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Search Results for " phenylephrine "

18

Compounds

8

Natural Products

Cat No. Product Name Synonyms Targets
T0453L DL-Phenylephrine HCl Eyelo,DL-Phenylephrine hydrochloride
DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.
T35576 Phenylephrine-3-O-Sulfate
Phenylephrine-3-O-sulfate is metabolite of the α1A-adrenergic receptor agonist phenylephrine formed via sulfation.
T68997 L-Phenylephrine
L-Phenylephrine is an alpha-adrenergic agonist used as a mydriatic, nasal decongestant, and cardiotonic agent.
T22033 ARC 239 dihydrochloride Norepinephrine
ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).
T12913 Siguazodan SKF 94836 PDE
Siguazodan (SKF 94836) is an effective, selective, orally active phosphodiesterase III ((PDE-III)) inhibitor with an IC50 of 117 nM. Siguazodan inhibited phenylephrine induced 5-HT release with an IC50 value of 4.2 μM。 S...
T4563 Thonzylamine neohetramine Histamine Receptor
Thonzylamine (neohetramine) is an antihistamine and anticholinergic drug. It is available as combination products with Clofedanol or Phenylephrine for temporary relief of symptoms of common cold, hay fever (allergic rhin...
T23557 Talibegron hydrochloride ZD2079 hydrochloride,ZD 2079 Adrenergic Receptor
Talibegron hydrochloride (ZD2079 hydrochloride) is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Relaxes rat mesenteric artery and isolated aorta in vitro. In...
T30427 Berefrine
Berefrine is an Oxazolidine prodrug of phenylephrine.
T40563 Sandaracopimaric acid
Sandaracopimaric acid is an anti-inflammatory diterpenoid compound that effectively reduces the contraction of phenylephrine-induced pulmonary arteries. With an EC50 of 43.93 μM, it exhibits noteworthy anti-inflammatory ...
T27164 DHP-218 PAK-9,PAK9,PAK 9,DHP218
DHP-218 is a calcium channel antagonist. DHP-218 inhibits Calcium-induced contraction of the rat aorta in high K+ solution with the pA2 value of 9.11. The IC50 value for the inhibitory effects of DHP-218 in high K+-induc...
TP2086 AdTx1
Selective, high affinity, non-competitive α1A adrenoceptor antagonist (Ki = 0.35 nM). Exhibits no significant activity against a range of other GPCRs, including α2A, β1 and β2 adrenoceptors. Antagonizes effects of phenyl...
T73083 Nipradolol KT 210 ; K 351 ; Hypadil,Hypadil,KT 210,K 351
Nipradolol (KT-210; K-351) is a potent blocker of alpha-1-adrenergic receptors . Nipradolol inhibits the increase of intraocular pressure (IOP) in an albino rabbit model induced by Phenylephrine . Nipradolo suppresses th...
T39281 AM404
AM404 is a chemical compound that functions as an inhibitor of endocannabinoid reuptake. It effectively blocks the transport of anandamide, with IC50 values measured in the low micromolar range. Moreover, AM404 exhibits ...
T69127 Moxisylyte
Moxisylyte, also known as thymoxamine, is a drug used in urology for the treatment of erectile dysfunction. It is an α1-adrenergic antagonist. Moxisylyte is also used for the short-term treatment of primary Reynaud's syn...
T35989 CAY10565
S-Nitrosothiols (RSNOs) are a class of molecules that function as exogenous and endogenous nitric oxide (NO) donors. RSNOs found in vivo include proteins such as S-nitrosohemoglobin and S-nitrosoalbumin, as well as low m...
T35987 CAY10563 CAY10563
S-Nitrosothiols (RSNOs) are a class of molecules that function as exogenous and endogenous nitric oxide (NO) donors. RSNOs found in vivo include proteins such as S-nitrosohemoglobin and S-nitrosoalbumin, as well as low m...
T35988 CAY10564
S-Nitrosothiols (RSNOs) are a class of molecules that function as exogenous and endogenous nitric oxide (NO) donors. RSNOs found in vivo include proteins such as S-nitrosohemoglobin and S-nitrosoalbumin, as well as low m...
T36070 (±)5(6)-EET
5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes. In solution, 5(6)-EET degrades into 5,6-DiHET and 5(6)-δ-lactone, which can be converted to 5...
Cat No. Product Name Synonyms Targets
T17310 Phenylephrine L-Phenylephrine,(R)-(-)-Phenylephrine Adrenergic Receptor
Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
T0453 Phenylephrine hydrochloride NCI-c55641,Phenylephrine HCl,(R)-(-)-Phenylephrine hydrochloride Endogenous Metabolite , Adrenergic Receptor
Phenylephrine hydrochloride (NCI-c55641) is a selective agonist of the α1-adrenergic receptor.
T7634 3-Hydroxymandelic Acid Endogenous Metabolite
3-Hydroxymandelic Acid is a metabolite of Phenylephrine.
T5263 P-Hydroxymandelic acid 4-Hydroxymandelic acid Others , Endogenous Metabolite
p-Hydroxymandelic acid (4-Hydroxymandelic acid) is an acidic metabolite of p-octopamine and p-synephrine (p-phenylephrine). It is also a naturally occurring metabolite of tyramine.
T2944 Danshensu sodium salt Sodium Danshensu,(±)-DanShenSu sodium salt,(±)-DanShenSu sodium sal P450 , Autophagy
Danshensu sodium salt (Sodium Danshensu) is sodium salt of danshensu from the widely used Chinese herb Danshen. It can inhibited phenylephrine- and CaCl2-induced vasoconstriction in Ca2+-free medium.
TN1624 Ethyl cinnamate Calcium Channel , ROS , NO Synthase
Ethyl cinnamate has antifungal, and vasorelaxant effects. Ethyl cinnamate can lead to the damage of cell membrane system and metabolic disorder through inducing lipid peroxidation via initiating ROS overproduction. Ethyl...
TN1724 Harmalol hydrochloride Harmidol hydrochloride P450 , Antioxidant
Harmalol hydrochloride (Harmidol hydrochloride) is a β-carboline alkaloid that can be extracted from the seeds of Peganum harmala L. Harmalol hydrochloride is the major metabolite of Harmaline and significantly inhibits ...
TN5061 Stephanine Adrenergic Receptor , Antifection
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of 6.76. Stephanine shows significant antiplasmodial activitie...
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