vmat2 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T24941	VMAT2-IN-I HCl	VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride
	VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A.
T79061	VMAT2-IN-2 tosylate		Monoamine Transporter
	VMAT2-IN-2 tosylate is a potent inhibitor of VMAT2 and is applicable in the research of tardive dyskinesia [1].		Monoamine Transporter
T7147	Valbenazine	NBI-98854	Monoamine Transporter
	Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.		Monoamine Transporter
T0719	Tetrabenazine	Xenazine,Ro 1-9569	Others , Dopamine Receptor , Monoamine Transporter
	Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders. Tetrabenazine blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high...		Others , Dopamine Receptor , Monoamine Transporter
T7563	NBI-98782	(+)-α-Dihydrotetrabenazine,(+)-α-DHTBZ,(+)-DTBZ	Monoamine Transporter
	NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)		Monoamine Transporter
T13133	Tetrabenazine Metabolite	(-)-β-Dihydrotetrabenazine,(-)-β-HTBZ	Monoamine Transporter
	Tetrabenazine Metabolite ((-)-β-HTBZ), a vesicles monoamine transporter 2 (VMAT2) inhibitor, is an active metabolite of Tetrabenazine. Tetrabenazine Metabolite has a high affinity for VMAT2 with a Ki of 13.4 nM. Tetraben...		Monoamine Transporter
T41195	FFN 206 dihydrochloride
	FFN 206 dihydrochloride is a fluorescent VMAT2 substrate that can be used to detect VMAT2 subcellular sites in cell culture and shows no detectable inhibition of DAT.
T13134	(+)-Tetrabenazine	(+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ	Monoamine Transporter
	(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1.		Monoamine Transporter
T41194	FFN 102 mesylate		Others
	FFN 102 mesylate is a pH responsive fluorescent false neurotransmitter (FFN), a selective dopamine transporter (DAT) and VMAT2 substrate. Exhibits no significant binding to a panel of 38 CNS receptors, including dopamine...		Others
T77549	Nurr1 agonist 2		Others
	Nurr1 agonist 2 is a Nurr1 agonist with an EC50 value of 0.07 μM. Nurr1 agonist 2 increases the mRNA expression of the Nurr1-regulated genes tyrosine hydroxylase (TH) and vesicular amino acid transporter 2 (VMAT2). Nurr1...		Others
T22452	Valbenazine tosylate	NBI-98854	Monoamine Transporter
	Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM).		Monoamine Transporter
T25750	Lobelane Hydrochloride
	Lobelane Hydrochloride is a vesicular monoamine transporter-2 (VMAT2) inhibitor.
T31791	FFN246 HCl	FFN 246,FFN246 hydrochloride,FFN246,FFN-246
	FFN246 is a fluorescent substrate for both the serotonin transporter and the vesicular monoamine transporter 2 (VMAT2).
T31790	FFN200 dihydrochloride	FFN200 HCl,FFN200,FFN 200,FFN-200
	FFN200 is a vesicular monoamine transporter 2 (VMAT2) substrate that selectively traces monoamine exocytosis in both neuronal cell culture and brain tissue.
T70322	Valbenazine dihydrochloride
	Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.
T12190	Trans (2,3)-Dihydrotetrabenazine	(2R,3R,11bR)-rel-DHTBZ,(2R,3R,11bR)-rel-Dihydrotetrabenazine	Others
	Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2).		Others
T23983	Deutetrabenazine metabolite M4	SD-1018,Deuterated monohydroxy tetrabenazine,D6-tetrabenazine metabolite M4
	Deutetrabenazine metabolite M4 is believed to be related to its effect as a reversible depletion of monoamines from nerve terminals. The major circulating metabolites of Deutetrabenazine, are reversible inhibitors of VM...
T78684	FFN246		5-HT Receptor
	FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation and emission spectra at 392/427 nm, respectively. It serves to label...		5-HT Receptor
T41193	FFN 270
	FFN 270 is a fluorescent false neurotransmitter (FFN). Fluorescent substrate for NET and VMAT2. Labels noradrenergic neurons and their synaptic vesicles, and enables imaging of synaptic vesicle content release from speci...