Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
Applied FilterClear all
TargetMol | Tags By Target
  • Androgen Receptor
    (136)
  • PROTACs
    (14)
  • Apoptosis
    (12)
  • Autophagy
    (8)
  • Endogenous Metabolite
    (7)
  • Estrogen/progestogen Receptor
    (7)
  • Estrogen Receptor/ERR
    (5)
  • Cytochromes P450
    (4)
  • Drug Metabolite
    (4)
  • Others
    (106)
Filter
Search Result
Results for "

androgen

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    300
    TargetMol | Inhibitors_Agonists
  • Compound Libraries
    1
    TargetMol | Compound_Libraries
  • Peptide Products
    7
    TargetMol | Peptide_Products
  • PROTAC Products
    33
    TargetMol | PROTAC
  • Natural Products
    44
    TargetMol | Natural_Products
  • Recombinant Protein
    25
    TargetMol | Recombinant_Protein
  • Isotope Products
    13
    TargetMol | Isotope_Products
  • Antibody Products
    23
    TargetMol | Antibody_Products
Prochloraz
Sporgon, Prelude
T2062567747-09-5
Prochloraz (Prelude) is a broad-spectrum contact imidazole fungicide. Prochloraz inhibits human placental microsomal aromatase in vitro (IC50 = 40 nM). Prochloraz also acts as an estrogen receptor (IC50s = 25 μM) and androgen receptor (IC50 = 4 μM) antagonist, and activates aryl hydrocarbon receptors (EC50 = 1 μM).
  • $34
In Stock
Size
QTY
D4-abiraterone
Δ4-Abiraterone, Delta4-Abiraterone, CB-7627, CB7627, Abiraterone D4A metabolite
T10946154229-21-7
D4-abiraterone is the active metabolite of abiraterone produced by 3β-HSD and is further metabolised by SRD5A.Δ4-Abiraterone is an inhibitor of CYP17A1, 3β-HSD and SRD5A, and an antagonist of the androgen receptor.
    7-10 days
    Inquiry
    Androgen receptor antagonist 1
    T103201338812-36-4In house
    Androgen receptor antagonist 1, an orally available full androgen receptor antagonist (IC50: 59 nM), is utilized in the synthesis of PROTAC AR degraders, achieving 24% and 47% AR protein degradation in LNCaP cells at concentrations of 1 μM and 10 μM, respectively.
    • $1,520
    6-8 weeks
    Size
    QTY
    Vosilasarm
    Testolone, RAD140
    T43581182367-47-0
    RAD140 is an investigational selective androgen receptor modulator (SARM) for the treatment of conditions such as muscle wasting and breast cancer.
    • $34
    In Stock
    Size
    QTY
    Androgen receptor degrader-5
    T2001972902679-11-0
    Androgen receptor degrader-5 (compound 14k) demonstrates superior capabilities, specifically in androgen receptor degradation and antiproliferative activity, showcasing its promising properties.
    • $1,520
    6-8 weeks
    Size
    QTY
    Androgen receptor antagonist 11
    T2012692719816-32-5
    Androgen receptor antagonist 11 (compound N29) is a selective, orally available antagonist.
    • $1,670
    8-10 weeks
    Size
    QTY
    Androgen receptor antagonist 12
    T2016046605-17-0
    Compound EF2 (Androgen receptor antagonist 12) is an orally active antagonist of the androgen receptor (AR) with an IC50 of 0.30 µM. It inhibits the transcriptional activity of mutant AR and the proliferation of AR-positive PCa (prostate cancer) cell lines. Additionally, Compound EF2 blocks the nuclear translocation of AR and suppresses tumor growth in the C4-2B xenograft mouse model. This compound is used for research in prostate cancer.
    • Inquiry Price
    10-14 weeks
    Size
    QTY
    Androgen receptor modulator 3
    T2045931018971-95-3
    Androgen receptormodulator 3 is a selective modulator of the androgen receptor, applied in the study of muscle atrophy.
    • Inquiry Price
    10-14 weeks
    Size
    QTY
    Androgen receptor antagonist 3
    T60987353484-46-5
    Androgen receptor antagonist 3 (Compound C18) exhibits anticancer activity as an antagonist of the androgen receptor (AR) with an IC50 value of 2.4 μM [1].
    • $2,140
    6-8 weeks
    Size
    QTY
    Androgen receptor antagonist 4
    T60988354815-43-3
    Androgen receptor antagonist 4 (Compound AT2) exhibits anticancer activities by potently antagonizing AR transcriptional activity, inhibiting downstream AR target genes, and blocking DHT-induced nuclear translocation of AR. It is an antagonist of the androgen receptor (AR) with an IC50 of 0.15 μM [1].
    • $2,140
    6-8 weeks
    Size
    QTY
    Androgen receptor antagonist 5
    T633242586195-28-8
    Androgen receptor antagonist 5 is a potent antagonist of the androgen receptor (AR) (IC50: 6.17 μM). Androgen receptor antagonist 5 inhibited the proliferation of prostate cancer cells LNCaP and showed antitumor effect in LNCaP xenograft mice model, which can be used to study prostate cancer.
    • $2,140
    8-10 weeks
    Size
    QTY
    Androgen receptor-IN-5
    T790241391944-16-3
    Androgen receptor-IN-5 is a potent inhibitor of the androgen receptor with anticancer properties. It additionally suppresses the synthesis of IL-17A, IL-17F, and INF-γ.
    • Inquiry Price
    8-10 weeks
    Size
    QTY
    Androgen receptor degrader-3
    T798912753650-84-7
    Androgen Receptor Degrader-3 (ARD-3) is a compound that inhibits androgen receptor signaling and promotes the degradation of the receptor, with potential applications in prostate cancer research [1].
    • Inquiry Price
    8-10 weeks
    Size
    QTY
    Androgen receptor degrader-1
    T806332616553-35-4
    Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in cancer research [1].
    • Inquiry Price
    8-10 weeks
    Size
    QTY
    Androgen receptor degrader-2
    T806472616553-33-2
    Androgen Receptor Degrader-2 (Compound 9) is a potent degrader of androgen receptors, with potential application in cancer research [1].
    • Inquiry Price
    8-10 weeks
    Size
    QTY
    Androgen receptor antagonist 9
    T83119915086-32-7
    Androgen Receptor Antagonist 9 (compound 28) serves as an antagonist to the androgen receptor [1].
    • Inquiry Price
    Size
    QTY
    Androgen receptor antagonist 10
    T85648876759-87-4
    Androgen receptor antagonist 10 (compound 6h) serves as an androgen receptor antagonist that effectively reduces wax esters in the golden Syrian hamster model [1].
    • Inquiry Price
    10-14 weeks
    Size
    QTY
    Androgen receptor degrader-4
    T856492505495-83-8
    Androgen receptor degrader-4 (compound 99) is a potent androgen receptor degrader, demonstrating an IC 50 of 3 nM. This compound effectively inhibits the proliferation of prostate cancer cells [1].
    • Inquiry Price
    Inquiry
    Size
    QTY
    A-485
    T140731889279-16-6
    A-485 is a potent and selective catalytic p300 CBP inhibitor with IC50 values of 9.8 nM for p300 and 2.6 nM for CBP.
    • $89
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Hot
    Enzalutamide
    MDV3100
    T6002915087-33-1
    Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP) that activates autophagy, exhibits antitumor activity, and is commonly used in treating desmoplasia-resistant prostate cancer.
    • $40
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Hot
    CSRM617 hydrochloride
    CSRM617 hydrochloride(787504-88-5 Free base)
    T10896L1353749-74-2In house
    CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 (OC2, a master regulator of androgen receptor), with a Kd of 7.43 µM in SPR assays, directly binding to the OC2-HOX domain. CSRM617 hydrochloride induces apoptosis through the appearance of cleaved Caspase-3 and PARP and is well tolerated in the mouse model of prostate cancer [1].
    • $35
    In Stock
    Size
    QTY
    celiprolol hydrochloride
    Selectrol, Selecor
    T124457470-78-7In house
    Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity. It is used in the management of ANGINA PECTORIS and HYPERTENSION.
    • $71
    3-6 months
    Size
    QTY
    Topterone
    Win 17665
    T1318760607-35-4In house
    Topterone (Win 17,665) is a potent topical antiandrogen that inhibits the stimulation of lumbar organ development by testosterone and dihydrotestosterone in castrated immature male hamsters.
    • $700
    In Stock
    Size
    QTY
    Seviteronel
    VT-464
    T13312L1610537-15-9In house
    Seviteronel (VT-464) is a novel CYP17 cleavage enzyme inhibitor and androgen receptor antagonist used in breast and prostate cancer research.
    • $113 TargetMol
    In Stock
    Size
    QTY