GPCR-G Protein-Others

Cat.No.	Product Name	Information	Area
T5150	Treprostinil	Treprostinil is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).	Cardiovascular system
T5148	Atosiban acetate	Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an i...	Others
T4996	Atosiban	Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as a...
T5018	Leuprorelin	Leuprolide is an agonist at pituitary GnRH receptors.GnRH receptor Leuprorelin is a g...
T5014	Prostaglandin E2 (PGE2)	Prostaglandin E2 is a hormone-like substance that participate in a wide range of body...
T5100	DJ-V159	DJ-V159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6...
T4546	Dinoprost Tromethamine	Dinoprost(Prostaglandin F2α) tromethamine salt is a naturally occurring prostaglandin...	Others
T4648	TC-G-1008	TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat ...	Metabolic Disease
T4390	ML221	ML221 is a potent?apelin /APJ?functional antagonist, inhibiting apelin-13-mediated ac...
T1418	Bucladesine sodium salt	Bucladesine, PKA activator, is a cyclic nucleotide derivative that mimics the action ...	anti-infection
T4278	AM966	AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses L...	cancer
T4300	AZD2098	AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research...	Inflammation
T7040	Angiotensin II human	Angiotensin II is mediated by AT1 and AT2 receptors. AT1 and AT2 receptors have seven...	cancer
T4186	AC-264613	AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 s...	Others
T4540	ML 18	ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of...	Others
T4500	ADX88178	ADX88178 is a potent positive allosteric modulator for metabotropic glutamate recepto...	Others
T4352	SB-756050	SB756050 is a specific TGR5 agonist.	Others
T4119	Octreotide Acetate	Octreotide acetate is a potent, long-acting synthetic somatostatin octapeptide analog...	Metbolism/ Cancer
T4102	Goserelin acetate	Goserelin acetate is a synthetic long-acting agonist of gonadotropin-releasing hormon...	Cancer
T4083	BAR 501	BAR501 is an effective and specific GPBAR1 agonist (EC50: 1 μM).	Other
T3520	Setipiprant	Setipiprant is an orally available, selective CRTH2 antagonist (IC50: 6.0 nM). CRTH2 ...	Others
T4016	BMS-986020	BMS-986020 is a selective antagonist of LPA1.	Others
T3993	BQCA	BQCA a highly selective allosteric modulator of the M1 mAChR.	Others
T3967	Exendin-4	Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). E...	Others
T3965	Fevipiprant	Fevipiprant is a selective, potent, reversible competitive CRTh2 antagonist.	Others
T3565	UV0155041	UV0155041 is an effective and positive allosteric modulator/allosteric agonist at mGl...	Others
T3422	GRA-Ex-25	GRA-Ex-25 is an inhibitor of glucagon receptor.	Other
T3148	Verlukast sodium	MK-571 is a selective, orally active?antagonist of the CysLT1 receptor. MK571 is a mu...	Respiratory system/ Cardiovascular system
T3630	Relugolix	Relugolix is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or...	Cancer/ Nervous system
T7013	Vorapaxar	Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) an...	Others

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