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GPCR/G Protein Glucagon Receptor

Glucagon Receptor

The glucagon receptor is a 62 kDa protein that is activated by glucagon and is a member of the class B G-protein coupled family of receptors, coupled to G alpha i, Gs and to a lesser extent G alpha q. Stimulation of the receptor results in activation of adenylate cyclase and increased levels of intracellular cAMP. In humans, the glucagon receptor is encoded by the GCGR gene.
Cat No. product name
TP1452L1 HAEGTFTSD acetate(926018-45-3 free base) HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from in...
TQ0239 PF-06291874 PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
T6876 Liraglutide Liraglutide is a long-acting GLP-1 receptor agonist.
T0294 Methylprodnisolone Sodium Succinate METHYLPREDNISOLONE, a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.
T3422 GRA-Ex-25 GRA-Ex-25 is an inhibitor of glucagon receptor.
T3896 Shanzhiside methyl ester Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38...
T3984 GLP-1(7-36) GLP-1 (7-36) amide is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays vari...
T7364 NNC-0640 NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
TQ0124 BETP BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
TP1469 Lixisenatide acetate (320367-13-3 free base) Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
TP1419L HAEGTFT acetate(926018-95-3 free base) HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
TP1796 Albiglutide TFA (782500-75-8 free base) Albiglutide TFA is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
T19850 Semaglutide Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
T12431 PF-06882961 PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
T12878 Semaglutide TFA (910463-68-2 free base) Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
T11408 GLP-1 receptor agonist 1 GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .
T11845 LGD-6972 LGD-6972 is an antagonist of glucagon receptor.
T8748 Exendin-4 acetate Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).
T8876 PF-06882961 Tris PF-06882961 Tris is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
T3967 Exendin-4 Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer ...
HAEGTFTSD acetate(926018-45-3 free base)
TP1452L1CAS TP1452L1
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from in...
PF-06291874
TQ0239CAS 1393124-08-7
PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
Liraglutide
T6876CAS 204656-20-2
Liraglutide is a long-acting GLP-1 receptor agonist.
Methylprodnisolone Sodium Succinate
T0294CAS 2375-03-3
METHYLPREDNISOLONE, a water-soluble ester, is used for allergic, cardiac, and hypoxic emergencies.
GRA-Ex-25
T3422CAS 307983-31-9
GRA-Ex-25 is an inhibitor of glucagon receptor.
Shanzhiside methyl ester
T3896CAS 64421-28-9
Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38...
GLP-1(7-36)
T3984CAS 107444-51-9
GLP-1 (7-36) amide is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays vari...
NNC-0640
T7364CAS 307986-98-7
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
BETP
TQ0124CAS 1371569-69-5
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
Lixisenatide acetate (320367-13-3 free base)
TP1469CAS 1997361-87-1
Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
HAEGTFT acetate(926018-95-3 free base)
TP1419LCAS TP1419L
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
Albiglutide TFA (782500-75-8 free base)
TP1796CAS TP1796
Albiglutide TFA is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
Semaglutide
T19850CAS 910463-68-2
Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
PF-06882961
T12431CAS 2230198-02-2
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Semaglutide TFA (910463-68-2 free base)
T12878CAS T12878
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
GLP-1 receptor agonist 1
T11408CAS 2212020-52-3
GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .
LGD-6972
T11845CAS 1207989-09-0
LGD-6972 is an antagonist of glucagon receptor.
Exendin-4 acetate
T8748CAS 914454-01-6
Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).
PF-06882961 Tris
T8876CAS 2230198-03-3
PF-06882961 Tris is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Exendin-4
T3967CAS 141758-74-9
Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer ...