T1681

Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.

RWJ-51204 is a selective adenosine A2A receptor antagonist and a partial agonist of GABA(A) receptor (IC50: 0.2-2 nM). It has neuroprotective and movement-improving effects and can be used in research related to Parkinson's disease.

S 18986 is a selective, orally active, brain-penetrant positive allosteric modulator of AMPA-type receptors that enhances cognition in rodents by inducing the release of noradrenaline and acetylcholine in the rat hippocampus, subsequently improving object-recognition memory.

S-2474, an inhibitor of COX-2 and 5-lipoxygenase, has anti-inflammatory and neuroprotective activities and inhibits Abeta (25 - 35) and Abeta (1 - 40) induced cell death.

Ruzadolane (formerly known as UP 26-91) is a 5-hydroxytryptamine receptor antagonist developed as a non-narcotic central analgesic for the treatment of anxiety disorders and pain.

RWJ-67657 (JNJ 3026582) is an orally active, selective p38α and p38β MAPK inhibitor (IC50s: 1 and 11 μM, respectively), with no activity at p38γ and p38δ, and demonstrates cardioprotective effects.

RX-3117 (fluorocyclopentenylcytosine) is a novel a cytidine analog. RX-3117 displays anticancer activity in several cancer cell lines, including gemcitabine-resistant variants.

RX 67668 is a muscle relaxant used to relieve skeletal muscle fatigue. RX 67668 is an effective cholinesterase inhibitor (IC50: 5 μM for both acetylcholinesterase and butyrylcholinesterase). RX 67668 can reverse the neuromuscular blockade induced by D-tub

RY796 is a selective voltage-gated potassium (KV2) channel inhibitor that inhibits KV2.1 and KV2.2, used in research on neurological disorders.

S-8921 is an inhibitor of ileal Na+/bile acid cotransporter.

S-acetyl-PEG3-alcohol, a PEG-based linker (PROTACs), connects essential ligands to form PROTAC molecules, facilitating selective protein degradation via the ubiquitin-proteasome system within cells.

Aminophylline-D6 is a deuterated compound of Aminophylline. Aminophylline (T1681) has a CAS number of 317-34-0. Aminophylline (T1681) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.