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Viral Proteins •   Coronavirus (CoV) Proteins •   Influenza Proteins Fluorescent Proteins Others

Search Result

Search Results for " activating "

Targets

Protease-activated Receptor

358

Compounds

84

Natural Products

440

Recombinant Proteins

4

Libraries

Cat No. Product Name Synonyms Targets
TP1046L PAR-2 Activating Peptide acetate SLIGRL-NH2 acetate,PAR-2 Activating Peptide acetate(171436-38-7 free base),Protease-Activated Receptor-2 Activating Peptide acetate Protease-activated Receptor
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).
TP2411 Sperm-activating peptide 1
Sperm-activating peptide 1 is a bioactive chemical.
T2503 PAC-1 Procaspase activating compound 1 Apoptosis , Caspase , Autophagy
PAC-1 (Procaspase activating compound 1) has been used in trials studying the treatment of Lymphoma, Melanoma, Solid Tumors, Breast Cancer, and Thoracic Cancers, among others.
TP1046 SLIGRL-NH2 Protease-Activated Receptor-2 Activating Peptide Protease-activated Receptor
SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) is a protease-activated receptor-2 (PAR-2) agonist that induces non-histaminergic pruritus.
T81372 Proteasome-activating peptide 1
Proteasome-activating peptide 1 enhances chymotrypsin-like proteasomal catalytic activity, boosting proteolytic rates both in vitro and within cultured cells. Additionally, it inhibits protein aggregation in a cellular m...
T76243 Proteasome-activating peptide 1 TFA
Proteasome-activating peptide 1 TFA is a potent activator of the proteasome, enhancing chymotrypsin-like proteasomal catalytic activity and thereby increasing proteolytic rates both in vitro and in culture. Additionally,...
T5374 NAcM-OPT E1/E2/E3 Enzyme , NEDD8
NAcM-OPT is a specific, reversible inhibitor targeting N-Acetyl-UBE2M interaction with DCN1 （IC50: 79 nM).
T24136 Heclin E1/E2/E3 Enzyme
Heclin is an inhibitor of HECT E3 ubiquitin ligase that acts by inhibiting Smurf2, Nedd4, and WWP1 with IC50 values of 6.8, 6.3, and 6.9 μM, respectively.
T80069 PACAP (6-27) (human, ovine, rat) Pituitary adenylate cyclase-activating peptide (6-27)
PACAP (6-27) (human, ovine, rat) serves as an antagonist for the PACAP receptor, inhibiting the catecholamine response of the canine adrenal gland to vasoactive intestinal peptide (VIP). This compound holds promise for r...
T5199 COH000 E1/E2/E3 Enzyme
COH000 is a covalent and irreversible inhibitor of small ubiquitin-like modifier (SUMO)-activating enzyme and inhibited SUMOylation (IC50: ~ 0.2 μM in vitro).
T16699 PYZD-4409 Others , E1/E2/E3 Enzyme
PYZD-4409 is a selective UBA1 inhibitor with an IC50 of 20 μM. PYZD-4409 induces cell death in malignant cells and is preferentially cytotoxic to malignant cells over normal hematopoietic cells.
T16102 ML-792 E1/E2/E3 Enzyme
ML-792 is a specific small ubiquitin-like modifier (SUMO)-activating enzyme (SAE) inhibitor. Compared with NAE/NEDD8 and UAE/ubiquitin (IC50s of 32 μM and >100 μM, respectively), ML-792 is an effective and selective inhi...
T16901 SMIP004 Apoptosis , Others , E1/E2/E3 Enzyme
SMIP004 is an SKP2 E3 ligase inhibitor. SMIP004 is a cancer cell-selective apoptosis inducer of human prostate cancer cells.
T3517 RO8994 Mdm2 , E1/E2/E3 Enzyme , p53
RO8994 is a highly effective and specific inhibitor of spiroindolinone small-molecule MDM2, with IC50 of 20 nM (MTT proliferation assays) and 5 nM (HTRF binding assays).
T8428 Subasumstat TAK-981 E1/E2/E3 Enzyme
Subasumstat (TAK-981) is a selective the SUMOylation enzymatic cascade inhibitor, has potential immune-activating and antineoplastic activities.
T75902 SLIGRL-NH2 TFA Protease-Activated Receptor-2 Activating Peptide TFA
SLIGRL-NH2 TFA, also known as Protease-Activated Receptor-2 Activating Peptide TFA, is a Protease-Activated Receptor-2 (PAR-2) agonist [1].
T6629 PYR-41 PYR41,PYR 41 Apoptosis , E1/E2/E3 Enzyme
PYR-41 is the first cell-permeable inhibitor of ubiquitin-activating enzyme E1, with no activity at E2.
T7379 2-D08 E1/E2/E3 Enzyme , TAM Receptor
2-D08 is a synthetic flavone that inhibits sumoylation, also inhibits Axl with an IC50 of 0.49 nM.2-D08 showed anti-aggregatory and neuroprotective effect.
T12261 NSC232003 E1/E2/E3 Enzyme
NSC232003 is a highly potent and cell-permeable inhibitor of UHRF1.
T13244 Ubiquitination-IN-1 Others
Ubiquitination-IN-1 is an inhibitor of ubiquitination and Cksl-Skp2 protein-protein interaction (IC50: 0.17 μM).
T9236 WSB1 Degrader 1 Others , E1/E2/E3 Enzyme
WSB1 Degrader 1 is a potent, orally active degrader of WD repeat and SOCS box-containing 1, exhibiting anti-cancer metastatic effects.
T7415 DKM 2-93 E1/E2/E3 Enzyme
DKM 2-93 is a relatively selective inhibitor of UBA5(IC50 : 430 μM).
TP1054 PACAP (1-38), human, ovine, rat TFA Pituitary Adenylate Cyclase Activating Polypeptide 38 (TFA)
PACAP (1-38), a novel neuropeptide isolated from the bovine hypothalamus is more active than vasoactive intestinal peptide (VIP) in stimulating adenylate cyclase (EC50=7 nM). PACAP 1-38 (10-9 M) increased substance P (SP...
T3317 SZL P1-41 Apoptosis , Others , E1/E2/E3 Enzyme
SZL P1-41, a skp2 inhibitor, can prevent assembly of Skp2-Skp1 complexes. It selectively suppresses Skp2 SCF E3 ligase activity but exhibits no effect on the activity of other SCF complexes. It also inhibits Skp2-mediate...
T2158 Nutlin-3 Nutlin3 E1/E2/E3 Enzyme
Nutlin-3 is an MDM2 antagonist.Nutlin-3 inhibits the MDM2-p53 interaction (IC50: 0.09 μM) and activates p53. Antiproliferative agent; chemotherapeutic agent; induces apoptosis in Y cells.
T11980 MD-224 Mdm2 , E1/E2/E3 Enzyme , PROTACs
MD-224 is a highly potent and efficacious MDM2 degrader based on the proteolysistargeting chimera (PROTAC) concept,and as a new class of anticancer agent.
T7889 C25-140 Others , TNF , E1/E2/E3 Enzyme , NF-κB
C25-140 is a small-molecule inhibitor of TRAF6-Ubc13.
T16888 SJ-172550 Mdm2 , E1/E2/E3 Enzyme
SJ-172550 is a small molecule inhibitor of MDMX (EC50: 5 μM).
TP1878 PACAP (1-38), human, ovine, rat Pituitary Adenylate Cyclase Activating Polypeptide 38,PACAP 1-38 PACAP
PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.
T3653 MX69 Mdm2 , E1/E2/E3 Enzyme , IAP
MX69 is the MDM2/XIAP inhibitor, blocking the MDM2 protein-XIAP RNA interaction, leading to MDM2 degradation.
T6149 YH239-EE Apoptosis , E1/E2/E3 Enzyme
YH239-EE, the ethyl ester of YH239, is a potent p53-MDM2 antagonist and an apoptosis inducer.
T23371 SMER3 SMER 3 Others , Ligand for E3 Ligase
SMER3 is an inhibitor of the Skp1-Cullin-F-box (SCF)(Met30) ubiquitin ligase, a member of the SCF E3-ligase family, which regulates diverse cellular processes including transcription, cell-cycle control and immune respon...
T8564 BC-1382 Others , E1/E2/E3 Enzyme
BC-1382 is a potent ubiquitin E3 ligase HECTD2 inhibitor that specificly disrupts the HECTD2/PIAS1 interaction(IC50 of 5 nM).
T4253 Skp2 Inhibitor C1 SKPin C1 Others , E1/E2/E3 Enzyme
Skp2 Inhibitor C1 (SKPin C1)(SKPin C1) is a specific small molecule inhibitor of Skp2-mediated p27 degradation.
T6332 Pevonedistat MLN4924 E1/E2/E3 Enzyme , NEDD8
Pevonedistat (MLN4924) is a potent and selective NEDD8 activating enzyme (NAE) inhibitor (IC50=4.7 nM). Pevonedistat can be used for the treatment of myelodysplastic syndromes (MDS) and also has antitumor activity.
T8844 Diflapolin Others , FLAP , Epoxide Hydrolase
Diflapolin is a highly active dual 5-lipoxygenase-activating protein (FLAP)/soluble epoxide hydrolase (sEH) inhibitor with marked anti-inflammatory efficacy and high target selectivity.
T10703 Mezigdomide CC-92480 Apoptosis , E1/E2/E3 Enzyme , Molecular Glues
Mezigdomide (CC-92480) is a potent, novel, selective and active cereblon E3 ubiquitin ligase modulator (CELMoD) that often acts as a molecular glue. Mezigdomide has antimyeloma activity.
T13349 WS-383 E1/E2/E3 Enzyme
WS-383 is a selective, potent and reversible DCN1-UBC12 interaction inhibitor(IC50 of 11 nM).
T3110 PRT4165 NSC600157,PRT 4165 BMI-1 , Others , E1/E2/E3 Enzyme
PRT4165 (NSC600157) is a potent PRC1-mediated H2A ubiquitylation inhibitor.
T3549 Avadomide CC 122 Apoptosis , E1/E2/E3 Enzyme , Ligand for E3 Ligase
Avadomide (CC 122) is an orally available pleiotropic pathway modulator with potential antineoplastic activity.
T5555 Siremadlin NVP-HDM 201 E1/E2/E3 Enzyme
Siremadlin (NVP-HDM 201) is a potent, orally bioavailable and highly specific p53-MDM2 interaction inhibitor.
T16974 TAK-243 MLN7243 Apoptosis , E1/E2/E3 Enzyme , NF-κB
TAK-243 (MLN7243) is a selective inhibitor of the ubiquitin-activating enzyme UAE (IC50=1 nM). TAK-243 blocks ubiquitin binding and disrupts mono-ubiquitin signaling as well as overall protein ubiquitination. TAK-243 exh...
T9023 Atuliflapon AZD5718 FLAP
Atuliflapon (AZD5718) is a novel 5-Lipoxygenase Activating Protein(FLAP) inhibitor for Treatment of Coronary Artery Disease.
T1493 BH3I-1 BHI1 BCL , E1/E2/E3 Enzyme
BH3I-1 (BHI1) is a Bcl-2 antagonist.
T6254 Idasanutlin RG7388,Ro 5503781 Mdm2 , E1/E2/E3 Enzyme
Idasanutlin (Ro 5503781) (RG-7388) is an effective and specific p53-MDM2 inhibitor (IC50: 6 nM).
T6965 RG7112 RG-7112,RG 7112,RO5045337 Mdm2 , E1/E2/E3 Enzyme
RG7112 (RO5045337) (RO5045337) is an orally bioavailable and selective p53-MDM2 inhibitor.
T6611 NSC697923 2-[(4-methylphenyl)sulfonyl]-5-nitrofuran E1/E2/E3 Enzyme
NSC-697923 (2-[(4-methylphenyl)sulfonyl]-5-nitrofuran), a potent inhibitor of UBE2N (ubiquitin-conjugating enzyme E2 N, Ubc13), exhibits its role in inducing cell death in neuroblastoma (NB) cells through two distinct me...
TQ0231 NVP-CGM097 CGM097 Mdm2 , E1/E2/E3 Enzyme
NVP-CGM097 (CGM097) is an effective and specific MDM2 inhibitor (IC50: 1.7 nM for hMDM2).
TQ0127 Navtemadlin AMG232,CS-1300 Mdm2 , E1/E2/E3 Enzyme
Navtemadlin (AMG232) is a potent, selective and orally available inhibitor of p53-MDM2 interaction (IC50: 0.6 nM). It binds to MDM2 with a Kd of 0.045 nM.
T13090 TAS4464 hydrochloride E1/E2/E3 Enzyme , NEDD8
TAS4464 hydrochloride is a highly potent and selective NEDD8 activating enzyme (NAE) inhibitor(IC50 of 0.955 nM).

Compounds

PAR-2 Activating Peptide acetate
TP1046L
Synonym: SLIGRL-NH2 acetate,PAR-2 Activating Peptide acetate(171436-38-7 free base),Protease-Activated Receptor-2 Activating Peptide acetate
Target: Protease-activated Receptor
Sperm-activating peptide 1
TP2411
Synonym:
Target:
PAC-1
T2503
Synonym: Procaspase activating compound 1
Target: Apoptosis, Caspase, Autophagy
SLIGRL-NH2
TP1046
Synonym: Protease-Activated Receptor-2 Activating Peptide
Target: Protease-activated Receptor
Proteasome-activating peptide 1
T81372
Synonym:
Target:
Proteasome-activating peptide 1 TFA
T76243
Synonym:
Target:
NAcM-OPT
T5374
Synonym:
Target: E1/E2/E3 Enzyme, NEDD8
Heclin
T24136
Synonym:
Target: E1/E2/E3 Enzyme
PACAP (6-27) (human, ovine, rat)
T80069
Synonym: Pituitary adenylate cyclase-activating peptide (6-27)
Target:
COH000
T5199
Synonym:
Target: E1/E2/E3 Enzyme
PYZD-4409
T16699
Synonym:
Target: Others, E1/E2/E3 Enzyme
ML-792
T16102
Synonym:
Target: E1/E2/E3 Enzyme
SMIP004
T16901
Synonym:
Target: Apoptosis, Others, E1/E2/E3 Enzyme
RO8994
T3517
Synonym:
Target: Mdm2, E1/E2/E3 Enzyme, p53
Subasumstat
T8428
Synonym: TAK-981
Target: E1/E2/E3 Enzyme
SLIGRL-NH2 TFA
T75902
Synonym: Protease-Activated Receptor-2 Activating Peptide TFA
Target:
PYR-41
T6629
Synonym: PYR41,PYR 41
Target: Apoptosis, E1/E2/E3 Enzyme
2-D08
T7379
Synonym:
Target: E1/E2/E3 Enzyme, TAM Receptor
NSC232003
T12261
Synonym:
Target: E1/E2/E3 Enzyme
Ubiquitination-IN-1
T13244
Synonym:
Target: Others
WSB1 Degrader 1
T9236
Synonym:
Target: Others, E1/E2/E3 Enzyme
DKM 2-93
T7415
Synonym:
Target: E1/E2/E3 Enzyme
PACAP (1-38), human, ovine, rat TFA
TP1054
Synonym: Pituitary Adenylate Cyclase Activating Polypeptide 38 (TFA)
Target:
SZL P1-41
T3317
Synonym:
Target: Apoptosis, Others, E1/E2/E3 Enzyme
Nutlin-3
T2158
Synonym: Nutlin3
Target: E1/E2/E3 Enzyme
MD-224
T11980
Synonym:
Target: Mdm2, E1/E2/E3 Enzyme, PROTACs
C25-140
T7889
Synonym:
Target: Others, TNF, E1/E2/E3 Enzyme, NF-κB
SJ-172550
T16888
Synonym:
Target: Mdm2, E1/E2/E3 Enzyme
PACAP (1-38), human, ovine, rat
TP1878
Synonym: Pituitary Adenylate Cyclase Activating Polypeptide 38,PACAP 1-38
Target: PACAP
MX69
T3653
Synonym:
Target: Mdm2, E1/E2/E3 Enzyme, IAP
YH239-EE
T6149
Synonym:
Target: Apoptosis, E1/E2/E3 Enzyme
SMER3
T23371
Synonym: SMER 3
Target: Others, Ligand for E3 Ligase
BC-1382
T8564
Synonym:
Target: Others, E1/E2/E3 Enzyme
Skp2 Inhibitor C1
T4253
Synonym: SKPin C1
Target: Others, E1/E2/E3 Enzyme
Pevonedistat
T6332
Synonym: MLN4924
Target: E1/E2/E3 Enzyme, NEDD8
Diflapolin
T8844
Synonym:
Target: Others, FLAP, Epoxide Hydrolase
Mezigdomide
T10703
Synonym: CC-92480
Target: Apoptosis, E1/E2/E3 Enzyme, Molecular Glues
WS-383
T13349
Synonym:
Target: E1/E2/E3 Enzyme
PRT4165
T3110
Synonym: NSC600157,PRT 4165
Target: BMI-1, Others, E1/E2/E3 Enzyme
Avadomide
T3549
Synonym: CC 122
Target: Apoptosis, E1/E2/E3 Enzyme, Ligand for E3 Ligase
Siremadlin
T5555
Synonym: NVP-HDM 201
Target: E1/E2/E3 Enzyme
TAK-243
T16974
Synonym: MLN7243
Target: Apoptosis, E1/E2/E3 Enzyme, NF-κB
Atuliflapon
T9023
Synonym: AZD5718
Target: FLAP
BH3I-1
T1493
Synonym: BHI1
Target: BCL, E1/E2/E3 Enzyme
Idasanutlin
T6254
Synonym: RG7388,Ro 5503781
Target: Mdm2, E1/E2/E3 Enzyme
RG7112
T6965
Synonym: RG-7112,RG 7112,RO5045337
Target: Mdm2, E1/E2/E3 Enzyme
NSC697923
T6611
Synonym: 2-[(4-methylphenyl)sulfonyl]-5-nitrofuran
Target: E1/E2/E3 Enzyme
NVP-CGM097
TQ0231
Synonym: CGM097
Target: Mdm2, E1/E2/E3 Enzyme
Navtemadlin
TQ0127
Synonym: AMG232,CS-1300
Target: Mdm2, E1/E2/E3 Enzyme
TAS4464 hydrochloride
T13090
Synonym:
Target: E1/E2/E3 Enzyme, NEDD8
1 2 3 4 5 6 7 8
Cat No. Product Name Synonyms Targets
T4S0181 Hinokiflavone MMP , BCL , E1/E2/E3 Enzyme
Hinokiflavone, a novel modulator of pre-mRNA splicing activity both in vitro and in cellulo, inhibits the assembly of the spliceosome, particularly blocking the formation of the B complex. Additionally, it acts as a SUMO...
T9352 Hydrocotarnine Others
hydrocotarnine is an inhibitor of Cbl.
T4036 Solasodine Solancarpidine,Purapuridine,Solasodin Apoptosis , Others , E1/E2/E3 Enzyme , Antifungal
Solasodine (Purapuridine)(Purapuridine) is a poisonous alkaloid chemical compound that occurs in plants of the Solanaceae family. Solasodine showed selective cytotoxicity against cervical cancer cell line (HeLa) and huma...
T2947 Indole-3-carbinol I3C,3-Indolemethanol,Indole-3-Methanol E1/E2/E3 Enzyme , NF-κB , Aryl Hydrocarbon Receptor , Endogenous Metabolite , p53
Indole-3-carbinol (I3C), a naturally occurring, orally available cleavage product of the glucosinolate glucobrassicanin, inhibits NF-κB and IκBα kinase activation.
T6S2123 Ginkgolic Acid Romanicardic acid,Ginkgolic acid I,Ginkgolic acid (15:1),Ginkgolic acid C15:1 Others , E1/E2/E3 Enzyme
Ginkgolic Acid (Romanicardic acid) C15:1 represses curli genes and prophage genes in EHEC.
T8288 14-Deoxyandrographolide Apoptosis , Others
14-Deoxyandrographolide is a bioactive compound of Andrographis paniculata with hepatoprotective efficacy. It desensitizes hepatocytes to TNF-α-mediated apoptosis through the release of TNFRSF1A release.
TN4222 Homoeriodictyol 7-O-β-D-glucoside Homoeriodictyol 7-O-glucoside Others , Platelet aggregation
Homoeriodictyol 7-O-β-D-glucoside (Homoeriodictyol 7-O-glucoside) is a natural product from Viscum coloratum(Kom.)Nakai. Homoeriodictyol 7-O-β-D-glucoside is an antagonist of platelet-activating factor (PAF).
T0800 Danthron Dantron,1,8-Dihydroxyanthraquinone,Chrysazin,Antrapurol Virus Protease , Antibacterial , AMPK , Autophagy
Danthron (Antrapurol) is a natural product, regulates glucose, and lipid metabolism by activating AMPK.
T4950 1,2-Dipalmitoyl-sn-glycerol (S)-1,2-Dipalmitin Endogenous Metabolite , PKC
1,2-Dipalmitoyl-sn-glycerol ((S)-1,2-Dipalmitin) is an analog of the PKC-activating second messenger diacylglycerol (DAG). It weakly activates PKC.
TN4114 Gardenin A ERK , LDL , MAPK , PKA , PKC
Gardenin A shows neurotrophic effects via activating MAPK/ERK, PKC, and PKA. Gardenin A exhibits antidepressant, anticonvulsant and anxiolytic effects.
TN2346 Mogrol ERK , AMPK , STAT
Mogrol, a biometabolite of mogrosides, functions by inhibiting the ERK1/2 and STAT3 pathways, diminishing CREB activation, and activating AMPK signaling.
T0129 Sanguinarine chloride Pseudochelerythrine chloride,Sanguinarium chloride Apoptosis , EGFR , VEGFR , Antibacterial , Parasite , Autophagy
Sanguinarine chloride (Pseudochelerythrine chloride), a benzophenanthridine alkaloid, stimulates apoptosis by activating the production of reactive oxygen species (ROS).
T3896 Shanzhiside methyl ester Glucagon Receptor
Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38 MAPK signaling.
T5281 Skatole Scatole,3-Methylindole,3-​Methylindole,3-Methyl-1H-indole,beta-Methylindole AhR , p38 MAPK , Aryl Hydrocarbon Receptor , Endogenous Metabolite , Antibacterial , Autophagy , Antifungal
Skatole (3-Methyl-1H-indole) is produced by intestinal bacteria. Skatole regulates intestinal epithelial cellular functions through activating aryl hydrocarbon receptors and p38.
T2A2497 L-Glutamic acid (S)-Glutamic acid,glutamic acid,(+)-L-Glutamic acid,Aciglut,glutacid,Glutaminol Apoptosis , Ferroptosis , Endogenous Metabolite , iGluR
L-Glutamic acid (Glutaminol) acts as an excitatory transmitter, shows a direct activating effect on the release of DA from dopaminergic terminals.
T5S2178 Fargesin (+/-)-Fargesin Adrenergic Receptor
1. Fargesin ((+/-)-Fargesin) as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Fargesin improves dyslipidemia and hyperglycemia by activating...
T3S0335 Soyasaponin Bb Soyasaponin I NF-κB , Caspase
1. Soyasaponin Bb (Soyasaponin I) can suppress Eca-976 cell growth, reverse effects on over expression of c-met, VEGF, and induce cell apoptosis through inhibiting HDAC1-NF-kappaB and activating PETEN and caspase-3 signa...
T3916 Ginsenoside F2 Apoptosis , Endogenous Metabolite , Autophagy
Ginsenoside F2 has antiproliferative activity against breast cancer stem cells (CSCs). It induces apoptosis in breast CSCs by activating the intrinsic apoptotic pathway and mitochondrial dysfunction.
T13818 Phytohemagglutinin PHA-M Apoptosis
Phytohemagglutinin (PHA-M) is a lectin, isolated from the red kidney bean , induces apoptosis via increasing proapoptotic protein Bax and activating caspases-3. Anti-tumor activity
TN4379 Kansuinine A IL Receptor , STAT , Interleukin
Kansuinine A possesses analgesic props, it also shows NGF inducing activity.
TN1461 (-)-Butin Butin Akt , PI3K , Nrf2
(-)-Butin (Butin) has antioxidant activity, can protect cells against H2O2-induced apoptosis, oxidative DNA damage and oxidative mitochondrial dysfunction; it attenuates oxidative stress by activating Nrf2-mediated Mn SO...
T0627 β-Alanine beta-Alanine,3-Aminopropanoic acid,2-Carboxyethylamine GABA Receptor , Endogenous Metabolite
β-Alanine (3-Aminopropanoic acid) is a naturally occurring beta amino acid formed in vivo by the degradation of dihydrouracil and carnosine. It acts as a neurotransmitter by activating glycine and GABA receptors.
T3665 Tectoridin Shekanin Estrogen Receptor/ERR , Reductase
Tectoridin (Shekanin) possesses an estrogenic and thyroid hormone-like agent by activating estrogen and thyroid hormone receptors. Tectoridin has anti-oxidant, anti-inflammatory and hypoglycemic activities; Tectoridin an...
T5764 Alliin (S)-3-(Allylsulphinyl)-L-alanine NF-κB , PPAR
Alliin ((S)-3-(Allylsulphinyl)-L-alanine) is a garlic organosulfur compound that possesses various pharmacological properties.alliin protected against LPS-induced ALI by activating PPARγ, which subsequently inhibited LPS...
T2978 Mogroside V AMPK
Mogroside V is a widely used sweetener, has in vitro AMPK activating effect, it also has anti-inflammatory potential in murine macrophages and a murine ear edema model, and has the potential to protect against LPS-induce...
TN7036 N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide (9Z,12Z,15Z)-N-[(3-Methoxyphenyl)methyl]-9,12,15-octadecatrienamide,Macamide Impurity 14 Wnt/beta-catenin
N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide (Macamide Impurity 14) induces osteogenic differentiation and subsequent bone formation of mesenchymal stem cells by activating the canonical Wnt/β-catenin signaling pa...
TN2322 Yangambin Calcium Channel , PAFR
Yangambin is a selective antagonist of the cardiovascular effects of platelet activating factor (PAF); it has hypotensive effect, which is probably due to a peripheral vasodilatation that involves, at least, the inhibiti...
TN2080 Pinoresinol (+)-Pinoresinol Apoptosis , NF-κB , CDK , p53
Pinoresinol ((+)-Pinoresinol) has antiinflammatory, hepatoprotective, and fungicidal activities, it can protect pial microcirculation from I-reperfusion injury, to increase nitric oxide release and to reduce oxidative st...
TN1873 Lirinidine Others
(+)-Lirinidine has antioxidative activity, and it can significantly inhibit the proliferation of melanoma cells; it also shows potent inhibition of melanogenesis. Lirinidine exhibits significant inhibition of collagen, a...
T4S1335 Daphnoretin Dephnoretin,Thymelol Influenza Virus , Caspase , PKC
1. Daphnoretin (Thymelol) has strong antiviral activity, mainly on the later phase of the replication cycle. 2. Daphnoretin has anticancer effects on leukemia, osteosarcoma and uterine cervix cancer cells, might through ...
T3867 Alpinetin (-)-alpinetin BCL , PPAR
Alpinetin ((-)-alpinetin) has antibacterial activity.Alpinetin has anti-inflammatory activity.Alpinetin can enhance the sensitivity of HepG2 hepatoma cells to the chemotherapeutic agent CDDP. Alpinetin has strong anti-he...
T2S2173 (E)-Naringenin chalcone Isosalipurpol,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone Others
Naringenin chalcone (Isosalipurpol) has antiallergic activity Naringenin chalcone suppresses asthmatic symptoms by inhibiting Th2 cytokine production from CD4 T cells. Naringenin chalcone is a potent tomato flavonoid tha...
T3923 Calycosin Cyclosin,3'-Hydroxyformononetin Apoptosis , Tyrosinase
Calycosin (Cyclosin) acts as a selective estrogen receptor modulator. Calycosin induces apoptosis in human ovarian cancer SKOV3 cells by activating caspases and Bcl-2 family proteins. Calycosin suppresses breast cancer c...
T5S2358 Dehydrocorydaline Dehydrocorydalin,13-Methylpalmatine BCL , PARP , p38 MAPK , Caspase , Parasite , Autophagy
1. Dehydrocorydaline (13-Methylpalmatine) exerts anti-metastatic potential via suppression of MMPs and Bcl-2 signaling in NSC-LC cells. 2. Dehydrocorydaline stimulates p38 MAPK activation, which can enhance heterodimeriz...
T5S1805 5,7-Dihydroxychromone 5,7-Dihydroxy-4H-Chromen-4-One Others , Virus Protease , PARP , Caspase , Nrf2
1. 5,7-Dihydroxychromone (5,7-Dihydroxy-4H-Chromen-4-One) isolated from DME is one of the active compounds that may contribute to regulate blood glucose levels. 2. 5,7-Dihydroxychromone exerts neuroprotective effect agai...
T3229 Cytochalasin D ATPase , p38 MAPK , Calcium Channel , Akt , PI3K
Cytochalasin D is an actin inhibitor, the removal of actin stress fibers is crucial for the chondrogenic differentiation. It may be an inhibitor of some fertilization processes such as sperm penetration or sperm head dec...
T2S2264 Linalool Linalol,(±)-Linalool,Phantol Apoptosis , IL Receptor , TNF , Endogenous Metabolite , iGluR
1. Linalool (Linalol), a natural compound of the essential oils, has been shown to have antinociceptive, antimicrobial, and anti-inflammatory properties. 2. Linalool was protected against LPS/GalN-induced liver injury th...
TN5171 Tricetin Apoptosis , Others , Nrf2
Tricetin is a flavonoid isolated from pomegranate.Tricetin is a potent competitive inhibitor of Keap1-Nrf2 protein-protein interaction (PPI) and protects Parkinson's disease patients from 6-OHDA-induced neurotoxicity by ...
T25983 Prehispanolone LC 5504,LC5504,LC-5504
Prehispanolone is a platelet activating factor antagonist from Chinese medicinal herb Leonurus heterophyllus.
TN3520 Bisdethiobis(methylthio)gliotoxin PAFR
Bisdethiobis(methylthio)gliotoxin is a platelet activating factor (PAF) antagonist.
TN5045 Spiradine F PAFR
Spiradine F can significantly inhibit platelet-activating factor(PAF)-induced platelet aggregation in a concentration-dependent manner.
T13559 Astragaloside VI EGFR
Astragaloside VI could improve wound healing by activating the EGFR/ERK signaling pathway.
TN4821 Pregomisin PAFR
Pregomisin shows platelet-activating factor (PAF) antagonistic activity and the IC 50 value is 4.8x10(-5) M.
TN4367 Kadsurin A PAFR
Kadsurin A has anti-platelet activating factor activities.
T28021 Meso-Dihydroguaiaretic acid
meso-Dihydroguaiaretic acid is an LXR-α antagonist, it inhibits hepatic lipid accumulation by activating AMP-activated protein kinase in human HepG2 cells.
TN1654 Futoquinol Others , ROS , PAFR
Futoquinol is an anti-platelet activating factor principle from the stem part of Piper futokadsura (Piperaceae), the Chinese drug haifengteng.
T7711 Uridine triphosphate UTP,Uridine 5'-triphosphate Others , Endogenous Metabolite
Uridine triphosphate (Uridine 5'-triphosphate) increases proliferation of human cancerous pancreatic duct epithelial cells by activating P2Y2 receptor.
T15541 Hyperforin dicyclohexylammonium salt Hyperforin DCHA Others
Hyperforin dicyclohexylammonium salt is a transient receptor canonical 6 channel activator with antidepressant effect. It modulates Ca2+ levels by activating Ca2+-conducting non-selective canonical TRPC6 channels.
T13716 (+)-Guaiacin Others
(+)-Guaiacin is a compound isolated from the bark of Machilus wangchiana Chun. It shows potent in vitro activities against the release of β-glucuronidase in rat polymorphonuclear leukocytes (PMNs) induced by platelet-act...
TN1570 Deoxyvasicinone Others
Deoxyvasicinone derivatives can be considered as promising lead molecules for the development of more potent inhibitors of NEDD8-activating enzyme.
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Natural Products

Hinokiflavone
T4S0181
Synonym:
Target: MMP, BCL, E1/E2/E3 Enzyme
hydrocotarnine
T9352
Synonym:
Target: Others
Solasodine
T4036
Synonym: Solancarpidine,Purapuridine,Solasodin
Target: Apoptosis, Others, E1/E2/E3 Enzyme, Antifungal
Indole-3-carbinol
T2947
Synonym: I3C,3-Indolemethanol,Indole-3-Methanol
Target: E1/E2/E3 Enzyme, NF-κB, Aryl Hydrocarbon Receptor, Endogenous Metabolite, p53
Ginkgolic Acid
T6S2123
Synonym: Romanicardic acid,Ginkgolic acid I,Ginkgolic acid (15:1),Ginkgolic acid C15:1
Target: Others, E1/E2/E3 Enzyme
14-Deoxyandrographolide
T8288
Synonym:
Target: Apoptosis, Others
Homoeriodictyol 7-O-β-D-glucoside
TN4222
Synonym: Homoeriodictyol 7-O-glucoside
Target: Others, Platelet aggregation
Danthron
T0800
Synonym: Dantron,1,8-Dihydroxyanthraquinone,Chrysazin,Antrapurol
Target: Virus Protease, Antibacterial, AMPK, Autophagy
1,2-Dipalmitoyl-sn-glycerol
T4950
Synonym: (S)-1,2-Dipalmitin
Target: Endogenous Metabolite, PKC
Gardenin A
TN4114
Synonym:
Target: ERK, LDL, MAPK, PKA, PKC
Mogrol
TN2346
Synonym:
Target: ERK, AMPK, STAT
Sanguinarine chloride
T0129
Synonym: Pseudochelerythrine chloride,Sanguinarium chloride
Target: Apoptosis, EGFR, VEGFR, Antibacterial, Parasite, Autophagy
Shanzhiside methyl ester
T3896
Synonym:
Target: Glucagon Receptor
Skatole
T5281
Synonym: Scatole,3-Methylindole,3-​Methylindole,3-Methyl-1H-indole,beta-Methylindole
Target: AhR, p38 MAPK, Aryl Hydrocarbon Receptor, Endogenous Metabolite, Antibacterial, Autophagy, Antifungal
L-Glutamic acid
T2A2497
Synonym: (S)-Glutamic acid,glutamic acid,(+)-L-Glutamic acid,Aciglut,glutacid,Glutaminol
Target: Apoptosis, Ferroptosis, Endogenous Metabolite, iGluR
Fargesin
T5S2178
Synonym: (+/-)-Fargesin
Target: Adrenergic Receptor
Soyasaponin Bb
T3S0335
Synonym: Soyasaponin I
Target: NF-κB, Caspase
Ginsenoside F2
T3916
Synonym:
Target: Apoptosis, Endogenous Metabolite, Autophagy
Phytohemagglutinin
T13818
Synonym: PHA-M
Target: Apoptosis
Kansuinine A
TN4379
Synonym:
Target: IL Receptor, STAT, Interleukin
(-)-Butin
TN1461
Synonym: Butin
Target: Akt, PI3K, Nrf2
β-Alanine
T0627
Synonym: beta-Alanine,3-Aminopropanoic acid,2-Carboxyethylamine
Target: GABA Receptor, Endogenous Metabolite
Tectoridin
T3665
Synonym: Shekanin
Target: Estrogen Receptor/ERR, Reductase
Alliin
T5764
Synonym: (S)-3-(Allylsulphinyl)-L-alanine
Target: NF-κB, PPAR
Mogroside V
T2978
Synonym:
Target: AMPK
N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide
TN7036
Synonym: (9Z,12Z,15Z)-N-[(3-Methoxyphenyl)methyl]-9,12,15-octadecatrienamide,Macamide Impurity 14
Target: Wnt/beta-catenin
Yangambin
TN2322
Synonym:
Target: Calcium Channel, PAFR
Pinoresinol
TN2080
Synonym: (+)-Pinoresinol
Target: Apoptosis, NF-κB, CDK, p53
Lirinidine
TN1873
Synonym:
Target: Others
Daphnoretin
T4S1335
Synonym: Dephnoretin,Thymelol
Target: Influenza Virus, Caspase, PKC
Alpinetin
T3867
Synonym: (-)-alpinetin
Target: BCL, PPAR
(E)-Naringenin chalcone
T2S2173
Synonym: Isosalipurpol,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone
Target: Others
Calycosin
T3923
Synonym: Cyclosin,3'-Hydroxyformononetin
Target: Apoptosis, Tyrosinase
Dehydrocorydaline
T5S2358
Synonym: Dehydrocorydalin,13-Methylpalmatine
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
5,7-Dihydroxychromone
T5S1805
Synonym: 5,7-Dihydroxy-4H-Chromen-4-One
Target: Others, Virus Protease, PARP, Caspase, Nrf2
Cytochalasin D
T3229
Synonym:
Target: ATPase, p38 MAPK, Calcium Channel, Akt, PI3K
Linalool
T2S2264
Synonym: Linalol,(±)-Linalool,Phantol
Target: Apoptosis, IL Receptor, TNF, Endogenous Metabolite, iGluR
Tricetin
TN5171
Synonym:
Target: Apoptosis, Others, Nrf2
Prehispanolone
T25983
Synonym: LC 5504,LC5504,LC-5504
Target:
Bisdethiobis(methylthio)gliotoxin
TN3520
Synonym:
Target: PAFR
Spiradine F
TN5045
Synonym:
Target: PAFR
Astragaloside VI
T13559
Synonym:
Target: EGFR
Pregomisin
TN4821
Synonym:
Target: PAFR
Kadsurin A
TN4367
Synonym:
Target: PAFR
meso-Dihydroguaiaretic acid
T28021
Synonym:
Target:
Futoquinol
TN1654
Synonym:
Target: Others, ROS, PAFR
Uridine triphosphate
T7711
Synonym: UTP,Uridine 5'-triphosphate
Target: Others, Endogenous Metabolite
Hyperforin dicyclohexylammonium salt
T15541
Synonym: Hyperforin DCHA
Target: Others
(+)-Guaiacin
T13716
Synonym:
Target: Others
Deoxyvasicinone
TN1570
Synonym:
Target: Others
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Recombinant Proteins

Species：
Human (255)
Mouse (83)
Rat (25)
Cynomolgus (24)
Rhesus (5)
Staphylococcus aureus (5)
Rhesus macaque (3)
Apis mellifera (2)
Bacillus subtilis (2)
Canine (2)
Expression System：
HEK293 (228)
E. coli (119)
Human Cells (40)
Baculovirus-Insect Cells (29)
Yeast (12)
Baculovirus (6)
CHO (3)
in vitro E. coli expression system (3)
Tag：
His (96)
hFc (47)
N-terminal 6xHis-tagged (33)
Tag Free (32)
C-6His (21)
C-His-Avi (21)
N-terminal 10xHis-tagged and C-terminal Myc-tagged (20)
C-His (16)
C-hFc (14)
N-terminal 6xHis-SUMO-tagged (13)
Cat No. Product Name Species Expression System
TMPY-02840 Ubiquitin Activating Enzyme E1/UBA1 Protein, Human, Recombinant (His & GST) Human Baculovirus-Insect Cells
UBE1, also known as UBA1, belongs to the ubiquitin-activating E1 family. UBE1 gene complements an X-linked mouse temperature-sensitive defect in DNA synthesis, and thus may function in DNA repair. It is part of a gene cl...
TMPY-03441 SAE1 Protein, Human, Recombinant Human Baculovirus-Insect Cells
SAE1 belongs to the ubiquitin-activating E1 family. It is a heterodimer that acts as a E1 ligase for SUMO1, SUMO2, SUMO3, and probably SUMO4. It functions as a UBLI E1 ligase mediating the ATP-dependent activation of UBL...
TMPJ-01011 FGF-9 Protein, Mouse, Recombinant (His) Mouse E. coli
Fibroblast growth factor-9 (FGF-9) is an approximately 26 kDa secreted glycoprotein of the FGF family. Secreted mouse FGF-9 lacks the N-terminal 1-3 aa and shares >98% sequence identity with rat, human, equine, porcine a...
TMPJ-00090 FGF-9 Protein, Human, Recombinant Human E. coli
Fibroblast Growth Factor 9 (FGF-9) belongs to the Fibroblast growth factor (FGF) family. FGF family members possess broad mitogenic and cell survival activities, and are involved in a variety of biological processes, inc...
TMPY-01481 FLAP Protein, Human, Recombinant (His) Human Baculovirus-Insect Cells
Arachidonate 5-Lipoxygenase-Activating Protein (ALOX5AP), also known as FLAP, belongs to the MAPEG family. ALOX5AP/FLAP is an essential partner of 5-LO for this process. The FLAP (ALOX5AP) gene has been linked to risk fo...
TMPJ-01324 UBA5 Protein, Human, Recombinant (His) Human E. coli
UBA5 is a member of the ubiquitin-activating E1 family and UBA5 subfamily. Ubiquitin and ubiquitin-like proteins are recognized as covalently conjugated to various cellular substrates by a three-step enzymatic pathway. T...
TMPJ-01391 BAFF/TNFSF13B Protein, Mouse, Recombinant (mFc) Mouse Human Cells
TNFSF13B/TNFSF20 belongs to the tumor necrosis factor family. It abundantly is expressed in peripheral blood Leukocytes and is specifically expressed in monocytes and macrophages. Also found in the spleen, lymph node, bo...
TMPY-03062 SAE1 Protein, Human, Recombinant (His & GST) Human Baculovirus-Insect Cells
SAE1 belongs to the ubiquitin-activating E1 family. It is a heterodimer that acts as a E1 ligase for SUMO1, SUMO2, SUMO3, and probably SUMO4. It functions as a UBLI E1 ligase mediating the ATP-dependent activation of UBL...
TMPJ-01116 HABP2 Protein, Human, Recombinant (His) Human Human Cells
Hyaluronan-binding protein 2（HABP2） is an extracellular serine protease which binds hyaluronic acid. It secreted as an inactive single-chain precursor and is then activated to a heterodimeric form, which consists of a 50...
TMPH-03456 CAK1 Protein, S. cerevisiae, Recombinant (His & Myc) Saccharomyces cerevisiae Baculovirus
CAK1 Protein, S. cerevisiae, Recombinant (His & Myc) is expressed in Baculovirus with N-terminal 10xHis tag and C-terminal Myc tag. The predicted molecular weight is 46.1 kDa. Accession number: P43568
TMPJ-00611 SFP Protein, B.subtilis, Recombinant (His) B.subtilis E. coli
The Bacillus subtilis enzyme Sfp, required for production of the lipoheptapeptide antibiotic surfactin, posttranslationally phosphopantetheinylates a serine residue in each of the seven peptidyl carrier protein domains o...
TMPY-02444 ATF2 Protein, Human, Recombinant (His & GST) Human Baculovirus-Insect Cells
Activating transcription factor 2, also known as ATF2, is a member of the leucine zipper family of DNA-binding proteins that binds to the cAMP response element. Its activity is enhanced after phosphorylation by stress-ac...
TMPY-06748 UBA6 Protein, Human, Recombinant (GST) Human Baculovirus-Insect Cells
UBA6 (Ubiquitin Like Modifier Activating Enzyme 6) is a Protein Coding gene. The UBA6 gene, located on 4q13.2, is conserved in chimpanzee, Rhesus monkey, dog, cow, mouse, rat, chicken, zebrafish, and frog. Uba6 is a homo...
TMPH-01163 CXCL5 Protein, Human, Recombinant (His) Human E. coli
CXCL5 Protein, Human, Recombinant (His) is expressed in E. coli.
TMPH-03457 CAK1 Protein, S. cerevisiae, Recombinant (E. coli, His & Myc) Saccharomyces cerevisiae E. coli
CAK1 Protein, S. cerevisiae, Recombinant (E. coli, His & Myc) is expressed in E. coli with N-terminal 10xHis tag and C-terminal Myc tag. The predicted molecular weight is 49.6 kDa. Accession number: P43568
TMPH-03520 ACP Protein, S. aureus, Recombinant (His & SUMO) Staphylococcus aureus E. coli
Carrier of the growing fatty acid chain in fatty acid biosynthesis. Is able to confer high methicillin resistance to S.aureus when overproduced.
TMPH-00164 4'-phosphopantetheinyl transferase ffp Protein, Bacillus subtilis, Recombinant (His & Myc) Bacillus subtilis E. coli
4'-phosphopantetheinyl transferase ffp Protein, Bacillus subtilis, Recombinant (His & Myc) is expressed in E. coli.
TMPH-00572 ACP Protein, E. coli, Recombinant (His & SUMO) E. coli E. coli
Carrier of the growing fatty acid chain in fatty acid biosynthesis.
TMPH-03518 ACP Protein, S. aureus, Recombinant (GST) Staphylococcus aureus E. coli
Carrier of the growing fatty acid chain in fatty acid biosynthesis. Is able to confer high methicillin resistance to S.aureus when overproduced.
TMPJ-00425 NCR1 Protein, Mouse, Recombinant (hFc) Mouse Human Cells
Natural cytotoxicity triggering receptor 1(NKp46/NCR1) is a single-pass type I membrane protein. It consists of two extracellular Ig-like domains followed by a short stalk region, a transmembrane domain containing a posi...
TMPH-03519 ACP Protein, S. aureus, Recombinant (His) Staphylococcus aureus Yeast
Carrier of the growing fatty acid chain in fatty acid biosynthesis. Is able to confer high methicillin resistance to S.aureus when overproduced.
TMPJ-00218 SLAMF6 Protein, Human, Recombinant (His & Avi), Biotinylated Human Human Cells
SLAM Family Member 6 (SLAMF6) is a 60 kD single-pass type I membrane protein that belongs to the SLAM subgroup of the CD2 family. Human SLAMF6/ NTB-A contains a 205 amino acid extracellular domain (ECD) with one Ig-like ...
TMPY-02648 PACAP receptor/ADCYAP1R1 Protein, Human, Recombinant (hFc) Human HEK293
Pituitary adenylate cyclase activating polypeptide (PACAP, Adcyap1) activation of PAC1 receptors ( Adcyap1r1) significantly increases excitability of guinea pig cardiac neurons. This modulation of excitability is mediate...
TMPH-02997 Dps Protein, Mycobacterium smegmatis, Recombinant (His & SUMO) Mycobacterium smegmatis E. coli
Protects DNA from oxidative damage by sequestering intracellular Fe(2+) ion and storing it in the form of Fe(3+) oxyhydroxide mineral. One hydrogen peroxide oxidizes two Fe(2+) ions, which prevents hydroxyl radical produ...
TMPY-02949 AP2 Gamma/TFAP2C Protein, Human, Recombinant (His) Human E. coli
TFAP2C, also known as AP2-GAMMA, is a member of the activating protein 2 family of transcription factors. AP-2 factors bind to the consensus sequence 5'-GCCNNNGGC-3' and activate genes involved in a large spectrum of imp...
TMPJ-00886 ATF1 Protein, Human, Recombinant (His) Human E. coli
Cyclic AMP-dependent transcription factor ATF-1(ATF1) which contains 1 bZIP (basic-leucine zipper) domain and 1 KID (kinase-inducible) domain, belongs to the bZIP family. It influences cellular physiologic processes by r...
TMPH-01164 ATF-3 Protein, Human, Recombinant (His) Human E. coli
ATF3 Protein, Human, Recombinant (His) is expressed in E. coli.
TMPH-00794 Dps Protein, Helicobacter pylori, Recombinant (His & SUMO) Helicobacter pylori E. coli
Protects DNA from oxidative damage by sequestering intracellular Fe(2+) ion and storing it in the form of Fe(3+) oxyhydroxide mineral. One hydrogen peroxide oxidizes two Fe(2+) ions, which prevents hydroxyl radical produ...
TMPJ-01054 PAFAHB Protein, Human, Recombinant (His) Human E. coli
Platelet-Activating Factor Acetylhydrolase IB Subunit β (PAFAHB) is a cytoplasmic hydrolase. PAFAHB is a member of the GDSL lipolytic enzyme family. It also belongs to Platelet-activating factor acetylhydrolase IB beta/g...
TMPJ-01041 FGF-12 Protein, Human, Recombinant Human E. coli
Fibroblast Growth Factor 12 (FGF-12) is a member of the fibroblast growth factor (FGF) family. FGF-12 is probably involved in nervous system development and function. FGF-12 lacks the N-terminal signal sequence present i...
TMPH-00886 ATF7IP2 Protein, Human, Recombinant (His) Human E. coli
Recruiter that couples transcriptional factors to general transcription apparatus and thereby modulates transcription regulation and chromatin formation. Can both act as an activator or a repressor depending on the conte...
TMPJ-00120 NKp80/KLRF1 Protein, Human, Recombinant (His) Human Human Cells
Killer cell lectin-like receptor subfamily F member 1 (KLRF1) is known as NKp80. Human NKp80, a member of the C-type lectin family of proteins (1 - 3), is 231 aa in length with a 38 amino acid (aa) cytoplasmic region, a ...
TMPH-03274 ATF-4 Protein, Rat, Recombinant (His & Myc) Rat E. coli
Transcription factor that binds the cAMP response element (CRE) (consensus: 5'-GTGACGT[AC][AG]-3') and displays two biological functions, as regulator of metabolic and redox processes under normal cellular conditions, an...
TMPJ-00920 CD40 Ligand Protein, Mouse, Recombinant (aa 112-260, His) Mouse Human Cells
CD40 Ligand, also known as TNFSF5, CD154, is a type II transmembrane glycoprotein member of the TNF superfamily. Mature mouse CD40 Ligand consists of a 22 amino acid (aa) cytoplasmic domain, a transmembrane segment, and ...
TMPH-03740 DCL Protein, Bacillus subtilis, Recombinant (His) Bacillus subtilis E. coli
Catalyzes the first step in the D-alanylation of lipoteichoic acid (LTA), the activation of D-alanine and its transfer onto the D-alanyl carrier protein (Dcp) DltC. In an ATP-dependent two-step reaction, forms a high ene...
TMPJ-01442 SLAMF7 Protein, Rhesus macaque, Recombinant (His) Rhesus Macaque Human Cells
SLAMF7 is a single-pass type I membrane protein and contains 1 Ig-like C2-type (immunoglobulin-like) domain. SLAMF7 is expressed in NK cells, activated B-cells, NK-cell line but not in promyelocytic, B-cell lines, or T-c...
TMPJ-00083 NCR3 Protein, Human, Recombinant (hFc) Human Human Cells
Natural Cytotoxicity Triggering Receptor 3 (NCR3) along with NKp44 and NKp46 constitute a group of receptors termed “Natural Cytotoxicity Receptors”. They play a major role in triggering NK-mediated killing of most tumor...
TMPJ-00553 Lp-PLA2/PLA2G7 Protein, Human, Recombinant (aa 22-441, His) Human Human Cells
Platelet-Activating Factor Acetylhydrolase (PAFAH) is a secreted enzyme which belongs to the AB hydrolase superfamily and Lipase family and catalyzes the degradation of platelet-activating factor to biologically inactive...
TMPJ-00178 BAFF/TNFSF13B Protein, Human, Recombinant (His) Human Human Cells
TNFSF13B/TNFSF20 belongs to the tumor necrosis factor family. It abundantly is expressed in peripheral blood Leukocytes and is specifically expressed in monocytes and macrophages. Also found in the spleen, lymph node, bo...
TMPJ-00222 SLAMF7 Protein, Human, Recombinant (mFc) Human Human Cells
SLAMF7 is a single-pass type I membrane protein and contains 1 Ig-like C2-type (immunoglobulin-like) domain. SLAMF7 is expressed in NK cells, activated B-cells, NK-cell line but not in promyelocytic, B-cell lines, or T-c...
TMPJ-00221 SLAMF7 Protein, Human, Recombinant (His & Avi), Biotinylated Human Human Cells
SLAMF7 is a single-pass type I membrane protein and contains 1 Ig-like C2-type (immunoglobulin-like) domain. SLAMF7 is expressed in NK cells, activated B-cells, NK-cell line but not in promyelocytic, B-cell lines, or T-c...
TMPJ-00567 NCR1 Protein, Human, Recombinant (hFc) Human Human Cells
Natural cytotoxicity triggering receptor 1(NCR1) is a single-pass type I membrane protein .It contains 2 Ig-like (immunoglobulin-like) domains and belongs to the natural cytotoxicity receptor (NCR) family. The protein is...
TMPJ-00009 CCL2 Protein, Human, Recombinant Human E. coli
The chemokine (C-C motif) ligand 2 (CCL2), also known as monocyte chemoattractant protein (MCP)-1 and small inducible cytokine A2 (SCYA2)), is a small cytokine that belongs to the CC chemokine family responsible for mono...
TMPJ-00177 BAFF/TNFSF13B Protein, Human, Recombinant (Avi & hFc), Biotinylated Human Human Cells
B-cell activating factor (BAFF), also known as BLyS, TALL-1, THANK, and TNFSF13B, is a transmembrane glycoprotein in the TNF ligand superfamily. BAFF is a cytokine and serves as a ligand for receptors TNFRSF13B (TACI), T...
TMPH-02488 ACSS2 Protein, Mouse, Recombinant (His) Mouse E. coli
Catalyzes the synthesis of acetyl-CoA from short-chain fatty acids. Acetate is the preferred substrate but can also utilize propionate with a much lower affinity.
TMPH-01173 CDK7 Protein, Human, Recombinant Human E. coli
CDK7 Protein, Human, Recombinant is expressed in E. coli.
TMPH-01172 CDK7 Protein, Human, Recombinant (His) Human Baculovirus
CDK7 Protein, Human, Recombinant (His) is expressed in Baculovirus.
TMPH-02613 ATF-5 Protein, Mouse, Recombinant (His & Myc) Mouse E. coli
Transcription factor that either stimulates or represses gene transcription through binding of different DNA regulatory elements such as cAMP response element (CRE) (consensus: 5'-GTGACGT[AC][AG]-3'), ATF5-specific respo...
TMPJ-00097 NKG2D/CD314 Protein, Cynomolgus, Recombinant (hFc) Cynomolgus Human Cells
NKG2-D type II integral membrane protein (NKG2D) is a type II transmembrane glycoprotein which belongs to the CD94/NKG2 family. NKG2D is expressed on natural killer (NK) cells, CD8+ alpha-beta and gamma-delta T-cells. As...
TMPJ-00122 NKG2D/CD314 Protein, Mouse, Recombinant (His) Mouse Human Cells
NKG2-D type II integral membrane protein (NKG2D) is a type II transmembrane glycoprotein which belongs to the CD94/NKG2 family. NKG2D is expressed on natural killer (NK) cells, CD8+ alpha-beta and gamma-delta T-cells. As...
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Ubiquitin Activating Enzyme E1/UBA1 Protein, Human, Recombinant (His & GST)
TMPY-02840
Species: Human
Expression System: Baculovirus-Insect Cells
SAE1 Protein, Human, Recombinant
TMPY-03441
Species: Human
Expression System: Baculovirus-Insect Cells
FGF-9 Protein, Mouse, Recombinant (His)
TMPJ-01011
Species: Mouse
Expression System: E. coli
FGF-9 Protein, Human, Recombinant
TMPJ-00090
Species: Human
Expression System: E. coli
FLAP Protein, Human, Recombinant (His)
TMPY-01481
Species: Human
Expression System: Baculovirus-Insect Cells
UBA5 Protein, Human, Recombinant (His)
TMPJ-01324
Species: Human
Expression System: E. coli
BAFF/TNFSF13B Protein, Mouse, Recombinant (mFc)
TMPJ-01391
Species: Mouse
Expression System: Human Cells
SAE1 Protein, Human, Recombinant (His & GST)
TMPY-03062
Species: Human
Expression System: Baculovirus-Insect Cells
HABP2 Protein, Human, Recombinant (His)
TMPJ-01116
Species: Human
Expression System: Human Cells
CAK1 Protein, S. cerevisiae, Recombinant (His & Myc)
TMPH-03456
Species: Saccharomyces cerevisiae
Expression System: Baculovirus
SFP Protein, B.subtilis, Recombinant (His)
TMPJ-00611
Species: B.subtilis
Expression System: E. coli
ATF2 Protein, Human, Recombinant (His & GST)
TMPY-02444
Species: Human
Expression System: Baculovirus-Insect Cells
UBA6 Protein, Human, Recombinant (GST)
TMPY-06748
Species: Human
Expression System: Baculovirus-Insect Cells
CXCL5 Protein, Human, Recombinant (His)
TMPH-01163
Species: Human
Expression System: E. coli
CAK1 Protein, S. cerevisiae, Recombinant (E. coli, His & Myc)
TMPH-03457
Species: Saccharomyces cerevisiae
Expression System: E. coli
ACP Protein, S. aureus, Recombinant (His & SUMO)
TMPH-03520
Species: Staphylococcus aureus
Expression System: E. coli
4'-phosphopantetheinyl transferase ffp Protein, Bacillus subtilis, Recombinant (His & Myc)
TMPH-00164
Species: Bacillus subtilis
Expression System: E. coli
ACP Protein, E. coli, Recombinant (His & SUMO)
TMPH-00572
Species: E. coli
Expression System: E. coli
ACP Protein, S. aureus, Recombinant (GST)
TMPH-03518
Species: Staphylococcus aureus
Expression System: E. coli
NCR1 Protein, Mouse, Recombinant (hFc)
TMPJ-00425
Species: Mouse
Expression System: Human Cells
ACP Protein, S. aureus, Recombinant (His)
TMPH-03519
Species: Staphylococcus aureus
Expression System: Yeast
SLAMF6 Protein, Human, Recombinant (His & Avi), Biotinylated
TMPJ-00218
Species: Human
Expression System: Human Cells
PACAP receptor/ADCYAP1R1 Protein, Human, Recombinant (hFc)
TMPY-02648
Species: Human
Expression System: HEK293
Dps Protein, Mycobacterium smegmatis, Recombinant (His & SUMO)
TMPH-02997
Species: Mycobacterium smegmatis
Expression System: E. coli
AP2 Gamma/TFAP2C Protein, Human, Recombinant (His)
TMPY-02949
Species: Human
Expression System: E. coli
ATF1 Protein, Human, Recombinant (His)
TMPJ-00886
Species: Human
Expression System: E. coli
ATF-3 Protein, Human, Recombinant (His)
TMPH-01164
Species: Human
Expression System: E. coli
Dps Protein, Helicobacter pylori, Recombinant (His & SUMO)
TMPH-00794
Species: Helicobacter pylori
Expression System: E. coli
PAFAHB Protein, Human, Recombinant (His)
TMPJ-01054
Species: Human
Expression System: E. coli
FGF-12 Protein, Human, Recombinant
TMPJ-01041
Species: Human
Expression System: E. coli
ATF7IP2 Protein, Human, Recombinant (His)
TMPH-00886
Species: Human
Expression System: E. coli
NKp80/KLRF1 Protein, Human, Recombinant (His)
TMPJ-00120
Species: Human
Expression System: Human Cells
ATF-4 Protein, Rat, Recombinant (His & Myc)
TMPH-03274
Species: Rat
Expression System: E. coli
CD40 Ligand Protein, Mouse, Recombinant (aa 112-260, His)
TMPJ-00920
Species: Mouse
Expression System: Human Cells
DCL Protein, Bacillus subtilis, Recombinant (His)
TMPH-03740
Species: Bacillus subtilis
Expression System: E. coli
SLAMF7 Protein, Rhesus macaque, Recombinant (His)
TMPJ-01442
Species: Rhesus Macaque
Expression System: Human Cells
NCR3 Protein, Human, Recombinant (hFc)
TMPJ-00083
Species: Human
Expression System: Human Cells
Lp-PLA2/PLA2G7 Protein, Human, Recombinant (aa 22-441, His)
TMPJ-00553
Species: Human
Expression System: Human Cells
BAFF/TNFSF13B Protein, Human, Recombinant (His)
TMPJ-00178
Species: Human
Expression System: Human Cells
SLAMF7 Protein, Human, Recombinant (mFc)
TMPJ-00222
Species: Human
Expression System: Human Cells
SLAMF7 Protein, Human, Recombinant (His & Avi), Biotinylated
TMPJ-00221
Species: Human
Expression System: Human Cells
NCR1 Protein, Human, Recombinant (hFc)
TMPJ-00567
Species: Human
Expression System: Human Cells
CCL2 Protein, Human, Recombinant
TMPJ-00009
Species: Human
Expression System: E. coli
BAFF/TNFSF13B Protein, Human, Recombinant (Avi & hFc), Biotinylated
TMPJ-00177
Species: Human
Expression System: Human Cells
ACSS2 Protein, Mouse, Recombinant (His)
TMPH-02488
Species: Mouse
Expression System: E. coli
CDK7 Protein, Human, Recombinant
TMPH-01173
Species: Human
Expression System: E. coli
CDK7 Protein, Human, Recombinant (His)
TMPH-01172
Species: Human
Expression System: Baculovirus
ATF-5 Protein, Mouse, Recombinant (His & Myc)
TMPH-02613
Species: Mouse
Expression System: E. coli
NKG2D/CD314 Protein, Cynomolgus, Recombinant (hFc)
TMPJ-00097
Species: Cynomolgus
Expression System: Human Cells
NKG2D/CD314 Protein, Mouse, Recombinant (His)
TMPJ-00122
Species: Mouse
Expression System: Human Cells
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Cat No. Product Name
L1300 PI3K-AKT-mTOR Compound Library

425 compounds
A unique collection of 425 compounds targeting PI3K/Akt/mTOR signaling for research in PI3K/Akt/mTOR signaling, and drug discovery in diseases involved with PI3K/Akt/mTOR signaling;
L8600 Ubiquitination Compound Library

214 compounds
A unique collection of 214 ubiquitination related small chemicals can be used for high throughput and high content screening；
L8720 Pyroptosis Compound Library

1077 compounds
1077 types of active small molecules associated with pyroptosis for high-throughput and high-content screening.
L6750 PBCRBS Traditional Chinese Medicine Compound Library

588 compounds
A unique collection of 588 compounds derived from traditional Chinese medicines (TCMs) for promoting blood circulation and removing blood stasis.

Libraries

PI3K-AKT-mTOR Compound Library
L1300
Compounds: 425
Ubiquitination Compound Library
L8600
Compounds: 214
Pyroptosis Compound Library
L8720
Compounds: 1077
PBCRBS Traditional Chinese Medicine Compound Library
L6750
Compounds: 588
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