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  • RXFP receptor
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Results for "

rxfp1

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    13
    TargetMol | Inhibitors_Agonists
  • Peptide Products
    1
    TargetMol | Peptide_Products
AZD5462
T638382787501-83-9
AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.
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10-14 weeks
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TargetMol | Inhibitor Hot
RXFP1 receptor agonist-8
T812392941271-76-5
Example 2 (RXFP1 receptor agonist-8) is a potent RXFP1 receptor agonist that suppresses cAMP production in HEK293 cells expressing human RXFP1, exhibiting an EC50 of 1.8 nM [1].
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8-10 weeks
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RXFP1 receptor agonist-7
T812402941484-13-3
RXFP1 receptor agonist-7 (Example 2) is an RXFP1 receptor agonist that effectively inhibits cAMP production in HEK293 cells stably expressing the human RXFP1, with an EC50 of 4.2 nM [1].
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8-10 weeks
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RXFP1 receptor agonist-6
T812412941346-85-4
RXFP1 receptor agonist-6 (Example 7) acts as an agonist for the RXFP1 receptor and effectively suppresses cAMP production in HEK293 cells stably expressing the human RXFP1, with an EC50 of 12 nM [1].
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8-10 weeks
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RXFP1 receptor agonist-5
T812422941385-36-8
RXFP1 receptor agonist-5 (Example 98) is an agonist targeting the RXFP1 receptor, inhibiting cAMP production in HEK293 cells with stable human RXFP1 expression, with an EC50 of 1.3 nM [1].
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8-10 weeks
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RXFP1 receptor agonist-4
T812432941376-76-5
RXFP1 receptor agonist-4 (Example 268) is a potent RXFP1 receptor agonist, shown to effectively suppress cAMP production in HEK293 cells stably expressing the human RXFP1 receptor, with an effective concentration (EC50) of 4.9 nM [1].
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8-10 weeks
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RXFP1 receptor agonist-3
T812442924767-53-1
RXFP1 receptor agonist-3 (Example 223) is an RXFP1 receptor agonist that inhibits cyclic AMP (cAMP) production in HEK293 cells stably expressing human RXFP1, with an EC50 of 2 nM [1].
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8-10 weeks
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RXFP1 receptor agonist-2
T812452924460-54-6
RXFP1 Receptor Agonist-2 (Example 124), an EC50 value of 1 nM [1].
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8-10 weeks
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RXFP1 receptor agonist-1
T812462924619-64-5
RXFP1 receptor agonist-1 (Example 2), suppresses cAMP production in HEK293 cells constitutively expressing the human RXFP1, with an EC50 of 300 nM [1].
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8-10 weeks
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ML-290
T161011482500-76-4
ML-290 is an effective relaxin insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. It shows an EC50 of 94 nM.
    7-10 days
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    Relaxin H3 (human)
    T813001158181-62-4
    Relaxin H3 (human), a relaxin peptide, exhibits antifibrotic effects by activating RXFP1 [1].
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    AZ7976
    T857832813866-27-0
    AZ7976 (Compound 42), a potent and highly selective agonist for Relaxin Family Peptide Receptor 1 (RXFP1) with a pEC 50 value greater than 10.5, operates through an allosteric mechanism to enhance RXFP1's cAMP signaling, which physiologically elevates heart rate. This property makes AZ7976 a valuable tool in cardiovascular disease research [1].
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    3-6 months
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    B7-33
    TP29031818415-56-3
    B7-33 is a single-chain relaxin analog and a selective agonist for relaxin receptor 1 (RXFP1). It binds to RXFP1 and preferentially activates the pERK pathway in cells expressing RXFP1, rather than cAMP. B7-33 serves as an antifibrotic agent and provides cardioprotective effects.
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