T6293 |
Mycophenolate Mofetil
|
128794-94-5
|
98%
|
|
Mycophenolate mofetil, an immunosuppressive agent, is the 2-morpholinoethyl ester of mycophenolic acid (MPA), and an inhibitor of inosine monophosphate dehydroge...
|
T4710 |
3-Methoxytyramine hydrochloride
|
1477-68-5
|
98%
|
|
3-Methoxytyramine hydrochloride is an inactive metabolite of dopamine which can activate trace amine associated receptor 1 (TAAR1). 3-methoxytyramine can be foun...
|
T8217 |
Enzalutamide carboxylic acid
|
1242137-15-0
|
98%
|
|
Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .
|
T13539 |
Allopurinol riboside
|
16220-07-8
|
98%
|
|
Allopurinol riboside is a metabolite of allopurinol with potency against parasites. Allopurinol riboside competitively inhibits the action of purine nucleoside p...
|
T16338 |
Norgestimate metabolite Norelgestromin
|
53016-31-2
|
98%
|
|
Norelgestromin is one of the active metabolites of norgestimate.It is a steroidal progestin used in contraceptive patches, where it is combined with the estrogen...
|
T8339 |
16α-Hydroxyprednisolone
|
13951-70-7
|
98%
|
|
16alpha-Hydroxyprednisolone is a stereoselective metabolite of the 22(R) epimer of the glucocorticoid budesonide
|
T13808 |
P-Coumaric Acid Ethyl Ester
|
7362-39-2
|
98%
|
|
p-Coumaric Acid Ethyl Ester is the ethyl ester of p-Coumaric acid. p-Coumaric Acid is a common dietary polyphenol and also a potent immunosuppressive agent in tr...
|
T8945L |
AST5902 mesylate(2412155-74-7 free base)
|
T8945L
|
98%
|
|
AST5902 mesylate is principal metabolite of Alflutinib in vivo. AST5902 mesylate exerts antineoplastic activity.
|
T5420 |
Cycloguanil hydrochloride
|
152-53-4
|
98%
|
|
Cycloguanil is an active metabolite of the antimalarial compound proguanil. It acts as an inhibitor of dihydrofolate reductase (Kis: 0.3 and 1.5 nM for Plasmodiu...
|
T10157 |
Regorafénib N-oxyde (M2)
|
835621-11-9
|
98%
|
|
Regorafénib N-oxyde M2 is an active metabolite of Regorafenib. Regorafenib is a multi-target inhibitor for VEGFR1/2/3, PDGFRβ, RET, Kit, and Raf-1 (IC50s: 13/4.2...
|
T10147 |
4-Hydroxymephenytoin
|
61837-65-8
|
98%
|
|
4-Hydroxymephenytoin is the metabolism of an antiepileptic drug mephenytoin. Mephenytoin is used as a CYP2C19 substrate.
|
T8547 |
DCBA
|
72236-23-8
|
98%
|
|
DCBA is a endogenous metabolite of insect repellent N-N-diethyl-meta-toluamide (DEET). The concentration of DCBA in urine can assess exposure to DEET.
|
T16339 |
Norverapamil hydrochloride
|
67812-42-4
|
98%
|
|
Norverapamil hydrochloride ((±)-Norverapamil hydrochloride) is an N-demethylated metabolite of Verapamil and it is an L-type calcium channel blocker and a P-glyc...
|
T7174 |
Urolithin A
|
1143-70-0
|
98%
|
|
Urolithin A is a secondary metabolite of ellagic acid, a polyphenolic antioxidant, that has antiproliferative, anti-inflammatory, and anti-oxidant properties.
|
T4281 |
Endoxifen
|
110025-28-0
|
98%
|
|
(E/Z)-Endoxifen is an active metabolite of tamoxifen produced by the sequential action of cytochrome P450 (CYP) isoforms, including CYP2D6. It is a strong anti-e...
|
T36061 |
N-Desmethyl Sildenafil
|
139755-82-1
|
98%
|
|
N-Desmethyl Sildenafil (Desmethylsildenafil) is a major metabolite of Sildenafil. Sildenafil is a potent phosphodiesterase type 5 (PDE5) inhibitor.
|
Fr13756 |
Isonicotinic acid
|
55-22-1
|
98%
|
|
Isonicotinic acid is a metabolite of Isoniazid.Isonicotinic acid is a useful isomer of nicotinic acid. Isoniazid is converted to Isonicotinic acid by hydrazinoly...
|
T13621 |
CNDAC hydrochloride
|
134665-72-8
|
98%
|
|
CNDAC hydrochloride, a nucleoside analog, is a metabolite of the sapacitabine.
|
T16045 |
Methotrexate metabolite
|
19741-14-1
|
98%
|
|
Methotrexate metabolite (DAMPA) is the active metabolite of Methotrexate. Methotrexate is a folic acid antagonist. Methotrexate is used as a chemotherapeutic age...
|
T1327 |
Nortriptyline hydrochloride
|
894-71-3
|
98%
|
|
Nortriptyline hydrochloride is a metabolite of AMITRIPTYLINE that is also used as an antidepressive agent. Nortriptyline is used in major depression, dysthymia, ...
|