Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.

Cat. No.	Product name	CAS No.	Purity
T0031	Ziprasidone hydrochloride monohydrate	138982-67-9	99.95%
T0031	Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic ac...
T5511	L-765314	189349-50-6	99.95%
T5511	L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the ro...
T6600	Naftopidil dihydrochloride	57149-08-3	99.95%
T6600	Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
T0991	Desipramine hydrochloride	58-28-6	99.94%
T0991	Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervou...
T0210L	Tamsulosin	106133-20-4	99.94%
T0210L	Tamsulosin ((R)-(-)-YM12617 free base) is an alpha1A adrenergic receptor antagonist for the symptomatic treatment of benign prostatic hyperplasia (BPH). Tamsulos...
T0455	Clozapine	5786-21-0	99.93%
T0455	Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, an...
T0088	Urapidil hydrochloride	64887-14-5	99.93%
T0088	Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
T1567	Olanzapine	132539-06-1	99.92%
T1567	Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
T17310	Phenylephrine	59-42-7	99.92%
T17310	Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
T0103	Dipivefrin hydrochloride	64019-93-8	99.92%
T0103	Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
T1073	Dronedarone hydrochloride	141625-93-6	99.91%
T1073	Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
T1540	Doxepin hydrochloride	1229-29-4	99.91%
T1540	Doxepin hydrochloride (Aponal) is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation....
T3278	Piribedil	3605-01-4	99.91%
T3278	Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
T0197	Terazosin hydrochloride	63074-08-8	99.91%
T0197	Terazosin hydrochloride (Hytrin) , a selective alpha1-antagonist, can treat the benign prostatic hyperplasia (BPH). It also can lower blood pressure, so it is a ...
T26363L	Napitane	148152-63-0	99.91%
T26363L	napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the stud...
T1415	Gemfibrozil	25812-30-0	99.9%
T1415	Gemfibrozil (CI-719) interacts with peroxisome proliferator-activated receptors (PPARalpha) resulting in PPARalpha-mediated stimulation of fatty acid oxidation a...
T12829	Salmeterol	89365-50-4	99.9%
T12829	Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
T10631	Bucindolol	71119-11-4	99.9%
T10631	Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.
T1275	Phentolamine mesylate	65-28-1	99.9%
T1275	Phentolamine mesylate (Phentolamine methanesulfonate) is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive...
T1433	Ritodrine hydrochloride	23239-51-2	99.89%
T1433	Ritodrine hydrochloride (NSC 291565) binds to and activates beta-2 adrenergic receptors of myometrial cells in the uterus, which decreases the intensity and fre...