T0076 |
Paliperidone
|
144598-75-4
|
96.98%
|
|
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically,...
|
T8044 |
Ajmalicine
|
483-04-5
|
96.9%
|
|
Ajmalicine (Raubasine) (Raubasine) is a potent adrenolytic agent which preferentially blocks α1-adrenoceptor. Ajmalicine is an reversible but non-competitive nic...
|
T6579 |
Medetomidine hydrochloride
|
86347-15-1
|
96.72%
|
|
Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
|
T37906 |
Dibenamine hydrochloride
|
55-43-6
|
96.43%
|
|
Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.
|
T8580 |
Bupranolol
|
14556-46-8
|
95.85%
|
|
Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic....
|
T0445L |
Promethazine hydrochloride
|
58-33-3
|
95.36%
|
|
Promethazine hydrochloride (Promethazine HCl) , the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mA...
|
TN1015 |
Meranzin
|
23971-42-8
|
95.08%
|
|
Meranzin, a bioactive compound derived from the Traditional Chinese Medicine (TCM) Chaihu-Shugan-San (CSS) and isolated from Murraya exotica L. leaves, targets t...
|
T10364 |
Arbutamine
|
128470-16-6
|
95.06%
|
|
Arbutamine (GP 21213) is a novel potent non-selective beta-adrenoceptor agonist with alpha-1-sympathomimetic activity.Arbutamine promotes cardiac stress and incr...
|
T50081 |
Tiprenolol
|
26481-51-6
|
95.00%
|
|
Tiprenolol is a beta adrenergic receptor antagonist.[1]
|
T12343 |
Benzquinamide
|
63-12-7
|
94.86%
|
|
Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer ...
|
T0185 |
Escitalopram
|
128196-01-0
|
94.62%
|
|
Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing e...
|
T15688 |
L-771688
|
200050-59-5
|
94.15%
|
|
L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benign ...
|
T1680 |
Tolazoline hydrochloride
|
59-97-2
|
100%
|
|
Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hyp...
|
T16431 |
Pamatolol
|
59110-35-9
|
100%
|
|
Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.
|
T0173 |
Nylidrin hydrochloride
|
849-55-8
|
100%
|
|
Nylidrin hydrochloride (Buphenine HCl) was an effective inhibitor of the IgG1-mediated release of histamine from passively sensitized guinea pig lung slices, and...
|
T8304 |
Anisodamine Hydrobromide
|
55449-49-5
|
100%
|
|
Anisodamine Hydrobromide (6-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
|
T1056 |
Isoprenaline hydrochloride
|
51-30-9
|
100%
|
|
Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
|
T1180 |
Blonanserin
|
132810-10-7
|
100%
|
|
Blonanserin (AD-5423) is an atypical antipsychotic approved in Japan in January, 2008. Relative to many other antipsychotics, blonanserin has an improved tolerab...
|
T1132 |
Nicergoline
|
27848-84-6
|
100%
|
|
Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
|
T2320 |
Indacaterol
|
312753-06-3
|
100%
|
|
Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.
|