Methylcytidine [1] .
T37216 N-Arachidonoyl-L-Alanine
Several different arachidonoyl amino acids, including N-arachidonoyl-L-alanine (NALA), have been isolated and characterized from bovine brain. The glycine congener (NAGly) was further characterized and found to suppress ...
T37731 TPU-0037A
TPU-0037A is an antibiotic and a congener of lydicamycin . It inhibits the growth of Gram-positive bacteria, including methicillin-resistant S. aureus (MRSA), B. subtilis, and M. luteus (MICs = 1.56-12.5 μg/ml), but not ...
T36162 8-iso Prostaglandin F1α 8-iso Prostaglandin F1α
8-iso PGF1α is an isoprostane that was first identified in human semen. It is a member of the isoprostane family, which are eicosanoids of non-cyclooxygenase origin. 8-iso PGF1α is present along with its 19-hydroxy conge...
T38225 N-Arachidonoyl-3-hydroxy-γ-Aminobutyric Acid
Several different arachidonoyl amino acids, including N-arachidonoyl-3-hydroxy-γ-aminobutyric acid (NAG-3H-ABA), have been isolated and characterized from bovine brain. The glycine congener was further characterized and ...
T60728 M1 ligand 1
M1 ligand 1 (compound 3b-b) is a N-desmethyl congener of arecoline derivative that is a muscarinic acetylcholine receptor M1 ligand. M1 ligand 1 is able to be used as PET (positron emission tomography) radiotracer [1].
TargetMol