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GPCR/G Protein Vasopressin Receptor

Vasopressin Receptor

The actions of vasopressin are mediated by stimulation of tissue-specific G protein-coupled receptors (GPCRs) called vasopressin receptors that are classified into the V1 (V1A), V2, and V3 (V1B) receptor subtypes. These three subtypes differ in localization, function and signal transduction mechanisms.
Cat No. product name
TP2082L D[Cha4]-AVP acetate(500170-27-4 free base) d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 recept...
TP1192L Conopressin S acetate(111317-90-9 free base) Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
TP1192L Conopressin S acetate(111317-90-9 free base) Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
T13920L Terlipressin Acetate Terlipressin, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelia...
T14494 Balovaptan Balovaptan is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) ...
T7303 LIXIVAPTAN Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
T5144 Desmopressin acetate (16679-58-6 free base) Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led ...
T5019 Desmopressin Desmopressin(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic properties of desmopressin h...
T4141 RO 5028442 RO5028442 has been used in trials studying Autistic Disorder.
T4355 OPC 21268 OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
T2568 Felypressin Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activit...
T6453 Conivaptan hydrochloride Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
T2326 Tolvaptan Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
T6288 Mozavaptan Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
d[Cha4]-AVP acetate(500170-27-4 free base)
TP2082LCAS TP2082L
d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 recept...
Conopressin S acetate(111317-90-9 free base)
TP1192LCAS TP1192L
Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
Conopressin S acetate(111317-90-9 free base)
TP1192LCAS TP1192L
Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
Terlipressin Acetate
T13920LCAS 1884420-36-3
Terlipressin, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelia...
Balovaptan
T14494CAS 1228088-30-9
Balovaptan is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) ...
LIXIVAPTAN
T7303CAS 168079-32-1
Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
Desmopressin acetate (16679-58-6 free base)
T5144CAS 62288-83-9
Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led ...
Desmopressin
T5019CAS 16679-58-6
Desmopressin(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic properties of desmopressin h...
RO 5028442
T4141CAS 920022-47-5
RO5028442 has been used in trials studying Autistic Disorder.
OPC 21268
T4355CAS 131631-89-5
OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
Felypressin
T2568CAS 56-59-7
Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activit...
Conivaptan hydrochloride
T6453CAS 168626-94-6
Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
Tolvaptan
T2326CAS 150683-30-0
Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
Mozavaptan
T6288CAS 137975-06-5
Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.