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Search Results for " vasopressin-receptor "

Targets

60

Compounds

2

Recombinant Proteins

1

Libraries

Cat No. Product Name Synonyms Targets
T14494 Balovaptan RG7314 Vasopressin Receptor
Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors. It is used for the research of autism.
T64174 Vasopressin V2 receptor antagonist 1
Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD).
T6288 Mozavaptan OPC31260l,OPC-31260 Vasopressin Receptor
Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
T4355 Fuscoside OPC 21268 Vasopressin Receptor
Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
T11857 LIT-001 Oxytocin Receptor
LIT-001 improves social interaction in a mouse model of autism.It is the first nonpeptide oxytocin receptor agonist with EC50 of 55 nM and Ki of 226 nM.
T13920L Terlipressin Acetate Terlipressin diacetate anhydrous,Terlipressin acetate anhydrous Vasopressin Receptor
Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelial cells (IEC-6).Terlipressin acetate exerts anti-in...
T5148 Atosiban acetate RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164 Oxytocin Receptor , Vasopressin Receptor
Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban acetate (RW22164) inhibits...
T2326 Tolvaptan OPC-41061 Vasopressin Receptor , Autophagy
Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
T7303 LIXIVAPTAN VPA-985,WAY-VPA 985 Vasopressin Receptor
Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
T6453 Conivaptan hydrochloride Vaprisol,Conivaptan HCl,YM 087 Vasopressin Receptor
Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
T7434 Argipressin Arg8-vasopressin,Vasopressin,AVP Vasopressin Receptor
Argipressin (Vasopressin) is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth ...
T2568 Felypressin Octapressin,Felypressin Acetate,PLV-2,H-[Cys-Phe-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2 Vasopressin Receptor
Felypressin (Octapressin) is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activity.
T2568L Felypressin acetate 2-(L-Phenylalanine)-8-L-lysinevasopressin,PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond),PLV 2,PLV-2 Vasopressin Receptor
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.
T4996 Atosiban RWJ22164,RW22164 Oxytocin Receptor , Vasopressin Receptor
Atosiban (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban inhibits the oxytocin-mediated rel...
T4141 RG7713 RO 5028442 Vasopressin Receptor
RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.
T21308 Histrelin Supprelin LA,Histrelin Acetate Others
Histrelin (Supprelin LA) acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It is considered a GnRH agonist. Histrelin is used in the treatment of hormone-sensitive cancers of th...
T28153 Nelivaptan SSR149415,SR 149415,SR-149415 Vasopressin Receptor
Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist.
T7284 Argipressin acetate (113-79-1(free base)) Others
Vasopressin acetate is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth muscle...
T15682 L-371,257 Oxytocin Receptor , Vasopressin Receptor
L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.
T5144 Desmopressin acetate (16679-58-6 free base) Desmopressin acetate,DDAVP Vasopressin Receptor
Desmopressin acetate (16679-58-6 free base) (DDAVP) is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led to its use in polyur...
T15273 Fedovapagon VA483,A106483 Vasopressin Receptor
Fedovapagon (VA106483) is a selective and potent agonist of the vasopressin V2 receptor (V2R) that inhibits the growth of intersegmental vessels in zebrafish. Fedovapagon can be used to study overactive bladder, nocturia...
TP1192L Conopressin S acetate(111317-90-9 free base) Con-S acetate Vasopressin Receptor
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
TP1927L1 D[Leu4,Lys8]-VP acetate d[Leu4,Lys8]-VP acetate(42061-33-6 free base) Vasopressin Receptor
d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respectively. d[Leu4,Lys8]-VP acetate exhibits weak antidiuretic...
TP2082L D[Cha4]-AVP acetate(500170-27-4 free base) Vasopressin Receptor
d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secre...
T23393 SR 49059 Others
vasopressin V1A receptor antagonist
T28745 Selepressin FE 202158,FE202158
Selepressin, an analog of vasopressin, is a potent, selective vasopressin V1a receptor agonist.
T28629 RWJ 676070 RWJ676070,RWJ-676070
RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.
T29085 VA-111913 VA111913,VA 111913
VA-111913, a vasopressin receptor antagonist, is used potentially for the treatment of dysmenorrhea.
T70066 Pecavaptan
Pecavaptan is a vasopressin receptor antagonist.
T21465 Mozavaptan hydrochloride OPC-31260,OPC31260,Mozavaptan HCl,OPC 31260
Mozavaptan is a vasopressin receptor antagonist.
T34325 Ribuvaptan
Ribuvaptan is a antagonist of vasopressin receptor .
T29177 YM 218 YM218,YM-218
YM 218 is a novel, potent, selective antagonist of nonpeptide vasopressin V1A receptor.
T76509 Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), is a weak agonist at antidiuretic receptor . However, Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin is a potent agonist at pit...
T39611 Enuvaptan Enuvaptan,BAY-2327949
Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.
T29178 YM 471 YM-471,YM471
YM 471 is a non-peptide arginine vasopressin (AVP) V1A and V2 receptor antagonist with oral activity.
T24759 Satavaptan fumarate SR-121463A,SR 121463 A,SR-121463 A,SR121463A
Satavaptan fumarate is a selective antagonist of the non-peptide vasopressin V2 receptor.
T76633 (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin is a potent vasopressin V1 receptor (VP V1R) antagonist. (Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin significantly decreases the mean arterial pressure (MAP...
T27965 M-0002 RWJ-351647,SPD556,SPD-556,M0002,RWJ351647
M-0002, a vasopressin V2 receptor antagonist, is used potentially for the treatment of ascites.
T28664 Satavaptan SR121463,SR 121463,SR-121463
Satavaptan is a vasopressin V2 receptor antagonist. Satavaptan improves the control of ascites in cirrhosis.
T28854 SRX 251 SRX-251,SRX251
SRX 251, a vasopressin V1a receptor antagonist, is used potentially for the treatment of primary dysmenorrhea.
T80073 Dp[Tyr(methyl)2,Arg8]-Vasopressin Vasopressin Receptor
Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].
TP2136 (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonge...
T79173 PF-06478939 Oxytocin Receptor
PF-06478939 is a peptide that functions as an agonist at the oxytocin (OT) receptor and vasopressin receptor without crossing the blood-brain barrier. It exhibits EC50 values of 0.01 nM at the OT receptor and 0.078 nM at...
T24370 L-368899 free base L 368899,L 368,899,L368,899,L-368899,L368899,L-368,899
L-368899 is a non-peptide and orally active antagonist of oxytocin receptor (IC50: 8.9 nM). It displays 40-fold selectivity over vasopressin V1a and V2 receptors (IC50: 370 and 570 nM respectively).
T17251 VNA-932 WAY-VNA 932 Others
VNA-932 is an agonist of the vasopressin V2-receptor (IC50: 80.3 nM and 778 nM in human-V2 binding and V1a binding assay).
T30275 Azilsartan trimethylethanolamine Azilsartan,TAK-536
Azilsartan is an angiotensin II receptor antagonist for the treatment of hypertension and was developed by Takeda. Azilsartan Medoxomil lowers blood pressure by blocking the effects of angiotensin II, a type of vasopress...
T62906 Lazuvapagon
Lazuvapagon is a vasopressin V2 receptor agonist that can be used to study enuresis.
T80270 Invopressin OCE-205 Vasopressin Receptor
Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial peritonitis, HRS2, and refractory ascites [1].
T80137 (d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin d(CH2)5[Tyr(Me)2, Dab5]AVP Vasopressin Receptor
(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].
TP1192 Conopressin S Con-S
Conopressin S, isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.

Compounds

Balovaptan
T14494
Synonym: RG7314
Target: Vasopressin Receptor
Vasopressin V2 receptor antagonist 1
T64174
Synonym:
Target:
Mozavaptan
T6288
Synonym: OPC31260l,OPC-31260
Target: Vasopressin Receptor
Fuscoside
T4355
Synonym: OPC 21268
Target: Vasopressin Receptor
LIT-001
T11857
Synonym:
Target: Oxytocin Receptor
Terlipressin Acetate
T13920L
Synonym: Terlipressin diacetate anhydrous,Terlipressin acetate anhydrous
Target: Vasopressin Receptor
Atosiban acetate
T5148
Synonym: RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164
Target: Oxytocin Receptor, Vasopressin Receptor
Tolvaptan
T2326
Synonym: OPC-41061
Target: Vasopressin Receptor, Autophagy
LIXIVAPTAN
T7303
Synonym: VPA-985,WAY-VPA 985
Target: Vasopressin Receptor
Conivaptan hydrochloride
T6453
Synonym: Vaprisol,Conivaptan HCl,YM 087
Target: Vasopressin Receptor
Argipressin
T7434
Synonym: Arg8-vasopressin,Vasopressin,AVP
Target: Vasopressin Receptor
Felypressin
T2568
Synonym: Octapressin,Felypressin Acetate,PLV-2,H-[Cys-Phe-Phe-Gln-Asn-Cys]-Pro-Lys-Gly-NH2
Target: Vasopressin Receptor
Felypressin acetate
T2568L
Synonym: 2-(L-Phenylalanine)-8-L-lysinevasopressin,PLV2. H-Cys-Phe-Phe-Gln-Asn-Cys-Pro-Lys-Gly-NH2 (Disulfide bond),PLV 2,PLV-2
Target: Vasopressin Receptor
Atosiban
T4996
Synonym: RWJ22164,RW22164
Target: Oxytocin Receptor, Vasopressin Receptor
RG7713
T4141
Synonym: RO 5028442
Target: Vasopressin Receptor
Histrelin
T21308
Synonym: Supprelin LA,Histrelin Acetate
Target: Others
Nelivaptan
T28153
Synonym: SSR149415,SR 149415,SR-149415
Target: Vasopressin Receptor
Argipressin acetate (113-79-1(free base))
T7284
Synonym:
Target: Others
L-371,257
T15682
Synonym:
Target: Oxytocin Receptor, Vasopressin Receptor
Desmopressin acetate (16679-58-6 free base)
T5144
Synonym: Desmopressin acetate,DDAVP
Target: Vasopressin Receptor
Fedovapagon
T15273
Synonym: VA483,A106483
Target: Vasopressin Receptor
Conopressin S acetate(111317-90-9 free base)
TP1192L
Synonym: Con-S acetate
Target: Vasopressin Receptor
d[Leu4,Lys8]-VP acetate
TP1927L1
Synonym: d[Leu4,Lys8]-VP acetate(42061-33-6 free base)
Target: Vasopressin Receptor
d[Cha4]-AVP acetate(500170-27-4 free base)
TP2082L
Synonym:
Target: Vasopressin Receptor
SR 49059
T23393
Synonym:
Target: Others
Selepressin
T28745
Synonym: FE 202158,FE202158
Target:
RWJ 676070
T28629
Synonym: RWJ676070,RWJ-676070
Target:
VA-111913
T29085
Synonym: VA111913,VA 111913
Target:
Pecavaptan
T70066
Synonym:
Target:
Mozavaptan hydrochloride
T21465
Synonym: OPC-31260,OPC31260,Mozavaptan HCl,OPC 31260
Target:
Ribuvaptan
T34325
Synonym:
Target:
YM 218
T29177
Synonym: YM218,YM-218
Target:
Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
T76509
Synonym:
Target:
Enuvaptan
T39611
Synonym: Enuvaptan,BAY-2327949
Target:
YM 471
T29178
Synonym: YM-471,YM471
Target:
Satavaptan fumarate
T24759
Synonym: SR-121463A,SR 121463 A,SR-121463 A,SR121463A
Target:
(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
T76633
Synonym:
Target:
M-0002
T27965
Synonym: RWJ-351647,SPD556,SPD-556,M0002,RWJ351647
Target:
Satavaptan
T28664
Synonym: SR121463,SR 121463,SR-121463
Target:
SRX 251
T28854
Synonym: SRX-251,SRX251
Target:
Dp[Tyr(methyl)2,Arg8]-Vasopressin
T80073
Synonym:
Target: Vasopressin Receptor
(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
TP2136
Synonym:
Target:
PF-06478939
T79173
Synonym:
Target: Oxytocin Receptor
L-368899 free base
T24370
Synonym: L 368899,L 368,899,L368,899,L-368899,L368899,L-368,899
Target:
VNA-932
T17251
Synonym: WAY-VNA 932
Target: Others
Azilsartan trimethylethanolamine
T30275
Synonym: Azilsartan,TAK-536
Target:
Lazuvapagon
T62906
Synonym:
Target:
Invopressin
T80270
Synonym: OCE-205
Target: Vasopressin Receptor
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
T80137
Synonym: d(CH2)5[Tyr(Me)2, Dab5]AVP
Target: Vasopressin Receptor
Conopressin S
TP1192
Synonym: Con-S
Target:
1 2

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPH-02818 Osteocalcin Protein, Mouse, Recombinant (His & SUMO) Mouse E. coli
Receptor for arginine vasopressin. The activity of this receptor is mediated by G proteins which activate adenylate cyclase. Involved in renal water reabsorption.
TMPH-01589 KIR2DS3 Protein, Human, Recombinant (His) Human Yeast
Secreted polyprotein that is packaged and proteolytically processed by prohormone convertases PCSK1 and PCSK2 in a cell-type-specific manner. VGF and peptides derived from its processing play many roles in neurogenesis a...
Cat No. Product Name
L7110 Anti-Hypertension Compound Library

719 compounds
719 hypertension-related small molecules for high-throughput and high-content screening.
TargetMol