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Search Result

Search Results for " aromatase "

Targets

Aromatase Others

50

Compounds

11

Natural Products

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T60022 Aromatase-IN-2 Others
Aromatase-IN-2 has anti-inflammatory, antitumor and antiasthmatic effects.
T60006 Aromatase inhibitor 23 Others
Aromatase inhibitor 23 is an inhibitor that target protein-protein interactions in RAD51 family of recombinases.
T61444 Nonsteroidal aromatase inhibitor 1
Nonsteroidal aromatase inhibitor 1 (Compound 13h) effectively inhibits the enzyme CYP19A1 with an IC50 value of 0.09 nM. Due to its potent inhibitory activity, Nonsteroidal aromatase inhibitor 1 holds promise for researc...
T61463 Monoamine oxidase/Aromatase-IN-1
Monoamine oxidase/Aromatase-IN-1 (compound 2q) is a potent dual inhibitor of monoamine oxidase (MAO) and aromatase, with IC50 values of 39 nM and 31 nM for MAO-B and aromatase, respectively. It holds significant potentia...
T7197 Fadrozole Aromatase
Fadrozole is a nonsteroidal aromatase inhibitor with potential antineoplastic activity(IC50 : 6.4 nM)
T0393 Anastrozole ZD1033 Aromatase
Anastrozole (ZD1033)(ZD1033), a potent and highly selective aromatase (CYP19) inhibitor (IC50 = 15 nM), has no obvious effect on adrenocorticoid hormone synthesis.
T11991 Mefentrifluconazole P450 , Antifungal
Mefentrifluconazole is a potent, selective and orally active fungal CYP51 (Kd= 0.5 nM) inhibitor, but shows less inhibitory activity on human aromatase (IC50=0.92 μM). Mefentrifluconazole is a novel azole derivative and ...
T7556 Fadrozole hydrochloride CGS 16949A Aromatase
Fadrozole hydrochloride (CGS 16949A) is a model aromatase inhibitor that has been shown to suppress estrogen production in the ovaries of fish.
T1103 Aminoglutethimide DL-Aminoglutethimide,BA-16038,NSC-330915 Aromatase
Aminoglutethimide (BA-16038), an aromatase inhibitor, is used in the therapy of advanced BREAST Y.
T20625 Prochloraz Sporgon,Prelude Estrogen Receptor/ERR , AhR , Androgen Receptor , Antifungal
Prochloraz (Prelude) is a broad-spectrum contact imidazole fungicide. Prochloraz inhibits human placental microsomal aromatase in vitro (IC50 = 40 nM). Prochloraz also acts as an estrogen receptor (IC50s = 25 μM) and and...
T1587 Exemestane EXE,FCE 24304,PNU155971 Aromatase
Exemestane (EXE) is an Aromatase Inhibitor. The mechanism of action of exemestane is as an Aromatase Inhibitor.
T4281 Endoxifen (E/Z)-N-desmethyl-4-hydroxy Tamoxifen,(E/Z)-Endoxifen Estrogen Receptor/ERR , Aromatase , Estrogen/progestogen Receptor , Parasite , Drug Metabolite
(E/Z)-Endoxifen ((E/Z)-Endoxifen) is an active metabolite of tamoxifen produced by the sequential action of cytochrome P450 (CYP) isoforms, including CYP2D6. It is a strong anti-estrogen, as it has an approximately 100-f...
T71708 Minamestane Aromatase
Minamestane is a novel irreversible aromatase inhibitor.Minamestane induces time-dependent inhibition of human placental aromatase with a half-life of 4 minutes and a K of 59 nM.Minamestane has antitumor activity.
T27320 Finrozole MPV 2213ad,MPV-2213ad,MPV 2213,MPV-2213,MPV2213ad Aromatase
Finrozole (MPV 2213ad) is a novel selective aromatase inhibitor that is partially reversible for breast development.
T23549 YM 511 P450 , Aromatase
YM 511 is a highly specific non-steroidal aromatase inhibitor. YM 511 inhibits aromatase activities in microsomes from rat ovary and human placenta competitively (IC50s of 0.4 and 0.12 nM, respectively). YM 511 slightly ...
T27918 LY 43578 LY-43578,LY43578 P450 , Aromatase
LY 43578 is an orally active aromatase inhibitor. LY43578 could inhibit O-demethylation of P-450-dependent p-nitroanisole and N-demethylation of ethylmorphine (IC50 of 0.3 and 5 μm, respectively) in rat liver microsomes....
T72310 Antibacterial agent 132 Antifungal
Antibacterial agent 132 showed antimicrobial activity against C. parapsilosis (ATCC 22019) and C. krusei (ATCC 6258) with MIC90 values of <0.06 μg/mL and 62.50 μg/mL, respectively. Antibacterial agent 132 inhibited aroma...
T26322 Vorozole R83839,R 83839,R-83839,(+)-Vorozole,R83842 P450 , Aromatase
Vorozole (R83842) is an orally active, potent, and selective nonsteroidal aromatase inhibitor.Vorozole exhibits antitumor activity in vivo and may be used in the study of breast cancer.
T2280 Endoxifen (Z-isomer) Endoxifen Z-isomer Estrogen Receptor/ERR , EGFR , Potassium Channel , Estrogen/progestogen Receptor , HER
Endoxifen Z-isomer (EDX) is a key active metabolite of tamoxifen (TAM) with higher affinity and specificity to estrogen receptors that also inhibits aromatase activity.
T26322L (-)-Vorozole (-)-Vorozole(Isomer-129731-10-8) P450 , Aromatase
(-)-Vorozole is an orally active non-steroidal aromatase inhibitor with potency and selectivity. (-)-Vorozole has demonstrated antitumor activity in in vivo experiments. (-)-Vorozole is used in the study of breast cancer...
T6827L Endoxifen hydrochloride
Endoxifen hydrochloride, a principal active metabolite of Tamoxifen (TAM), exhibits heightened affinity and specificity towards the estrogen receptor and possesses aromatase inhibitory capability. It holds promise for br...
T11847L Liarozole R75251 dihydrochloride P450 , Retinoid Receptor
Liarozole (R75251 dihydrochloride) is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 1...
T12319 Org30958 Aromatase
Org30958 is a potent inhibitor of aromatase in vivo.
T27369 FR 901537 FR901537,FR-901537
FR 901537 is a new aromatase inhibitor with antitumor effects.
T70558 Org 33201
Org 33201 is a potent aromatase inhibitor.
T71410 Cgs 18320B
Cgs 18320B is a non-steroidal aromatase inhibitor
T27922 LY 56110 LY56110,LY-56110
LY 56110 is a novel nonsteroidal aromatase inhibitor.
T7197L Fadrozole HCl hydrate Fadrozole,CGS-16949A,Fadrozole hydrochloride hemihydrate,CGS16949A,CGS 16949A
Fadrozole is a selective inhibitor of aromatase. It also effective in the treatment of estrogen-dependent diseases including breast cancer.
T70404 MPV-2213AD
MPV-2213AD is an aromatase inhibitor.
T71897 Vatalanib succinate
Vatalanib succinate is a VEGFR, PDGFR-β, c-Kit, c-Fms, and aromatase inhibitor.
T30837 Cgp 47645 Leflutrozole,Cgp-47645,Cgp47645
CGP 47645 (Leflurozole) is an oral active non-steroidal aromatase inhibitor and antitumor agent with anti-tumor and endocrine effects.
T30834 Cgp 45688 Cgp45688,Cgp-45688
CGP 45688 is an oral active non-steroidal aromatase inhibitor with anti-tumor and endocrine effects on rat breast tumors.
T20683 Letrozole related compound B Letrozole specified impurity A
Letrozole related compound B is an impurity of aromatase inhibitor.
T25716 Liarozole fumarate Liazal,R85246,R-85246,R 85246
Liarozole fumarate is used as a retinoic acid metabolism blocking agent (RAMBA) and an aromatase inhibitor.
T27868 LY 113174 LY-113174,LY113174
LY 113174, a novel nonsteroidal aromatase inhibitor, may prove useful in the treatment of estrogen-dependent diseases.
T61787 SYN20028567
SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].
T81012 Testololactone
Testololactone, an aromatase inhibitor, may be utilized in breast carcinoma research [1].
T71073 Tan 931
Tan 931 is a nonsteroidal aromatase inhibitor that was first isolated from the culture filtrate of a soil isolate fungus, No. 8974
T6060L Anabasine HCl BB-NC-0036,CCG-38440,H-8174,AR-1H7273,ZX-BK000320,ST-24041653
Anabasine HCl is used as a clinical biomarker for tobacco smoke exposure and as an insecticide. It is also a depolarizing NMJ blocker, aromatase inhibitor, nAChr antagonist, and teratogen found in species of Nicotiana.
T38424 (R)-Fadrozole FAD286,(R)-CGS 16949A free base,(R)-Fadrozole
(R)-Fadrozole ((R)-CGS 16949A; FAD286) is a potent nonsteroidal inhibitor. (R)-Fadrozole also inhibits human placental aromatase (pIC 50 = 6.17) and aldosterone biosynthesis. (R)-Fadrozole reverses cardiac fibrosis in sp...
T71010 Norendoxifen
Norendoxifen, also known as 4-hydroxy-N, N-didesmethyltamoxifen, is a nonsteroidal aromatase inhibitor of the triphenylethylene group that was never marketed. It is an active metabolite of the selective estrogen receptor...
T80057 Cytochrome P450 reductase
Cytochrome P450 reductase, a NADPH-cytochrome reductase, facilitates an optimal conformation of aromatase for substrate binding [1].
T61919 Anticancer agent 78
Anticancer agent 78 has anti-aromatase activity (IC50=0.9 μM）。 Anticancer agent 78 is an effective anticancer agent, showing cytotoxicity. Anticancer agent 78 has research potential in breast cancer.
T11847 Liarozole dihydrochloride R75251 dihydrochloride Others
Liarozole dihydrochloride is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lya...
T35676 17β-hydroxy Exemestane
17β-hydroxy Exemestane is the primary active metabolite of exemestane . It is formed by metabolism of exemestane by the cytochrome P450 (CYP) isoforms CYP1A and CYP4A11. 17β-hydroxy Exemestane is an aromatase inhibitor (...
T25716L Liarozole HCl R75251,Liarozole hydrochloride,R 75251,R-75251
Liarozole HCl is a benzimidazole derivative with antineoplastic activity. As a retinoic acid metabolism blocking agent, liarozole inhibits CYP450-dependent all-trans-retinoic acid (ATRA)-4-hydroxylase, leading to an incr...
T83907 10-Chloroestra-1,4-diene-3,17-dione 10-chloro-1,4-Estradiene
10-Chloroestra-1,4-diene-3,17-dione acts as an estrogen receptor α (ERα) agonist, enhancing reporter gene expression in S. cerevisiae with an EC50 of 0.36 nM for the human receptor. Additionally, it functions as an aroma...
T71578 Endoxifen mesylate
Endoxifen, also known as N-desmethyl-4-hydroxytamoxifen, is a chemical that is under development for estrogen receptor-positive breast cancer. It is also being evaluated as an antipsychotic for treatment of mania and ot...
T37560 Nidulin
Nidulin is a depsidone originally isolated from A. nidulans. It is active against the bacteria M. tuberculosis and M. ranoe, as well as the fungi T. tonsurans and M. audouini. It also inhibits the growth of methicillin-r...
T78590 Dibenzylfluorescein DBF
Dibenzylfluorescein (DBF), a fluorogenic probe (Fluorescent dye), serves as a substrate for various cytochrome P450 (CYP) isoforms, such as CYP3A4, CYP2C8, CYP2C9, CYP2C19, and aromatase (CYP19). It is commonly utilized ...

Compounds

Aromatase-IN-2
T60022
Synonym:
Target: Others
Aromatase inhibitor 23
T60006
Synonym:
Target: Others
Nonsteroidal aromatase inhibitor 1
T61444
Synonym:
Target:
Monoamine oxidase/Aromatase-IN-1
T61463
Synonym:
Target:
Fadrozole
T7197
Synonym:
Target: Aromatase
Anastrozole
T0393
Synonym: ZD1033
Target: Aromatase
Mefentrifluconazole
T11991
Synonym:
Target: P450, Antifungal
Fadrozole hydrochloride
T7556
Synonym: CGS 16949A
Target: Aromatase
Aminoglutethimide
T1103
Synonym: DL-Aminoglutethimide,BA-16038,NSC-330915
Target: Aromatase
Prochloraz
T20625
Synonym: Sporgon,Prelude
Target: Estrogen Receptor/ERR, AhR, Androgen Receptor, Antifungal
Exemestane
T1587
Synonym: EXE,FCE 24304,PNU155971
Target: Aromatase
Endoxifen
T4281
Synonym: (E/Z)-N-desmethyl-4-hydroxy Tamoxifen,(E/Z)-Endoxifen
Target: Estrogen Receptor/ERR, Aromatase, Estrogen/progestogen Receptor, Parasite, Drug Metabolite
Minamestane
T71708
Synonym:
Target: Aromatase
Finrozole
T27320
Synonym: MPV 2213ad,MPV-2213ad,MPV 2213,MPV-2213,MPV2213ad
Target: Aromatase
YM 511
T23549
Synonym:
Target: P450, Aromatase
LY 43578
T27918
Synonym: LY-43578,LY43578
Target: P450, Aromatase
Antibacterial agent 132
T72310
Synonym:
Target: Antifungal
Vorozole
T26322
Synonym: R83839,R 83839,R-83839,(+)-Vorozole,R83842
Target: P450, Aromatase
Endoxifen (Z-isomer)
T2280
Synonym: Endoxifen Z-isomer
Target: Estrogen Receptor/ERR, EGFR, Potassium Channel, Estrogen/progestogen Receptor, HER
(-)-Vorozole
T26322L
Synonym: (-)-Vorozole(Isomer-129731-10-8)
Target: P450, Aromatase
Endoxifen hydrochloride
T6827L
Synonym:
Target:
Liarozole
T11847L
Synonym: R75251 dihydrochloride
Target: P450, Retinoid Receptor
Org30958
T12319
Synonym:
Target: Aromatase
FR 901537
T27369
Synonym: FR901537,FR-901537
Target:
Org 33201
T70558
Synonym:
Target:
Cgs 18320B
T71410
Synonym:
Target:
LY 56110
T27922
Synonym: LY56110,LY-56110
Target:
Fadrozole HCl hydrate
T7197L
Synonym: Fadrozole,CGS-16949A,Fadrozole hydrochloride hemihydrate,CGS16949A,CGS 16949A
Target:
MPV-2213AD
T70404
Synonym:
Target:
Vatalanib succinate
T71897
Synonym:
Target:
Cgp 47645
T30837
Synonym: Leflutrozole,Cgp-47645,Cgp47645
Target:
Cgp 45688
T30834
Synonym: Cgp45688,Cgp-45688
Target:
Letrozole related compound B
T20683
Synonym: Letrozole specified impurity A
Target:
Liarozole fumarate
T25716
Synonym: Liazal,R85246,R-85246,R 85246
Target:
LY 113174
T27868
Synonym: LY-113174,LY113174
Target:
SYN20028567
T61787
Synonym:
Target:
Testololactone
T81012
Synonym:
Target:
Tan 931
T71073
Synonym:
Target:
Anabasine HCl
T6060L
Synonym: BB-NC-0036,CCG-38440,H-8174,AR-1H7273,ZX-BK000320,ST-24041653
Target:
(R)-Fadrozole
T38424
Synonym: FAD286,(R)-CGS 16949A free base,(R)-Fadrozole
Target:
Norendoxifen
T71010
Synonym:
Target:
Cytochrome P450 reductase
T80057
Synonym:
Target:
Anticancer agent 78
T61919
Synonym:
Target:
Liarozole dihydrochloride
T11847
Synonym: R75251 dihydrochloride
Target: Others
17β-hydroxy Exemestane
T35676
Synonym:
Target:
Liarozole HCl
T25716L
Synonym: R75251,Liarozole hydrochloride,R 75251,R-75251
Target:
10-Chloroestra-1,4-diene-3,17-dione
T83907
Synonym: 10-chloro-1,4-Estradiene
Target:
Endoxifen mesylate
T71578
Synonym:
Target:
Nidulin
T37560
Synonym:
Target:
Dibenzylfluorescein
T78590
Synonym: DBF
Target:
Cat No. Product Name Synonyms Targets
T7999 7-Hydroxyflavanone Anti-infection
7-Hydroxyflavanone shows antimicrobial activity against Streptococcus pneumoniae clinical isolates.
T1590 Letrozole CGS 20267 Aromatase , Autophagy
Letrozole (CGS 20267) is an Aromatase Inhibitor. The mechanism of action of letrozole is as an Aromatase Inhibitor.
T2O2744 Alpha-Naphthoflavone 7,8-benzoflavone Aromatase
alpha-Naphthoflavone (7,8-benzoflavone), a synthetic flavonoid, is a potent inhibitor of aromatase with an I50 value of 0.5 μM.
T6917 Oleuropein Apoptosis , Aromatase , ROS , PPAR
Oleuropein is an antioxidant polyphenol isolated from olive leaf.
T0530 Flavanone 2-Phenyl-4-chromanone,4-Flavanone,2,3-Dihydroflavone,2-Phenylchroman-4-one Others , Aromatase
Flavanone (2-Phenylchroman-4-one)s from citrus fruits have also been shown to exert beneficial effects on human vascular function. In particular, chronic interventions with orange juice, or the pure flavanone hesperidin,...
TN3987 Eriodictyol chalcone Anti-infection , Aromatase
Eriodictyol chalcone has anti-plasmodial effects on P. falciparum growth.
T3899 Calceolarioside B Desrhamnosyl isoacteoside,Nuomioside A Aromatase
Calceolarioside B (Desrhamnosyl isoacteoside) displays inhibition of aromatase. Calceolarioside B displays inhibition of human recombinant PKCalpha.
T3390 Obacunone Apoptosis , Aromatase , p38 MAPK
Obacunone has cytotoxicity in androgen-dependent human prostate Y cells. Obacunone exerts an antivirulence effect on S. Typhimurium and may serve as a lead compound for development of antivirulence strategies for S. Typh...
TN1674 Garcinone D Reactive Oxygen Species , Nrf2 , STAT
Garcinone D shows significant cytotoxicity against the CEM-SS cell line, with IC(50) value of 3.2 microg/ml; it exhibits dose-dependent enzyme-based microsomal aromatase inhibitory activity. Garcinone D inhibits p65 acti...
TN4605 Myriceric acid B HIV Protease
Myriceric acid B is a potent HIV-1 entry inhibitor targeting gp41 and can serve as a lead compound for developing novel anti-HIV-1 drug. Myriceric acid B scavenges DPPH free radicals with IC50 value of 21.8 uM, it inhibi...
TN4307 Isolimonexic acid BCL , Caspase , COX , p53
Isolimonexic acid exhibits cytotoxicity on MCF-7 cell lines, it also inhibits Panc-28 cancer cell growth.

Natural Products

7-Hydroxyflavanone
T7999
Synonym:
Target: Anti-infection
Letrozole
T1590
Synonym: CGS 20267
Target: Aromatase, Autophagy
alpha-Naphthoflavone
T2O2744
Synonym: 7,8-benzoflavone
Target: Aromatase
Oleuropein
T6917
Synonym:
Target: Apoptosis, Aromatase, ROS, PPAR
Flavanone
T0530
Synonym: 2-Phenyl-4-chromanone,4-Flavanone,2,3-Dihydroflavone,2-Phenylchroman-4-one
Target: Others, Aromatase
Eriodictyol chalcone
TN3987
Synonym:
Target: Anti-infection, Aromatase
Calceolarioside B
T3899
Synonym: Desrhamnosyl isoacteoside,Nuomioside A
Target: Aromatase
Obacunone
T3390
Synonym:
Target: Apoptosis, Aromatase, p38 MAPK
Garcinone D
TN1674
Synonym:
Target: Reactive Oxygen Species, Nrf2, STAT
Myriceric acid B
TN4605
Synonym:
Target: HIV Protease
Isolimonexic acid
TN4307
Synonym:
Target: BCL, Caspase, COX, p53

Recombinant Proteins

Species：
Human (1)
Expression System：
E. coli (1)
Tag：
N-terminal 6xHis-tagged (1)
Cat No. Product Name Species Expression System
TMPH-00956 Aromatase/CYP19A1 Protein, Human, Recombinant (His) Human E. coli
Aromatase/CYP19A1 Protein, Human, Recombinant (His) is expressed in E. coli.
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