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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T12228 Niperotidine 84845-75-0 98%
Niperotidine
Niperotidine is an antagonist of histamine H2-receptor.
T10575 BMY-25271 78441-82-4 98%
BMY-25271
BMY-25271 is an antagonist of histamine H2 receptor.
T11532 H4R antagonist 1 1429375-54-1 98%
H4R antagonist 1
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
TN5279 Zeorin 22570-53-2 98%
Zeorin
Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
T12756 ROS 234 dioxalate 1781941-93-2 98%
ROS 234 dioxalate
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
T13040 SUN 1334H 607736-84-5 98%
SUN 1334H
SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
T11531 H3R-IN-1 Hydrochloride 2319790-07-1 98%
H3R-IN-1 Hydrochloride
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
TN1913 Marmin 14957-38-1 98%
Marmin
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
TN3062 4'-O-Methylnyasol 79004-25-4 98%
4'-O-Methylnyasol
4'-O-Methylnyasol may have potential to be developed as medicines for the treatment of allergies by inhibiting the activation of mast cells.
T19604 WZ4141 1222776-76-2 98%
WZ4141
WZ4141 is an intermediate in compound synthesis.
T11324 FRG8701 108498-50-6 98%
FRG8701
FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
TN2895 3,5-Dicaffeoyl-epi-quinic acid 879305-14-3 98%
3,5-Dicaffeoyl-epi-quinic acid
3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
T10911 H3 receptor antagonist 1 935840-13-4 98%
H3 receptor antagonist 1
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
T15565 Imetit dihydrobromide 32385-58-3 98%
Imetit dihydrobromide
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
T4099 S 38093 862896-30-8 99.98%
S 38093
S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
T1619 Trazodone hydrochloride 25332-39-2 99.98%
Trazodone hydrochloride
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients wi...
TN1154 Nepetin 520-11-6 99.96%
Nepetin
Nepetin (6-Methoxyluteolin) has antioxidant activity, it is a potent inhibitor of histamine release and calcium influx via down-regulation of the FcεRI α chain.
T0468 Lidocaine 137-58-6 99.95%
Lidocaine
Lidocaine (Alphacaine) is an amide local anesthetic with anti-inflammatory properties in vitro and in vivo. It has this functions perhaps due to an attenuation o...
T4499 Mequitazine 29216-28-2 99.95%
Mequitazine
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
T8822 JNJ-5207852 dihydrochloride 1782228-76-5 99.95%
JNJ-5207852 dihydrochloride
JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor....
Niperotidine
T12228
Niperotidine is an antagonist of histamine H2-receptor.
BMY-25271
T10575
BMY-25271 is an antagonist of histamine H2 receptor.
H4R antagonist 1
T11532
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to ot...
Zeorin
TN5279
Zeorin shows strong inhibition activity against bacteria and fungi. It markedly exhibits inhibitory activity on histamine release from mast cell induced by DNP24...
ROS 234 dioxalate
T12756
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
SUN 1334H
T13040
SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
H3R-IN-1 Hydrochloride
T11531
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
Marmin
TN1913
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and sec...
4'-O-Methylnyasol
TN3062
4'-O-Methylnyasol may have potential to be developed as medicines for the treatment of allergies by inhibiting the activation of mast cells.
WZ4141
T19604
WZ4141 is an intermediate in compound synthesis.
FRG8701
T11324
FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
3,5-Dicaffeoyl-epi-quinic acid
TN2895
3,5-Dicaffeoyl-epi-quinic acid shows anti-inflammatory activity, it may improve mast cell-mediated inflammatory diseases.
H3 receptor antagonist 1
T10911
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
Imetit dihydrobromide
T15565
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in trigg...
S 38093
T4099
S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
Trazodone hydrochloride
T1619
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients wi...
Nepetin
TN1154
Nepetin (6-Methoxyluteolin) has antioxidant activity, it is a potent inhibitor of histamine release and calcium influx via down-regulation of the FcεRI α chain.
Lidocaine
T0468
Lidocaine (Alphacaine) is an amide local anesthetic with anti-inflammatory properties in vitro and in vivo. It has this functions perhaps due to an attenuation o...
Mequitazine
T4499
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
JNJ-5207852 dihydrochloride
T8822
JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor....
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TargetMol