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Search Result

Search Results for " glucagon-receptor "

109

Compounds

2

Natural Products

9

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T37223 Glucagon Receptor Antagonist I
Glucagon receptor antagonist I is a competitive antagonist of the glucagon receptor (GCGR; IC50 = 181 nM). It blocks glucagon-induced glycogenolysis in primary human hepatocytes and isolated liver. Glucagon receptor anta...
T36580 Glucagon Receptor Antagonist Inactive Control
Glucagon Receptor Antagonist Inactive Control is a Glucagon receptor antagonist that can be used in related research in the field of life sciences. Its product number is T36580 and CAS number is 362482-00-6.
T11416 Glucagon receptor antagonists-5 Others
Glucagon receptor antagonists-5 is an orally bioavailable indazole-based glucagon receptor antagonist (Ki: 32 nM). It has potential for the treatment of type 2 diabetes mellitus (T2DM).
T11415 Glucagon receptor antagonists-3 Others
Glucagon receptor antagonist -3 is a highly effective glucagon receptor antagonist.
T11414 Glucagon receptor antagonists-2 Others
Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist.
T11413 Glucagon receptor antagonists-1 Others
Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.
TQ0239 PF-06291874 Glucagon receptor antagonists-4 Glucagon Receptor
PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
T15389L Glucagon (1-29), bovine, human, porcine hydrochloride Porcine glucagon hydrochloride,Glucagon hydrochloride Glucocorticoid Receptor , Glucagon Receptor
Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. It activates HNF4α and increases HNF4α phosphorylation. Glucagon (1-29), bovine, human, porcine hydrochloride(Po...
TQ0124 BETP Glucagon Receptor
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
T11845 LGD-6972 Glucagon Receptor
LGD-6972 is an antagonist of glucagon receptor.
T9579 GLP-1 receptor agonist 9 Glucagon Receptor
1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
T7364 NNC-0640 Glucagon Receptor
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
T8748 Exendin-4 acetate Glucagon Receptor
Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).
T3984 GLP-1(7-36), amide MKC 253,Human GLP-1-(7-36)-amide,Glucagon-like Peptide 1 (7-36) amide,Glucagon-Like Peptide (GLP) I (7-36), amide, human,GLP-1(7-36),GLP-1-(7-36)-amide Glucagon Receptor
GLP-1(7-36), amide (MKC 253) is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays various antidiabetic effects by potentiating glucose-...
T19850 Semaglutide Glucagon Receptor
Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
TP2252 GLP-1 (9-36) amide Glucagon Receptor
antagonist at the human GLP-1 receptor
T3422 GRA Ex-25 GRA-Ex-25 Glucagon Receptor
GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.
T3967 Exendin-4 Exenatide,Exenatide Acetate Glucagon Receptor
Exendin-4 (Exenatide) is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer half-life of 2.4 hours.
TP1039 Secretin (33-59), rat Secretin (rat) Glucagon Receptor
Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.
TP1469 Lixisenatide acetate (320367-13-3 free base) Lixisenatide acetate Glucagon Receptor
Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
T6876 Liraglutide Liraglutidum,Victoza,Liraglutida,NN2211 Glucagon Receptor
Liraglutide (Liraglutida) is a long-acting GLP-1 receptor agonist.
TP2100 Avexitide Exendin-3 (9-39) amide,Exendin (9-39) Glucagon Receptor
Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.
TP1376 GLP-1(7-37) acetate(106612-94-6 free base) GLP-1(7-37) acetate Others , Glucagon Receptor
Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.
T60047 V-0219 Glucagon Receptor
V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.
TP1103 Cotadutide acetate MEDI0382 acetate,Cotadutide acetate (1686108-82-6 Free base) Glucagon Receptor
Cotadutide acetate (MEDI0382 acetate) is a potent peptide dual agonist of glucagon-like peptide-1 (GLP-1) and glucagon receptor with EC50 of 6.9 pM and 10.2 pM, respectively.
T22893 L-168049 L-168,049 Glucagon Receptor
L-168049 is a selective and non-competitive antagonist of human glucagon receptor with IC50s of 3.7 nM, 63 nM, and 60 nM for human, murine, and canine, respectively.
T76559 Survodutide BI 456906 Glucagon Receptor
Survodutide (BI 456906) is a dual agonist of glucagon and glucagon-like peptide 1 (GLP-1) receptor (GLP Receptor) that reduces body weight in HbA1c16 diabetes.
T28182 NNC 92-1687 NNC92-1687,NNC-92-1687 Glucagon Receptor
NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.
T76279 Retatrutide LY3437943 Glucagon Receptor
Retatrutide (LY3437943) is a triple agonist of the glucagon receptor, glucose-dependent insulinotropic polypeptide receptor, and glucagon-like peptide-1 receptor (GLP-1R), and inhibits GCGR, GIPR, and GLP-1R.Retatrutide ...
T76279L1 Retatrutide sodium salt Retatrutide sodium salt(2381089-83-2 free base),LY3437943 sodium salt Glucagon Receptor
Retatrutide sodium salt is a potent triple agonist peptide for glucagon receptor (GCGR), glucose-dependent proinsulinotropic polypeptide receptor (GIPR), and glucagon-like peptide-1 receptor (GLP-1R) Retatrutide sodium s...
T8355 Exenatide Exendin-4,Extendin-4 Glucagon Receptor
Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.
T60047L V-0219 hydrochloride V-0219 hydrochloride（878453-71-5 Free base） Glucagon Receptor
V-0219 hydrochloride, an orally-active positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R), is utilized in obesity-associated diabetes research.
T11408 Orforglipron LY3502970,GLP-1 receptor agonist 1 Glucagon Receptor
Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1 diabetes in adults.
T12431 PF-06882961 Glucagon Receptor
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
T19850L Semaglutide Acetate Semaglutide Acetate(910463-68-2 Free base) Glucagon Receptor
Semaglutide Acetate is an agonist of a glucagon-like peptide 1 (GLP-1) receptor and can be used in studies about the treatment of type 2 diabetes.
T36579 GLP-1R Agonist DMB Glucagon Receptor
GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).
T8876 PF-06882961 Tris UNII-2HJV78O0SS Glucagon Receptor
PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
TP1976L Oxyntomodulin acetate Glucagon Receptor
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
T14130 Adomeglivant LY2409021 Glucagon Receptor
Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.
TP2100L Avexitide acetate Exendin 9-39 acetate,Avexitide acetate（133514-43-9 Free base） Glucagon Receptor
Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.
T63166L (S, R)-LSN 3318839 (S, R)-LSN 3318839(Isomer-2764704-18-7) Glucagon Receptor
(S, R)-LSN 3318839 is an allosteric modulator of the glucagon-like peptide-3318839 receptor (GLP-1R) that has demonstrated powerful hypoglycemic effects in animal models alone or in combination with sitagliptin.
T78097L Mazdutide acetate（2259884-03-0 free base） Mazdutide acetate（2259884-03-0 free base）,OXM-3 acetate,LY-3305677 acetate,IBI-362 acetate Glucagon Receptor
Mazdutide acetate is a potent co-agonist of glucagon-like peptide (GLP-1R) and glucagon receptor (GCGR), a gastrin-regulating hormone analog.Mazdutide acetate stimulates insulin secretion from mouse pancreatic islets, an...
T15387 GLP-1R Antagonist 1 Glucagon Receptor
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).
T63166 LSN3318839 LSN-3318839,LSN 3318839 Glucagon Receptor
LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can be used to lower blood glucose.
TP1111 Tirzepatide LY-3298176 Glucagon Receptor
Tirzepatide (LY-3298176) is a dual agonist of glucose-dependent polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor with neuroprotective activity for the study of diabetes and obesity.
T12055 MK 0893 Others
MK 0893 is a potent, selective antagonist of glucagon receptor.
T28057 MK3577 MK-3577,MK 3577
MK3577 is a glucagon receptor antagonist.
T30299 BAY-27-9955 BAY 279955,BAY27-9955,BAY-279955,BAY 27-9955
BAY-27-9955 is a glucagon receptor antagonist.
T25711 LGD-6972 sodium LGD 6972 sodium
LGD-6972 sodium is a glucagon receptor antagonist.
T70279 Cotadutide
Cotadutide is a dual receptor agonist that modifies the activity of glucagon and glucagon-like peptide-1 (GLP-1).

Compounds

Glucagon Receptor Antagonist I
T37223
Synonym:
Target:
Glucagon Receptor Antagonist Inactive Control
T36580
Synonym:
Target:
Glucagon receptor antagonists-5
T11416
Synonym:
Target: Others
Glucagon receptor antagonists-3
T11415
Synonym:
Target: Others
Glucagon receptor antagonists-2
T11414
Synonym:
Target: Others
Glucagon receptor antagonists-1
T11413
Synonym:
Target: Others
PF-06291874
TQ0239
Synonym: Glucagon receptor antagonists-4
Target: Glucagon Receptor
Glucagon (1-29), bovine, human, porcine hydrochloride
T15389L
Synonym: Porcine glucagon hydrochloride,Glucagon hydrochloride
Target: Glucocorticoid Receptor, Glucagon Receptor
BETP
TQ0124
Synonym:
Target: Glucagon Receptor
LGD-6972
T11845
Synonym:
Target: Glucagon Receptor
GLP-1 receptor agonist 9
T9579
Synonym:
Target: Glucagon Receptor
NNC-0640
T7364
Synonym:
Target: Glucagon Receptor
Exendin-4 acetate
T8748
Synonym:
Target: Glucagon Receptor
GLP-1(7-36), amide
T3984
Synonym: MKC 253,Human GLP-1-(7-36)-amide,Glucagon-like Peptide 1 (7-36) amide,Glucagon-Like Peptide (GLP) I (7-36), amide, human,GLP-1(7-36),GLP-1-(7-36)-amide
Target: Glucagon Receptor
Semaglutide
T19850
Synonym:
Target: Glucagon Receptor
GLP-1 (9-36) amide
TP2252
Synonym:
Target: Glucagon Receptor
GRA Ex-25
T3422
Synonym: GRA-Ex-25
Target: Glucagon Receptor
Exendin-4
T3967
Synonym: Exenatide,Exenatide Acetate
Target: Glucagon Receptor
Secretin (33-59), rat
TP1039
Synonym: Secretin (rat)
Target: Glucagon Receptor
Lixisenatide acetate (320367-13-3 free base)
TP1469
Synonym: Lixisenatide acetate
Target: Glucagon Receptor
Liraglutide
T6876
Synonym: Liraglutidum,Victoza,Liraglutida,NN2211
Target: Glucagon Receptor
Avexitide
TP2100
Synonym: Exendin-3 (9-39) amide,Exendin (9-39)
Target: Glucagon Receptor
GLP-1(7-37) acetate(106612-94-6 free base)
TP1376
Synonym: GLP-1(7-37) acetate
Target: Others, Glucagon Receptor
V-0219
T60047
Synonym:
Target: Glucagon Receptor
Cotadutide acetate
TP1103
Synonym: MEDI0382 acetate,Cotadutide acetate (1686108-82-6 Free base)
Target: Glucagon Receptor
L-168049
T22893
Synonym: L-168,049
Target: Glucagon Receptor
Survodutide
T76559
Synonym: BI 456906
Target: Glucagon Receptor
NNC 92-1687
T28182
Synonym: NNC92-1687,NNC-92-1687
Target: Glucagon Receptor
Retatrutide
T76279
Synonym: LY3437943
Target: Glucagon Receptor
Retatrutide sodium salt
T76279L1
Synonym: Retatrutide sodium salt(2381089-83-2 free base),LY3437943 sodium salt
Target: Glucagon Receptor
Exenatide
T8355
Synonym: Exendin-4,Extendin-4
Target: Glucagon Receptor
V-0219 hydrochloride
T60047L
Synonym: V-0219 hydrochloride（878453-71-5 Free base）
Target: Glucagon Receptor
Orforglipron
T11408
Synonym: LY3502970,GLP-1 receptor agonist 1
Target: Glucagon Receptor
PF-06882961
T12431
Synonym:
Target: Glucagon Receptor
Semaglutide Acetate
T19850L
Synonym: Semaglutide Acetate(910463-68-2 Free base)
Target: Glucagon Receptor
GLP-1R Agonist DMB
T36579
Synonym:
Target: Glucagon Receptor
PF-06882961 Tris
T8876
Synonym: UNII-2HJV78O0SS
Target: Glucagon Receptor
Oxyntomodulin acetate
TP1976L
Synonym:
Target: Glucagon Receptor
Adomeglivant
T14130
Synonym: LY2409021
Target: Glucagon Receptor
Avexitide acetate
TP2100L
Synonym: Exendin 9-39 acetate,Avexitide acetate（133514-43-9 Free base）
Target: Glucagon Receptor
(S, R)-LSN 3318839
T63166L
Synonym: (S, R)-LSN 3318839(Isomer-2764704-18-7)
Target: Glucagon Receptor
Mazdutide acetate（2259884-03-0 free base）
T78097L
Synonym: Mazdutide acetate（2259884-03-0 free base）,OXM-3 acetate,LY-3305677 acetate,IBI-362 acetate
Target: Glucagon Receptor
GLP-1R Antagonist 1
T15387
Synonym:
Target: Glucagon Receptor
LSN3318839
T63166
Synonym: LSN-3318839,LSN 3318839
Target: Glucagon Receptor
Tirzepatide
TP1111
Synonym: LY-3298176
Target: Glucagon Receptor
MK 0893
T12055
Synonym:
Target: Others
MK3577
T28057
Synonym: MK-3577,MK 3577
Target:
BAY-27-9955
T30299
Synonym: BAY 279955,BAY27-9955,BAY-279955,BAY 27-9955
Target:
LGD-6972 sodium
T25711
Synonym: LGD 6972 sodium
Target:
Cotadutide
T70279
Synonym:
Target:
1 2 3
Cat No. Product Name Synonyms Targets
T3896 Shanzhiside methyl ester Glucagon Receptor
Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38 MAPK signaling.
T37298 Spinacine Endogenous Metabolite
Spinacine has been isolated from spinach and the roots of Panax ginseng. This conformationally constrained amino acid is a structural element in certain biologically active compounds as glucagon antagonists and angiotens...

Natural Products

Shanzhiside methyl ester
T3896
Synonym:
Target: Glucagon Receptor
Spinacine
T37298
Synonym:
Target: Endogenous Metabolite

Recombinant Proteins

Species：
Human (6)
Mouse (2)
Rat (1)
Expression System：
E. coli (5)
HEK293 (4)
Tag：
N-terminal 6xHis-tagged (3)
N-terminal 10xHis-tagged and C-terminal Myc-tagged (2)
C-terminal 10xHis-tagged (1)
His,AVI (1)
N-terminal 6xHis-SUMO-tagged (1)
N-terminal GST-tagged (1)
Cat No. Product Name Species Expression System
TMPY-06864 GLP1R Protein, Human, Recombinant (His & Avi) Human HEK293
Glucagon-like peptide (GLP)-1 receptor is encoded by GLP1R. GLP1R plays a critical role in mediating the biological actions of GLP1 in mammals and fish. The neuronal GLP1Rs mediate body weight and anorectic effects of li...
TMPH-01386 GLP2R Protein, Human, Recombinant (His) Human HEK293
This is a receptor for glucagon-like peptide 2. The activity of this receptor is mediated by G proteins which activate adenylyl cyclase.
TMPH-03301 GLP1R Protein, Rat, Recombinant (E. coli, His) Rat E. coli
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ...
TMPH-02676 GLP1R Protein, Mouse, Recombinant (His & SUMO) Mouse E. coli
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ...
TMPH-01385 GLP1R Protein, Human, Recombinant (His) Human HEK293
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ...
TMPH-01384 GLP1R Protein, Human, Recombinant (E. coli, His) Human E. coli
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ...
TMPH-01382 GCGR Protein, Human, Recombinant (E. coli, His & Myc) Human E. coli
G-protein coupled receptor for glucagon that plays a central role in the regulation of blood glucose levels and glucose homeostasis. Regulates the rate of hepatic glucose production by promoting glycogen hydrolysis and g...
TMPH-02675 GCGR Protein, Mouse, Recombinant (GST) Mouse E. coli
G-protein coupled receptor for glucagon that plays a central role in the regulation of blood glucose levels and glucose homeostasis. Regulates the rate of hepatic glucose production by promoting glycogen hydrolysis and g...
TMPH-01383 GCGR Protein, Human, Recombinant (His & Myc) Human HEK293
G-protein coupled receptor for glucagon that plays a central role in the regulation of blood glucose levels and glucose homeostasis. Regulates the rate of hepatic glucose production by promoting glycogen hydrolysis and g...
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