TN4298 |
Isohyenanchin
|
19417-00-6
|
98%
|
|
Isohyenanchin is the potent antagonist of RDLac homo-oligomers, it is also a weak antagonist of ionotropic GABA receptors.
|
T12044 |
(-)-Bicuculline methochloride
|
53552-05-9
|
98%
|
|
(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.
|
T3927 |
Phellopterin
|
2543-94-4
|
98%
|
|
Phellopterin is a partial agonist of the central benzodiazepine receptors in vitro. Phellopterin shows a cytotoxic effect on RAW264.7 cell at the concentration f...
|
T2850 |
Bicuculline
|
485-49-4
|
98%
|
|
Bicuculline is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and has been isolated...
|
T1396 |
Bemegride
|
64-65-3
|
98%
|
|
Bemegride is a central nervous system stimulant and antidote for barbiturate poisoning.
|
T8572 |
CL 218872
|
66548-69-4
|
98%
|
|
CL 218872 is a benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 n...
|
T2S1464 |
Thiocolchicoside
|
602-41-5
|
98%
|
|
Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonis...
|
T5375 |
Loreclezole
|
117857-45-1
|
98%
|
|
Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.
|
T8639 |
Phenibut (hydrochloride)
|
3060-41-1
|
98%
|
|
Phenibut (hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing voltage-gated calcium channels, stimulates d...
|
T13536 |
Afoxolaner
|
1093861-60-9
|
98%
|
|
Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs. Afoxolaner acts on the insect GABA and glutamate receptors, inhibiting GABA...
|
T7699 |
AZD7325
|
942437-37-8
|
98%
|
|
AZD-7325 is a GABA-Aα2,3 -selective receptor modulator.
|
T4590 |
(+)-Kavain
|
500-64-1
|
98%
|
|
Kawain is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.
|
T8036 |
6-Methylflavone
|
29976-75-8
|
98%
|
|
6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.
|
T1065 |
Baclofen
|
1134-47-0
|
98%
|
|
Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing Baclofen act...
|
T8630 |
Baclofen hydrochloride
|
28311-31-1
|
98%
|
|
Baclofen hydrochloride is a GAMMA-AMINOBUTYRIC ACID derivative that is a specific GABA-B RECEPTORS agonist. It is used in the treatment of MUSCLE SPASTICITY, esp...
|
T11349 |
GABAA receptor agent 1
|
1571-87-5
|
98%
|
|
GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.
|
T11307 |
Fluxametamide
|
928783-29-3
|
98%
|
|
Fluxametamide is a novel isoxazoline insecticide that acts via distinctive antagonism of insect ligand-gated chloride channels, acts as an antagonist of GABA- an...
|
T0349 |
Riluzole
|
1744-22-5
|
98%
|
|
Riluzole is a glutamate antagonist (RECEPTORS, GLUTAMATE) used as an anticonvulsant (ANTICONVULSANTS) and to prolong the survival of patients with AMYOTROPHIC LA...
|
T4728 |
4-Acetamidobutanoic acid
|
3025-96-5
|
98%
|
|
4-Acetamidobutanoic acid can be found in blood, feces, and urine, as well as in human prostate tissue. 4-Acetamidobutanoic acid exists in all eukaryotes, ranging...
|
T2940 |
6-Hydroxyflavone
|
6665-83-4
|
98%
|
|
6-Hydroxyflavone is a noncompetitive inhibitors of cytochrome P450 2C9. It is a flavone, a type of chemical compound. It is reported in leaves of Barleria prioni...
|