Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T6652	Salbutamol hemisulfate	51022-70-9	99.39%
T6652	Salbutamol hemisulfate (Albuterol Sulfate) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
T10778	CGP 20712 A	105737-62-0	99.37%
T10778	CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
T1577	Midodrine hydrochloride	3092-17-9	99.36%
T1577	Midodrine is converted to its active metabolite, desglymidodrine by deglycination reaction. Desglymidodrine selectively binds to and activates alpha-1-adrenergic...
T6688	Synephrine hydrochloride	5985-28-4	99.36%
T6688	Synephrine hydrochloride (Oxedrine hydrochloride) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
T4983	Isoetharine mesylate salt	7279-75-6	99.35%
T4983	Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450...
T0031L	Ziprasidone hydrochloride	122883-93-6	99.34%
T0031L	Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic acti...
T10830	CL 316243	138908-40-4	99.34%
T10830	CL316243 is a highly potent selective agonist of β3-adrenoceptor, with a EC50 of 3 nM. CL316243 is an effective stimulant of adipocyte lipolysis and increases br...
T24064	Fipamezole	150586-58-6	99.32%
T24064	Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.
T26760	Bedoradrine sulfate	194785-31-4	99.31%
T26760	Bedoradrine sulfate (MN-221 sulfate) is a super-selective beta2 agonist for the treatment of asthma exacerbations and chronic obstructive pulmonary disease.
T1239	Indacaterol maleate	753498-25-8	99.31%
T1239	Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
T0324	Isoxsuprine hydrochloride	579-56-6	99.31%
T0324	Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
T0137	Mirtazapine	85650-52-8	99.3%
T0137	Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
T22406	Prazosin	19216-56-9	99.29%
T22406	Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T16798	RS 17053 hydrochloride	169505-93-5	99.27%
T16798	RS 17053 hydrochloride is a potent and selective antagonist of α1A adrenoceptor. RS 17053 hydrochloride exhibits a pKi value of 9.1 in native cell membrane and a...
T9762	Upidosin	152735-23-4	99.26%
T9762	Upidosin (SB-216469) is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenocepto...
T21445	Naphazoline	835-31-4	99.25%
T21445	Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity. Naphazoline can be used as a vasoconstrictor with a rapid action in ...
T0383	Fenspiride hydrochloride	5053-08-7	99.18%
T0383	Fenspiride hydrochloride (Decaspiride) , an oxazolidinone spiro compound, is a drug used in the therapy of certain respiratory diseases. It is approved for use i...
T10100	QF0301B	149247-12-1	99.16%
T10100	QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.
T21640	Talinolol	57460-41-0	99.15%
T21640	(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
T1671	Mirabegron	223673-61-8	99.14%
T1671	Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.