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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T9220 Naftopidil hydrochloride 1164469-60-6 99.95%
Naftopidil hydrochloride
Naftopidil hydrochloride (BM-15275 hydrochloride) is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adre...
T0031 Ziprasidone hydrochloride monohydrate 138982-67-9 99.95%
Ziprasidone hydrochloride monohydrate
Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic ac...
T5511 L-765314 189349-50-6 99.95%
L-765314
L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the ro...
T6600 Naftopidil dihydrochloride 57149-08-3 99.95%
Naftopidil dihydrochloride
Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
T0991 Desipramine hydrochloride 58-28-6 99.94%
Desipramine hydrochloride
Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervou...
T0210L Tamsulosin 106133-20-4 99.94%
Tamsulosin
Tamsulosin ((R)-(-)-YM12617 free base) is an alpha1A adrenergic receptor antagonist for the symptomatic treatment of benign prostatic hyperplasia (BPH). Tamsulos...
T0088 Urapidil hydrochloride 64887-14-5 99.93%
Urapidil hydrochloride
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
T17310 Phenylephrine 59-42-7 99.92%
Phenylephrine
Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
T0103 Dipivefrin hydrochloride 64019-93-8 99.92%
Dipivefrin hydrochloride
Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
T1073 Dronedarone hydrochloride 141625-93-6 99.91%
Dronedarone hydrochloride
Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
T3278 Piribedil 3605-01-4 99.91%
Piribedil
Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
T0197 Terazosin hydrochloride 63074-08-8 99.91%
Terazosin hydrochloride
Terazosin hydrochloride (Hytrin) , a selective alpha1-antagonist, can treat the benign prostatic hyperplasia (BPH). It also can lower blood pressure, so it is a ...
T26363L Napitane 148152-63-0 99.91%
Napitane
napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the stud...
T1500 Xylazine hydrochloride 23076-35-9 99.9%
Xylazine hydrochloride
Xylazine hydrochloride (BAY 1470 hydrochloride) is an adrenergic alpha-2 agonist used as a sedative, analgesic and centrally acting muscle relaxant in veterinary...
T1415 Gemfibrozil 25812-30-0 99.9%
Gemfibrozil
Gemfibrozil (CI-719) interacts with peroxisome proliferator-activated receptors (PPARalpha) resulting in PPARalpha-mediated stimulation of fatty acid oxidation a...
T12829 Salmeterol 89365-50-4 99.9%
Salmeterol
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
T1275 Phentolamine mesylate 65-28-1 99.9%
Phentolamine mesylate
Phentolamine mesylate (Phentolamine methanesulfonate) is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive...
T5105 1-(2-Pyridyl)piperazine 34803-66-2 99.89%
1-(2-Pyridyl)piperazine
1-(2-Pyridyl)piperazine (NSC-13778) is a selective α2-adrenoceptor antagonists. 1-(2-Pyridyl)piperazine shows sympatholytic activity. 1-(2-Pyridyl)piperazine is ...
T6464 Detomidine hydrochloride 90038-01-0 99.89%
Detomidine hydrochloride
Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.
T7045 Clonidine 4205-90-7 99.88%
Clonidine
Clonidine (Kapvay) is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Desp...
Naftopidil hydrochloride
T9220
Naftopidil hydrochloride (BM-15275 hydrochloride) is a selective alpha1-adrenoceptor antagonist with Ki of 3.7 nM, 20 nM and 1.2 nM for the cloned human α1a-adre...
Ziprasidone hydrochloride monohydrate
T0031
Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic ac...
L-765314
T5511
L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the ro...
Naftopidil dihydrochloride
T6600
Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
Desipramine hydrochloride
T0991
Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervou...
Tamsulosin
T0210L
Tamsulosin ((R)-(-)-YM12617 free base) is an alpha1A adrenergic receptor antagonist for the symptomatic treatment of benign prostatic hyperplasia (BPH). Tamsulos...
Urapidil hydrochloride
T0088
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
Phenylephrine
T17310
Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
Dipivefrin hydrochloride
T0103
Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
Dronedarone hydrochloride
T1073
Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
Piribedil
T3278
Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
Terazosin hydrochloride
T0197
Terazosin hydrochloride (Hytrin) , a selective alpha1-antagonist, can treat the benign prostatic hyperplasia (BPH). It also can lower blood pressure, so it is a ...
Napitane
T26363L
napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the stud...
Xylazine hydrochloride
T1500
Xylazine hydrochloride (BAY 1470 hydrochloride) is an adrenergic alpha-2 agonist used as a sedative, analgesic and centrally acting muscle relaxant in veterinary...
Gemfibrozil
T1415
Gemfibrozil (CI-719) interacts with peroxisome proliferator-activated receptors (PPARalpha) resulting in PPARalpha-mediated stimulation of fatty acid oxidation a...
Salmeterol
T12829
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
Phentolamine mesylate
T1275
Phentolamine mesylate (Phentolamine methanesulfonate) is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive...
1-(2-Pyridyl)piperazine
T5105
1-(2-Pyridyl)piperazine (NSC-13778) is a selective α2-adrenoceptor antagonists. 1-(2-Pyridyl)piperazine shows sympatholytic activity. 1-(2-Pyridyl)piperazine is ...
Detomidine hydrochloride
T6464
Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.
Clonidine
T7045
Clonidine (Kapvay) is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Desp...
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TargetMol