Select your Country or Region

  • TargetMol | Compound LibraryArgentinaArgentina
  • TargetMol | Compound LibraryAustraliaAustralia
  • TargetMol | Compound LibraryAustriaAustria
  • TargetMol | Compound LibraryBelgiumBelgium
  • TargetMol | Compound LibraryBrazilBrazil
  • TargetMol | Compound LibraryBulgariaBulgaria
  • TargetMol | Compound LibraryCroatiaCroatia
  • TargetMol | Compound LibraryCyprusCyprus
  • TargetMol | Compound LibraryCzechCzech
  • TargetMol | Compound LibraryDenmarkDenmark
  • TargetMol | Compound LibraryEgyptEgypt
  • TargetMol | Compound LibraryEstoniaEstonia
  • TargetMol | Compound LibraryFinlandFinland
  • TargetMol | Compound LibraryFranceFrance
  • TargetMol | Compound LibraryGermanyGermany
  • TargetMol | Compound LibraryGreeceGreece
  • TargetMol | Compound LibraryHong KongHong Kong
  • TargetMol | Compound LibraryHungaryHungary
  • TargetMol | Compound LibraryIcelandIceland
  • TargetMol | Compound LibraryIndiaIndia
  • TargetMol | Compound LibraryIrelandIreland
  • TargetMol | Compound LibraryIsraelIsrael
  • TargetMol | Compound LibraryItalyItaly
  • TargetMol | Compound LibraryJapanJapan
  • TargetMol | Compound LibraryKoreaKorea
  • TargetMol | Compound LibraryLatviaLatvia
  • TargetMol | Compound LibraryLebanonLebanon
  • TargetMol | Compound LibraryMalaysiaMalaysia
  • TargetMol | Compound LibraryMaltaMalta
  • TargetMol | Compound LibraryMoroccoMorocco
  • TargetMol | Compound LibraryNetherlandsNetherlands
  • TargetMol | Compound LibraryNew ZealandNew Zealand
  • TargetMol | Compound LibraryNorwayNorway
  • TargetMol | Compound LibraryPolandPoland
  • TargetMol | Compound LibraryPortugalPortugal
  • TargetMol | Compound LibraryRomaniaRomania
  • TargetMol | Compound LibrarySingaporeSingapore
  • TargetMol | Compound LibrarySlovakiaSlovakia
  • TargetMol | Compound LibrarySloveniaSlovenia
  • TargetMol | Compound LibrarySpainSpain
  • TargetMol | Compound LibrarySwedenSweden
  • TargetMol | Compound LibrarySwitzerlandSwitzerland
  • TargetMol | Compound LibraryTaiwan,ChinaTaiwan,China
  • TargetMol | Compound LibraryThailandThailand
  • TargetMol | Compound LibraryTurkeyTurkey
  • TargetMol | Compound LibraryUnited KingdomUnited Kingdom
  • TargetMol | Compound LibraryUnited StatesUnited States
  • TargetMol | Compound LibraryOther CountriesOther Countries
Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
Applied FilterClear all
TargetMol | Tags By Target
  • ADC Linker
    (2)
  • Adenosine Receptor
    (2)
  • Drug-Linker Conjugates for ADC
    (3)
  • Estrogen Receptor/ERR
    (2)
  • GABA Receptor
    (4)
  • Glucagon Receptor
    (2)
  • Histamine Receptor
    (3)
  • LPA Receptor
    (2)
  • Sigma receptor
    (6)
  • Others
    (63)
Filter
Search Result
Results for "

target/GABA_Receptor/1

" in TargetMol Product Catalog
  • Inhibitor Products
    103
    TargetMol | Activity
  • Peptides Products
    6
    TargetMol | inventory
  • Dye Reagents
    1
    TargetMol | natural
  • PROTAC Products
    1
    TargetMol | composition
  • Recombinant Protein
    5
    TargetMol | Activity
Y1 receptor antagonist 1
T12155221697-09-2In house
Y1 receptor antagonist 1 (H 409-22 isomer) is the active isomer of H-409/22, a neuropeptide Y (NPY) Y1 receptor antagonist that dose-dependently antagonizes the vascular response to exogenous and endogenous NPY in pigs. lagodeoxycholic acid (H 409-22 isomer) is the active isomer of H-409/22, an antagonist of neuropeptide Y (NPY) Y1 receptor.
  • $353
Backorder
Size
QTY
Edg-2 receptor inhibitor 1
T45211195941-38-8
Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).
  • $98
In Stock
Size
QTY
A2B receptor antagonist 1
T10058531506-36-2In house
A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.
  • $388
In Stock
Size
QTY
TargetMol | Inhibitor Sale
Protease-Activated Receptor-1, PAR-1 Agonist acetate
T38836L
Protease-Activated Receptor-1, PAR-1 Agonist acetate is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 Agonist acetate corresponds to PAR1 tethered ligand and which can selectively mimic theactions of thrombin via this receptor[1][2].
  • $133
In Stock
Size
QTY
AMPA receptor modulator-1
T103072036074-41-4In house
AMPA receptor modulator-1 can be activated by glutamate, thereby modulating ion channels.
  • $117
In Stock
Size
QTY
GLP-1 receptor agonist 9 citrate
T9579L
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
  • $195
In Stock
Size
QTY
TargetMol | Inhibitor Sale
LPA1 receptor antagonist 1
T157851396006-71-5In house
LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a selective and potent lysophosphatidic acid (LPA1) receptor antagonist (IC50 : 25 nM) for the study of idiopathic pulmonary fibrosis.
  • $147 TargetMol
In Stock
Size
QTY
A2A receptor antagonist 1
T37792443103-97-7In house
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
  • $31
In Stock
Size
QTY
Dopamine D2 receptor antagonist-1
T110771055411-77-2In house
Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.
  • $55
In Stock
Size
QTY
Sigma-1 receptor antagonist 2
T129111639220-15-7In house
Sigma-1 receptor antagonist 2 is a potent and selective antagonist of sigma 1 receptor (σ1 R) (σ1 and σ2 receptor with Kis of 3.88 and 1288 nM , respectively).
  • $97
In Stock
Size
QTY
Glucocorticoid receptor agonist-1
T379082166375-82-0In house
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].
  • $226
In Stock
Size
QTY
Androgen receptor antagonist 1
T103201338812-36-4In house
Androgen receptor antagonist 1 is an orally available full androgen receptor antagonist (IC50: 59 nM). It can be used in the synthesis of PROTAC AR degraders, which results in 24% and 47 % AR protein degradation in LNCaP cells at 1 μM and 10 μM, respectively.
  • $1,520
6-8 weeks
Size
QTY
Target 1
T9467 In house
Target 1 has a wide range of applications in life science related research.
    Inquiry
    TargetMol | Inhibitor Sale
    (E)-GABAB receptor antagonist 1
    T111371611483-29-4In house
    (E)-GABAB receptor antagonist 1 is a trans-GABAB receptor antagonist 1. (E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM. GABAB receptor antagonist 1 is a selective and negative allosteric modulator of GABAB (γ-Aminobutyric acid) receptors.
    • $195
    In Stock
    Size
    QTY
    H3 receptor antagonist 1
    T10911935840-13-4In house
    H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
    • $1,520
    8-10 weeks
    Size
    QTY
    Sigma-1 receptor antagonist 3
    T129121639220-17-9In house
    Sigma-1 receptor antagonist 3 is a potent and selective antagonist of Sigma-1 (σ1) receptor(Ki : 1.14 nM), has the potential for the neuropathic pain.
    • $81
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
    GP130 receptor agonist-1
    T9157339303-87-6
    GP130 receptor agonist-1 (N-(4-Fluorophenyl)-4-phenyl-2-thiazolami) is a potent, brain-penetrant and orally active GP130 receptor agonist.
    • $30
    In Stock
    Size
    QTY
    TargetMol | Citations Cited
    GABA receptor Antagonist 1
    T82357
    GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 of 7.08 nmol/L and demonstrates insecticidal efficacy against P. xylostella, S. frugiperda, S. exigua, and S. litura with respective LC50 values of 0.09, 0.84, 0.87, and 0.68 mg/L. Moreover, this compound exhibits moderate toxicity to honeybees (48 h, ID50 = 2.22 μg/adult) and low toxicity to zebrafish (LC50: 42.4 mg/L) [1].
    • Inquiry Price
    Size
    QTY
    TargetMol | Inhibitor Sale
    Interferon receptor inducer-1
    T137362215120-36-6
    Interferon receptor inducer-1 Used in the treatment of a disorder in which the induction of interferon is involved. is an interferon (IFN) receptor inducer.
    • $30
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
    Androgen receptor degrader-1
    T806332616553-35-4
    Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in cancer research [1].
    • Inquiry Price
    Size
    QTY
    TargetMol | Inhibitor Sale
    RXFP1 receptor agonist-1
    T812462924619-64-5
    RXFP1 receptor agonist-1 (Example 2), an agonist of the RXFP1 receptor, suppresses cAMP production in HEK293 cells that constitutively express the human RXFP1, exhibiting an EC50 of 300 nM [1].
    • Inquiry Price
    Size
    QTY
    TargetMol | Inhibitor Sale
    Histamine H4 receptor antagonist-1
    T386341246207-84-0
    Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.
    • Inquiry Price
    Size
    QTY
    TargetMol | Inhibitor Sale
    GLP-1 receptor agonist 4
    T114051187061-62-6
    GLP-1 receptor agonist 4 is a glucagon-like peptide-1 receptor (GLP-1R) agonist , has an EC50 of 64.5 nM. GLP-1 receptor agonist 4 can be used in the research for treatment of diabetes.
    • Inquiry Price
    Size
    QTY
    TargetMol | Inhibitor Sale
    Succinate/succinate receptor antagonist 1
    T679152361972-29-2
    Succinate/succinate receptor antagonist 1 is a potent succinate receptor antagonist. Succinate/succinate receptor antagonist 1 interrupts succinate signals in gingival tissue and inhibits the activation of SucnRl Antagonist 1. Its IC50 value is 20 μsouth of the coast. Succinate/succinate receptor antagonist 1 can be used to treat periodontal disease.
    • $34
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
    Glucocorticoid receptor agonist-1 phosphate Gly-Glu TFA
    T823032734877-83-7
    Glucocorticoid Receptor Agonist-1 Phosphate Gly-Glu (TFA) serves as a cleavable linker for the synthesis of Antibody-Drug Conjugates (ADCs).
    • Inquiry Price
    Size
    QTY
    TargetMol | Inhibitor Sale
    GABA-IN-1
    T82356
    GABA-IN-1 (Compound 6), a GABA inhibitor, exhibits larvicidal and insecticidal properties, achieving a mortality rate of 93% at a concentration of 50 mg/L [1].
    • Inquiry Price
    Size
    QTY
    TargetMol | Inhibitor Sale
    β2AR/M-receptor agonist-1
    T747082230520-62-2
    β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and muscarinic receptor. It demonstrates a significant affinity for the β2 adrenoceptor, indicated by an EC50 value of 9.2 nM, and for the muscarinic receptor with a Ki value of 30.2 nM. Furthermore, its MABA activity is highlighted by an EC50 value of 4.0 nM [1].
    • Inquiry Price
    Size
    QTY
    TargetMol | Inhibitor Sale
    σ1 Receptor antagonist-1
    T92441204401-49-9
    σ1 Receptor antagonist-1 is a selective sigma 1 receptor antagonist.
    • $39
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
    GABA-AT-IN-1
    T62185242148-96-5
    GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.
    • $2,140
    6-8 weeks
    Size
    QTY
    Vanilloid receptor antagonist 1
    T9247871814-52-7
    Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.
    • $117
    In Stock
    Size
    QTY
    Glucocorticoid receptor modulator 1
    T721022868357-11-1
    Glucocorticoid receptor modulator 1 is a potent, orally active, non-steroidal selective glucocorticoid receptor modulator, exhibiting IC50 values of 9 nM and 130 nM against NF-κB and AP-1, respectively. It effectively reduces the expression of inflammatory factors such as IL-6, IL-1β, and TNF-α, and alleviates dermatitis in mice.
    • $987
    6-8 weeks
    Size
    QTY
    Protease-Activated Receptor-1 antagonist 2
    T742661454588-34-1
    Protease-Activated Receptor-1 Antagonist 2 is an orally active antagonist of protease-activated receptor-1 (PAR-1), demonstrating significant potency with an IC 50 of 7 nM. It exhibits favorable pharmacokinetic characteristics, making it valuable in cardiovascular disease (CVD) research, including studies on atherosclerosis and restenosis [1].
    • Inquiry Price
    Size
    QTY
    Glucocorticoid receptor agonist-1 Ala-Ala-Mal
    T741162166376-51-6
    Glucocorticoid receptor agonist-1 Ala-Ala-Mal (compound 88), a glucocorticosteroid and glucocorticoid receptor agonist, can be conjugated with Adalimumab to formulate an ADC [1].
    • Inquiry Price
    Size
    QTY
    Protease-Activated Receptor-1, PAR-1 Agonist TFA
    T36288
    Protease-Activated Receptor-1 (PAR-1) Agonist TFA is a selective peptide that acts as an agonist for the proteinase-activated receptor-1 (PAR-1). Corresponding to the tethered ligand of PAR-1, this compound mimics the actions of thrombin through the PAR-1 receptor[1][2].
    • Inquiry Price
    Size
    QTY
    mGlu4 receptor agonist 1
    T617751678501-16-0
    mGlu4 receptor agonist 1 (compound 62) is a highly effective positive allosteric modulator of mGlu4 receptors, displaying an EC 50 of 308 nM. Additionally, it exhibits noteworthy anxiolytic and antipsychotic properties [1].
    • $1,520
    6-8 weeks
    Size
    QTY
    Glucocorticoid receptor-IN-1
    T635512662908-25-8
    Glucocorticoid receptor-IN-1 is a selective regulator of the glucocorticoid receptor (GR) and exhibits anti-inflammatory activity. glucocorticoid receptor-IN-1 has good transcriptional repression, acting on hMMP1 ( IC50: 2.11 nM) and also has a transcriptional activating effect on MMTV (EC50: 5.59 nM).
    • $1,520
    8-10 weeks
    Size
    QTY
    5-HT6/5-HT2A receptor ligand-1
    T612072411088-07-6
    5-HT6/5-HT2A receptor ligand-1 (compound 33) is a dual antagonist for the 5-HT6 and 5-HT2A receptors. It exhibits a K i value of 2 nM and 11 nM for the respective receptors. This compound holds promise for research in neurological and psychiatric disorders [1].
    • $1,520
    6-8 weeks
    Size
    QTY
    CCK-B Receptor Antagonist 1
    T13261168161-71-5
    CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.
    • $45
    5 days
    Size
    QTY
    Adenosine receptor inhibitor 1
    T618502550400-52-5
    Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR). It exhibits exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >1000, >1000 nM. This compound demonstrates notable antinociceptive, anti-inflammatory, and peripheral analgesic properties. Therefore, Adenosine receptor inhibitor 1 holds great promise for investigating cancer and neurodegenerative diseases [1].
    • $1,520
    6-8 weeks
    Size
    QTY
    Substance P Receptor Antagonist 1
    T10121225526-17-0
    Substance P Receptor Antagonist 1 has the potential function in gastrointestinal disorders, inflammatory diseases, respiratory, and central nervous system disorders.
    • $1,520
    6-8 weeks
    Size
    QTY
    Glucagon receptor antagonists-1
    T11413503559-84-0
    Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.
    • $766
    10-14 weeks
    Size
    QTY
    GLP-1 receptor agonist 3
    T114042230200-09-4
    GLP-1 receptor agonist 3 is a GLP-1 receptor agonist,Example 4A-1, has EC50s of 1.1 nM and 13 nM in Clone H6 and Clone C6 cell lines assay, respectively.
    • $1,820
    8-10 weeks
    Size
    QTY
    NOT Receptor Modulator 1
    T122471015231-98-7
    NOT Receptor Modulator 1 (2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol) is a modulator of nuclear receptor NOT.
    • $81
    In Stock
    Size
    QTY
    Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Br
    T778352344809-82-9
    Glucocorticoid Receptor Agonist-1 Phosphate (Gly-Glu-Br) is an antibody-drug conjugate (ADC) linker utilized in the synthesis of ABBV-154, ABBV-927, ABBV-368, and related analogs [1].
    • Inquiry Price
    Size
    QTY
    GLP-1 receptor agonist 13
    T79348
    Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1].
    • Inquiry Price
    Size
    QTY
    CCK-A receptor inhibitor 1
    T12404137004-80-9
    CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the study of diseases related to the digestive system.
    • $700
    6-8 weeks
    Size
    QTY
    Dopamine D3 receptor antagonist-1
    T64024
    Dopamine D3 receptor antagonist-1 is a dopamine D3 receptor selective or multi-targeting ligand with a Ki value of 1.58 nM that has demonstrated therapeutic potential for central nervous system disorders.
    • $1,520
    10-14 weeks
    Size
    QTY
    Dopamine D4 receptor antagonist-1
    T60917444724-92-9
    Dopamine D4 receptor antagonist-1 can be used in schizophrenia study. Dopamine D4 receptor antagonist-1 is a selective antagonist of Dopamine D4 receptor (DRD4). The Ki value of Dopamine D4 receptor antagonist-1 for Hd4.2 is 9.0 nM [1].
    • $1,520
    6-8 weeks
    Size
    QTY
    GIP/GLP-1 dual receptor agonist-1
    T751502807481-02-1
    GIP/GLP-1 dual receptor agonist-1 (compound 4), a receptor agonist for both GIP and GLP-1, shows potential for the research of metabolic disorders and fatty liver diseases, such as nonalcoholic steatohepatitis (NASH) and nonalcoholic fatty liver disease (NAFLD) [1].
    • Inquiry Price
    Size
    QTY
    Sigma-1 receptor antagonist 1
    T129101639220-19-1
    Sigma-1 receptor antagonist 1 is an effective and selective antagonist of sigma-1 receptor. Sigma-1 receptor antagonist 1 exhibits antineuropathic pain activity and can be used in the treatment of neuropathic pain studies.
    • $97
    In Stock
    Size
    QTY