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Cat.No. Product Name Information Area
T4528 Tyrphostin AG 528 Tyrphostin AG 528 is an inhibitor of EGFR (IC50: 4.9 μM) and ErbB2 (IC50: 2.1 μM).
T4205 AG 494 AG-494 is an inhibitor of epidermal growth factor receptor kinase.
T3506 Nazartinib Nazartinib (EGF816, NVS-816) is a covalent, irreversible, mutant-selective EGFR inhib... Others
T3545 RG 13022 RG13022 is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of ... Others
T3554 RG 14620 RG14620 is an epidermal growth factor receptor (EGFR) inhibitor. Cancer
T3870 Cyasterone Cyasterone, a natural EGFR inhibitor, can inhibit the growth of A549 and MGC823 cells... Others
T3721 Avitinib maleate Avitinib maleate is a pyrrolopyrimidine-based irreversible epidermal growth factor re... Cancer
T3634 Osimertinib mesylate AZD-9291 mesylate is an irreversible and mutant-selective EGFR inhibitor. Cancer
T3659 AZD3759 AZD3759 is an orally active, effective and central nervous system-penetrant EGFR inhi... Cancer
T3024 Avitinib Avitinib, also known as AC0010 or AC0010MA, is an orally available, irreversible, epi... Cancer
T6932 PD168393 PD168393 is an irreversible EGFR inhibitor (IC50: 0.70 nM), irreversibly alkylate Cys... Others
T6918 Olmutinib Olmutinib is an orally available small molecule, a mutant-selective inhibitor of epid... Others
T6908 NSC228155 NSC228155 is an activator of EGFR, binding to the sEGFR dimerization domain II and mo... Others
T6824 EAI045 EAI045, an allosteric inhibitor, targets towards drug-resistant EGFR mutants but avoi... Others
T3402 Ginsenoside Rg3new Ginsenoside Rg3 possess an ability to inhibit the lung metastasis of tumor cells via ... Others
T6734 WZ8040 WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor, does not inhibit... Cancer
T6733 WZ3146 WZ3146 is a mutant-selective irreversible inhibitor of EGFR(L858R) and EGFR(E746_A750... Cancer
T6619 OSI-420 OSI-420 is the active metabolite of Erlotinib (EGFR inhibitor with IC50 of 2 nM).
T6427 Butein Butein, a plant polyphenol, is isolated from Rhus verniciflua. It can inhibit the act... Cancer
T2501 Canertinib dihydrochloride Canertinib dihydrochloride is the hydrochloride salt of an orally bio-available quina... Cancer
T6238 WZ4002 WZ4002 is a mutant-selective EGFR inhibitor for EGFR(L858R) and EGFR(T790M) with IC50... Cancer
T6153 Icotinib Icotinib is an orally available quinazoline-based inhibitor of epidermal growth facto... Others
T6136 Canertinib Canertinib is a pan-erbB tyrosine kinase inhibitor which work against esophageal squa... Cancer
T6124 Mubritinibnew Mubritinib (TAK-165) is a potent inhibitor of HER2/ErbB2 with IC50 of 6 nM. Cancer
T6039 TAK-285 TAK-285 is a novel dual HER2 and EGFR(HER1) inhibitor with IC50 of 17 nM and 23 nM, >... Cancer
T6008 CNX-2006 CNX-2006 is a novel irreversible mutant-selective EGFR inhibitor with IC50 of < 20 nM... Cancer
T2995 Chrysophanic Acid Chrysophanic acid is an EGFR/mTOR pathway inhibitor, which can be found in rhubarb, a... Cancer
T2959 Ginsenoside Rh2 Ginsenoside Rh2, an extract of red Panax ginseng, is a potent anti-inflammatory and a... Cancer
T2859 Biochanin A Biochanin A is an isoflavone derivative isolated from red clover Trifolium pratense w... Metabolism system
T2851 Daphnetin Daphnetin, a natural coumarin derivative, is a protein kinase inhibitor with inhibito... Cancer