benzazepine

SKF83959, a benzazepine analog, is a selective and potent partial agonist of the dopamine D1 receptor with Ki values of 1.18, 7.56, 920, and 399 nM for rat D1, D5, D2, and D3 receptors, respectively.SKF83959 is a potent variant modulator of the sigma (σ)-1 receptor, which ameliorates cognitive dysfunction for the study depression and Alzheimer's disease.

Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).

SQ-31765 is a blocker of benzazepine calcium channel.

Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4 BETA2 NICOTINIC RECEPTOR partial agonist. It is used for SMOKING CESSATION.

Anilopam is an opioid analgesic belonging to the benzazepine class and acts as an agonist at opioid receptors.

Tienopramine is a benzazepine derivative and a tricyclic antidepressant. It is an analogue of Imipramine.

Trimopam is a dopamine receptor agonist of the benzazepine group.

Mozavaptan (OPC-31260) is a competitive antagonist of vasopressin receptors, targeting both V1 and V2 receptors, with IC50 values of 1.2 μM and 14 nM, respectively.