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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15411 | GPNA hydrochloride | Apoptosis , Others | |
GPNA hydrochloride is specific glutamine (Gln) transporter ASCT2(SLC1A5) inhibitor. GPNA reversibly induces apoptosis in A549 cells. GPNA hydrochloride is a well-known substrate of the enzyme γ-glutamyltransferase (GGT).... | |||
T5345 | V-9302 | Others | |
V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uM). | |||
T21102 | L-4FPG | L4FPG,L 4FPG | Others |
L-4FPG is a Glycine derivative, inhibits the neutral amino acid transporters ASCT1 and ASCT2. | |||
T77385 | Idactamab | INT-001 | |
Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2. | |||
T60642 | SN40 | ||
SN40 is a potent amino acid transport (AAT) inhibitor that can be used in anticancer research. SN40 has Kis of 7.29 μM, 2.42 μM, 2.94 μM, 5.55 μM, 24.43 μM and 5.55 μM for human ASCT1, rat ASCT2, human ASCT2, EAAT1, EAAT... | |||
T40064 | V-9302 hydrochloride | ||
V-9302 hydrochloride is a potent and selective competitive antagonist that inhibits transmembrane glutamine flux by specifically targeting the amino acid transporter ASCT2 (SLC1A5), and not ASCT1. In HEK-293 cells, V-930... | |||
T60768 | SN05 | ||
SN05 is a potent inhibitor of amino acid transport (AAT) that can be used in anticancer research. The Ki values of SN05 for human ASCT1, rat ASCT2, human ASCT2, EAAT1, EAAT2, EAAC1 and EAAT5 is 2.77 μM, 0.73 μM, 0.87 μM,... | |||
T31824 | Fluoroglutamine (2S,4R) | FDG | |
Fluoroglutamine (2S,4R) is a Glutamine analog, not metabolized in the TCA cycle, but it can be incorporated into proteins and peptides. Fluoroglutamine (2S,4R) can be used as assess transporter (ASCT2) activity or protei... |