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GPCR-G Protein-Others
Cat.No. Product Name Information Area
T5150 Treprostinil Treprostinil is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM). Cardiovascular system
T5148 Atosiban acetate Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an i... Others
T4996 Atosiban

Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as a...

T5018 Leuprorelin Leuprolide is an agonist at pituitary GnRH receptors.GnRH receptor Leuprorelin is a g...
T5014 Prostaglandin E2 (PGE2) Prostaglandin E2 is a hormone-like substance that participate in a wide range of body...
T5100 DJ-V159 DJ-V159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6...
T4546 Dinoprost Tromethamine Dinoprost(Prostaglandin F2α) tromethamine salt is a naturally occurring prostaglandin... Others
T4648 TC-G-1008 TC-G-1008 is a GPR39 (zinc receptor) agonist (EC50 values are 0.4 and 0.8 nM for rat ... Metabolic Disease
T4390 ML221 ML221 is a potent?apelin /APJ?functional antagonist, inhibiting apelin-13-mediated ac...
T1418 Bucladesine sodium salt Bucladesine, PKA activator, is a cyclic nucleotide derivative that mimics the action ... anti-infection
T4278 AM966 AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses L... cancer
T4300 AZD2098 AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research... Inflammation
T7040 Angiotensin II human Angiotensin II is mediated by AT1 and AT2 receptors. AT1 and AT2 receptors have seven... cancer
T4186 AC-264613 AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 s... Others
T4540 ML 18 ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of... Others
T4500 ADX88178 ADX88178 is a potent positive allosteric modulator for metabotropic glutamate recepto... Others
T4352 SB-756050 SB756050 is a specific TGR5 agonist. Others
T4119 Octreotide Acetate Octreotide acetate is a potent, long-acting synthetic somatostatin octapeptide analog... Metbolism/ Cancer
T4102 Goserelin acetate Goserelin acetate is a synthetic long-acting agonist of gonadotropin-releasing hormon... Cancer
T4083 BAR 501 BAR501 is an effective and specific GPBAR1 agonist (EC50: 1 μM). Other
T3520 Setipiprant Setipiprant is an orally available, selective CRTH2 antagonist (IC50: 6.0 nM). CRTH2 ... Others
T4016 BMS-986020 BMS-986020 is a selective antagonist of LPA1. Others
T3993 BQCA BQCA a highly selective allosteric modulator of the M1 mAChR. Others
T3967 Exendin-4

Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). E...

T3965 Fevipiprant Fevipiprant is a selective, potent, reversible competitive CRTh2 antagonist. Others
T3565 UV0155041 UV0155041 is an effective and positive allosteric modulator/allosteric agonist at mGl... Others
T3422 GRA-Ex-25 GRA-Ex-25 is an inhibitor of glucagon receptor. Other
T3148 Verlukast sodium MK-571 is a selective, orally active?antagonist of the CysLT1 receptor. MK571 is a mu... Respiratory system/ Cardiovascular system
T3630 Relugolix Relugolix is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or... Cancer/ Nervous system
T7013 Vorapaxar Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) an... Others