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Search Results for " pcsk9-in-9 "

8

Compounds

1

Natural Products

21

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T39528 PCSK9-IN-2 PCSK9-IN-2
PCSK9-IN-2 is a newly developed small molecule that effectively inhibits the protein-protein interaction (PPI) between PCSK9 and LDLR. It has been found to have a potent inhibitory activity with an IC50 value of 7.57 μM.
TP1881L1 Pep 2-8 ammonium salt(1541011-97-5 free base) Others
Pep 2-8 ammonium salt is Proprotein convertase subtilisin/kexin type 9 (PCSK9) inhibitor. Potent inhibitor of PCSK9 binding to LDL receptor (IC50 = 0.8 μM). Restores LDL uptake in HepG2 cells treated with PCSK9.
T72025 PCSK9-IN-10 Serine/threonin kinase
PCSK9-IN-10, a potent and orally active inhibitor of Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9), exhibits a half-maximal inhibitory concentration (IC50) of 6.4 µM. By enhancing the expression of Low-Density Li...
TP1881 Pep2-8 Pep 2-8
Proprotein convertase subtilisin/kexin type 9 (PCSK9) inhibitor. Potent inhibitor of PCSK9 binding to LDL receptor (IC50 = 0.8 μM). Restores LDL uptake in HepG2 cells treated with PCSK9.
T70069 MDK6465
MDK6465, also known as PCSK9-IN-8b, is a novel liver-targeted inhibitor of ribosomal synthesis of proprotein convertase subtilisin/kexin type 9 (PCSK9). MDK6465 has CAS#1900686-46-5. the last 4 digits are used in its na...
T72221 PF-06815345 hydrochloride
PF-06815345 hydrochloride, an orally active potent inhibitor of proprotein convertase subtilisin/kexin type 9 (PCSK9), has an IC50 value of 13.4 μM. It significantly decreases in vivo PCSK9 levels in mice.
T60541 PCSK9 modulator-2
PCSK9 modulator-2 (Compound 1) is a potent PCSK9 modulator (EC 50 = 202 nM) that has the potential to be used in hyperlipidemia research. Proprotein convertase subtilisin/kexin type 9 (PCSK9) is a recently validated ther...
T79051 PCSK9-IN-15
PCSK9-IN-15 (compound 5) is a potent inhibitor of proprotein convertase subtilisin/kexin 9 (PCSK9, K D <200 nM) that plays a crucial role in cholesterol metabolism by regulating blood levels of low-density lipoprotein ch...
Cat No. Product Name Synonyms Targets
T75545 PCSK9-IN-9
PCSK9-IN-9, a natural isocoumarin, inhibits proprotein convertase subtilisin-kexin type 9 (PCSK9), IDOL, and SREBP2 mRNA expression, demonstrating specificity by inhibiting PCSK9 with an IC50 value of 11.9 μM [1].

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-04966 PCSK9 Protein, Human, Recombinant (D374Y, His) Human HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPY-00408 PCSK9 Protein, Human, Recombinant (D374Y & V474I & G670E, His) Human HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPY-05131 PCSK9 Protein, Human, Recombinant (His & Avi), Biotinylated Human HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPJ-00369 PCSK9 Protein, Human, Recombinant (His & HA & Avi), Biotinylated Human Human Cells
Human Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) is a secretory subtilase belonging to the proteinase K subfamily. PCSK9 is synthesized as a soluble zymogen that undergoes autocatalytic intramolecular processi...
TMPJ-00443 PCSK9 Protein, Macaca nemestrina, Recombinant (His) Macaca nemestrina Human Cells
Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) is a secretory subtilase belonging to the proteinase K subfamily. PCSK9 is synthesized as a soluble zymogen that undergoes autocatalytic intramolecular processing in ...
TMPK-00483 PCSK9 Protein, Cynomolgus, Recombinant (His) Cynomolgus HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9) is an enzyme encoded by the PCSK9 gene in humans on chromosome 1.The first two PCSK9 inhibitors, alirocumab and evolocumab, were approved as once every two week injec...
TMPJ-00368 PCSK9 Protein, Human, Recombinant (Avi), Biotinylated Human Human Cells
Human Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) is a secretory subtilase belonging to the proteinase K subfamily. PCSK9 is synthesized as a soluble zymogen that undergoes autocatalytic intramolecular processi...
TMPY-05217 PCSK9 Protein, Mouse, Recombinant (mFc) Mouse HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPY-05114 PCSK9 Protein, Human, Recombinant (D374Y & V474I & G670E, His), Biotinylated Human HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPY-01245 PCSK9 Protein, Mouse, Recombinant (His) Mouse HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPY-00995 PCSK9 Protein, Rhesus, Recombinant (His) Rhesus HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPY-01565 PCSK9 Protein, Rat, Recombinant (His) Rat HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPY-05270 PCSK9 Protein, Human, Recombinant (D374Y, mFc), Biotinylated Human HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPY-05199 PCSK9 Protein, Human, Recombinant (D374Y, mFc) Human HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPY-05218 PCSK9 Protein, Human, Recombinant (mFc) Human HEK293
Proprotein convertase subtilisin/kexin type 9 (PCSK9), also known as NARC1 (neural apoptosis regulated convertase), which is a newly identified human secretory subtilase belonging to the proteinase K subfamily of the sec...
TMPJ-00865 VEGF121 Protein, Human, Recombinant (His) Human Human Cells
Human VEGF121, also known as Vascular endothelial growth factor A, VEGFA, Vascular permeability factor, VPF and VEGF, is a homodimeric, heparin-binding glycoprotein which belongs to the platelet-derived growth factor (PD...
TMPY-03698 VEGF121b Protein, Human, Recombinant Human HEK293
Vascular endothelial growth factor (VEGF), also known as vascular permeability factor (VPF) and VEGF-A, is a potent mediator of both angiogenesis and vasculogenesis in the fetus and adult. It is a member of the platelet-...
TMPH-00005 YAP1 Protein, Human, Recombinant (Isoform 9, His) Human Yeast
TMPK-00825 VEGF121 Protein, Human, Recombinant (His & Avi) Human HEK293
Vascular endothelial growth factor (VEGF or VEGF-A), also known as vascular permeability factor (VPF), is a potent mediator of both angiogenesis and vasculogenesis in the fetus and adult. VEGF165 appears to be the most a...
TMPK-00826 VEGF121 Protein, Human, Recombinant (His & Avi), Biotinylated Human HEK293
Vascular endothelial growth factor (VEGF or VEGF-A), also known as vascular permeability factor (VPF), is a potent mediator of both angiogenesis and vasculogenesis in the fetus and adult. VEGF165 appears to be the most a...
TMPY-05268 Neurofascin Protein, Human, Recombinant (hFc), Biotinylated Human HEK293
NFASC (Neurofascin, also known as NRCAML, NEDCPMD, and NF) is a Protein Coding gene. 13 alternatively spliced human isoforms have been reported. NFASC belongs to the immunoglobulin superfamily, L1/neurofascin/NgCAM famil...
PCSK9 Protein, Human, Recombinant (D374Y, His)
TMPY-04966
Species: Human
Expression System: HEK293
PCSK9 Protein, Human, Recombinant (D374Y & V474I & G670E, His)
TMPY-00408
Species: Human
Expression System: HEK293
PCSK9 Protein, Human, Recombinant (His & Avi), Biotinylated
TMPY-05131
Species: Human
Expression System: HEK293
PCSK9 Protein, Human, Recombinant (His & HA & Avi), Biotinylated
TMPJ-00369
Species: Human
Expression System: Human Cells
PCSK9 Protein, Macaca nemestrina, Recombinant (His)
TMPJ-00443
Species: Macaca nemestrina
Expression System: Human Cells
PCSK9 Protein, Cynomolgus, Recombinant (His)
TMPK-00483
Species: Cynomolgus
Expression System: HEK293
PCSK9 Protein, Human, Recombinant (Avi), Biotinylated
TMPJ-00368
Species: Human
Expression System: Human Cells
PCSK9 Protein, Mouse, Recombinant (mFc)
TMPY-05217
Species: Mouse
Expression System: HEK293
PCSK9 Protein, Human, Recombinant (D374Y & V474I & G670E, His), Biotinylated
TMPY-05114
Species: Human
Expression System: HEK293
PCSK9 Protein, Mouse, Recombinant (His)
TMPY-01245
Species: Mouse
Expression System: HEK293
PCSK9 Protein, Rhesus, Recombinant (His)
TMPY-00995
Species: Rhesus
Expression System: HEK293
PCSK9 Protein, Rat, Recombinant (His)
TMPY-01565
Species: Rat
Expression System: HEK293
PCSK9 Protein, Human, Recombinant (D374Y, mFc), Biotinylated
TMPY-05270
Species: Human
Expression System: HEK293
PCSK9 Protein, Human, Recombinant (D374Y, mFc)
TMPY-05199
Species: Human
Expression System: HEK293
PCSK9 Protein, Human, Recombinant (mFc)
TMPY-05218
Species: Human
Expression System: HEK293
VEGF121 Protein, Human, Recombinant (His)
TMPJ-00865
Species: Human
Expression System: Human Cells
VEGF121b Protein, Human, Recombinant
TMPY-03698
Species: Human
Expression System: HEK293
YAP1 Protein, Human, Recombinant (Isoform 9, His)
TMPH-00005
Species: Human
Expression System: Yeast
VEGF121 Protein, Human, Recombinant (His & Avi)
TMPK-00825
Species: Human
Expression System: HEK293
VEGF121 Protein, Human, Recombinant (His & Avi), Biotinylated
TMPK-00826
Species: Human
Expression System: HEK293
Neurofascin Protein, Human, Recombinant (hFc), Biotinylated
TMPY-05268
Species: Human
Expression System: HEK293
TargetMol