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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T23535L | Xanthine amine congener trihydrochloride | Xanthine amine congener trihydrochloride (96865-92-8 Free base) | Adenosine Receptor |
Xanthine amine congener trihydrochloride is a potent adenosine antagonist that reverses the reduction in urine flow, sodium excretion and heart rate produced by the adenosine agonist, N6-cyclohexyladenosine. | |||
T7683 | Adenosine amine congener | ADAC | Adenosine Receptor |
Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,. | |||
T39387 | Xanthine amine congener dihydrochloride | XAC dihydrochloride,Xanthine amine congener dihydrochloride | |
Xanthine amine congener dihydrochloride (XAC dihydrochloride), a potent antagonist for both Adenosine A1 and A2 receptors, exhibits IC50 values of 1.8 nM for A1 and 114 nM for A2 receptors. Additionally, it functions as ... | |||
T23535 | Xanthine amine congener | Adenosine Receptor | |
Xanthine amine congener is an Adenosine receptor antagonist. | |||
T62963 | Xanthine amine congener hydrochloride | ||
Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice. | |||
T3421 | Nordihydrocapsaicin | Others | |
Nordihydrocapsaicin is an analog and congener of capsaicin, belonging to the capsaicinoid class of compounds found in Capsicum chili peppers. | |||
T0797 | Cimetidine | SKF-92334 | Histamine Receptor |
Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological actions. It inhibits GASTRIC ACID secretion, as well as PEP... | |||
T1378 | Tegafur | Fluorafur,FT-207,NSC 148958,FT 207 | Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis |
Tegafur (FT 207) is a congener of the antimetabolite fluorouracil with antineoplastic activity. Tegafur is a prodrug that is gradually converted to fluorouracil in the liver by the cytochrome P-450 enzyme. | |||
T1591 | Ancitabine hydrochloride | NSC 145668 HCl,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C | Others , DNA/RNA Synthesis , Autophagy |
Ancitabine hydrochloride (NSC 145668 HCl) is the hydrochloride salt of a cytarabine congener prodrug with antineoplastic activity. Upon administration, ancitabine is slowly hydrolyzed into cytarabine. Subsequently, cytar... | |||
T21161 | Ancitabine | ||
Ancitabine, a congener of cyterabine, is metabolized to cytarabine, thereby maintains a more constant antineoplastic action. | |||
T61409 | CXCR4 antagonist 3 | ||
CXCR4 antagonist 3 (compound 12a), an effective antagonist of CXCR4, exhibits an IC50 of 11 nM. It is a congener of TIQ15, showcasing exceptional properties such as CXCR4 antagonism, CYP 2D6 inhibition, metabolic stabili... | |||
T72682 | Lankacyclinone C | ||
Lankacyclinone C, a congener of lankacidin C devoid of the δ-lactone moiety, exhibits antitumor activity. | |||
T74722 | Demethyl bleomycin A2 | ||
Demethyl bleomycin A2 is a Bleomycin congener. The DNA cleavage of demethyl bleomycin A2 is insensitive to the presence of 5-Methylcytidine [1] . | |||
T37216 | N-Arachidonoyl-L-Alanine | ||
Several different arachidonoyl amino acids, including N-arachidonoyl-L-alanine (NALA), have been isolated and characterized from bovine brain. The glycine congener (NAGly) was further characterized and found to suppress ... | |||
T37731 | TPU-0037A | ||
TPU-0037A is an antibiotic and a congener of lydicamycin . It inhibits the growth of Gram-positive bacteria, including methicillin-resistant S. aureus (MRSA), B. subtilis, and M. luteus (MICs = 1.56-12.5 μg/ml), but not ... | |||
T36162 | 8-iso Prostaglandin F1α | 8-iso Prostaglandin F1α | |
8-iso PGF1α is an isoprostane that was first identified in human semen. It is a member of the isoprostane family, which are eicosanoids of non-cyclooxygenase origin. 8-iso PGF1α is present along with its 19-hydroxy conge... | |||
T38225 | N-Arachidonoyl-3-hydroxy-γ-Aminobutyric Acid | ||
Several different arachidonoyl amino acids, including N-arachidonoyl-3-hydroxy-γ-aminobutyric acid (NAG-3H-ABA), have been isolated and characterized from bovine brain. The glycine congener was further characterized and ... | |||
T60728 | M1 ligand 1 | ||
M1 ligand 1 (compound 3b-b) is a N-desmethyl congener of arecoline derivative that is a muscarinic acetylcholine receptor M1 ligand. M1 ligand 1 is able to be used as PET (positron emission tomography) radiotracer [1]. |