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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T1696 2-(1-Piperazinyl)pyrimidine 20980-22-7 98.86%
2-(1-Piperazinyl)pyrimidine
2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
T13655 DL-Norepinephrine hydrochloride 55-27-6 98.86%
DL-Norepinephrine hydrochloride
DL-Norepinephrine hydrochloride (DL-lysine) is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 ...
T68051L RS 15385-198 121961-55-5 98.81%
RS 15385-198
RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor antagonist.
T68051 Delequamine 119905-05-4 98.75%
Delequamine
Delequamine (RS 15385-197) is a selective and potent TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study men...
T3232 Higenamine hydrochloride 11041-94-4 98.75%
Higenamine hydrochloride
Higenamine hydrochloride (norcoclaurine HCl) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class...
T3431 Pardoprunox hydrochloride 269718-83-4 98.73%
Pardoprunox hydrochloride
Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) an...
T77566 (3aR,9aR)-Fluparoxan 105182-47-6 98.68%
(3aR,9aR)-Fluparoxan
(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental diso...
T10066 2',5'-Dideoxyadenosine 6698-26-6 98.66%
2',5'-Dideoxyadenosine
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
T19769 Cimaterol 54239-37-1 98.64%
Cimaterol
Cimaterol is a potent β-adrenoceptor agonist. cimaterol binds to the L6β-receptor with a Kd value of 26 nM, which is consistent with its EC50 for stimulating pro...
T14490 Talipexole dihydrochloride 36085-73-1 98.64%
Talipexole dihydrochloride
Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and intestinal...
T22612 BMY-14802 hydrochloride 105565-55-7 98.64%
BMY-14802 hydrochloride
BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects. BMY-14802 hydrochloride is...
T20157 Brimonidine 59803-98-4 98.60%
Brimonidine
Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P. It is used to treat open-angle glaucoma or ocular hypertensi...
T2535 Ivabradine hydrochloride 148849-67-6 98.6%
Ivabradine hydrochloride
Ivabradine hydrochloride (S 16257-2) is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioav...
T22369 Midodrine 42794-76-3 98.57%
Midodrine
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.
T13804 OPC-28326 167626-17-7 98.56%
OPC-28326
OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of...
T31175 Dabelotine 118976-38-8 98.55%
Dabelotine
Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.
T8899 Metipranolol 22664-55-7 98.54%
Metipranolol
Metipranolol is a useful organic compound for research related to life sciences. The catalog number is T8899 and the CAS number is 22664-55-7.
T26923 Bunazosin Hydrochloride 52712-76-2 98.48%
Bunazosin Hydrochloride
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
T10952 Dabuzalgron 219311-44-1 98.47%
Dabuzalgron
Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicit...
T6519 Gramine 87-52-5 98.44%
Gramine
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4...
2-(1-Piperazinyl)pyrimidine
T1696
2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
DL-Norepinephrine hydrochloride
T13655
DL-Norepinephrine hydrochloride (DL-lysine) is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 ...
RS 15385-198
T68051L
RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor antagonist.
Delequamine
T68051
Delequamine (RS 15385-197) is a selective and potent TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study men...
Higenamine hydrochloride
T3232
Higenamine hydrochloride (norcoclaurine HCl) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class...
Pardoprunox hydrochloride
T3431
Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) an...
(3aR,9aR)-Fluparoxan
T77566
(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental diso...
2',5'-Dideoxyadenosine
T10066
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
Cimaterol
T19769
Cimaterol is a potent β-adrenoceptor agonist. cimaterol binds to the L6β-receptor with a Kd value of 26 nM, which is consistent with its EC50 for stimulating pro...
Talipexole dihydrochloride
T14490
Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and intestinal...
BMY-14802 hydrochloride
T22612
BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects. BMY-14802 hydrochloride is...
Brimonidine
T20157
Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P. It is used to treat open-angle glaucoma or ocular hypertensi...
Ivabradine hydrochloride
T2535
Ivabradine hydrochloride (S 16257-2) is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioav...
Midodrine
T22369
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.
OPC-28326
T13804
OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of...
Dabelotine
T31175
Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.
Metipranolol
T8899
Metipranolol is a useful organic compound for research related to life sciences. The catalog number is T8899 and the CAS number is 22664-55-7.
Bunazosin Hydrochloride
T26923
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
Dabuzalgron
T10952
Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicit...
Gramine
T6519
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4...
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TargetMol