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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
TP1902L1 G-Protein antagonist peptide acetate 98.06%
G-Protein antagonist peptide acetate
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide aceta...
T1158 Phenoxybenzamine hydrochloride 63-92-3 98.04%
Phenoxybenzamine hydrochloride
Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihyp...
T21787L Azepexole hydrochloride 147663-20-5 98.03%
Azepexole hydrochloride
Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic ...
T1045 Trimipramine maleate 521-78-8 98.02%
Trimipramine maleate
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepineph...
T6860 (RS)-ICI-118551 Hydrochloride 1217094-53-5 98.02%
(RS)-ICI-118551 Hydrochloride
ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors...
T21371 Apraclonidine hydrochloride 73218-79-8 98.01%
Apraclonidine hydrochloride
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist. Apraclonidine hydrochloride lowers intraocular pre...
T0394 Moxisylyte hydrochloride 964-52-3 98%
Moxisylyte hydrochloride
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
T1287 Synephrine 94-07-5 98%
Synephrine
Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
T1504 Silodosin 160970-54-7 98%
Silodosin
Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
T1459 Cisatracurium besylate 96946-42-8 98%
Cisatracurium besylate
Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.
T0365 Thioridazine hydrochloride 130-61-0 98%
Thioridazine hydrochloride
Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selecti...
T6641 Rilmenidine Phosphate 85409-38-7 98%
Rilmenidine Phosphate
Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.
T3158 Harmane 486-84-0 97.89%
Harmane
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T11726 JP1302 dihydrochloride 1259314-65-2 97.83%
JP1302 dihydrochloride
JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a...
T3046 BMY 7378 dihydrochloride 21102-95-4 97.67%
BMY 7378 dihydrochloride
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
T6241 Quetiapine hemifumarate 111974-72-2 97.63%
Quetiapine hemifumarate
Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I dep...
T0446 Naphazoline hydrochloride 550-99-2 97.6%
Naphazoline hydrochloride
Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant.
T68164 Tolamolol 38103-61-6 97.58%
Tolamolol
Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in the trea...
T70047 Bedoradrine 194785-19-8 97.53%
Bedoradrine
Bedoradrine free base is a novel, highly selective β2-adrenoceptor agonist for the treatment of asthma and chronic obstructive pulmonary disease (COPD).
T28829 Soquinolol 61563-18-6 97.48%
Soquinolol
Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long durat...
G-Protein antagonist peptide acetate
TP1902L1
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide aceta...
Phenoxybenzamine hydrochloride
T1158
Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihyp...
Azepexole hydrochloride
T21787L
Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic ...
Trimipramine maleate
T1045
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepineph...
(RS)-ICI-118551 Hydrochloride
T6860
ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors...
Apraclonidine hydrochloride
T21371
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist. Apraclonidine hydrochloride lowers intraocular pre...
Moxisylyte hydrochloride
T0394
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
Synephrine
T1287
Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
Silodosin
T1504
Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
Cisatracurium besylate
T1459
Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.
Thioridazine hydrochloride
T0365
Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selecti...
Rilmenidine Phosphate
T6641
Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.
Harmane
T3158
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
JP1302 dihydrochloride
T11726
JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a...
BMY 7378 dihydrochloride
T3046
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
Quetiapine hemifumarate
T6241
Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I dep...
Naphazoline hydrochloride
T0446
Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant.
Tolamolol
T68164
Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in the trea...
Bedoradrine
T70047
Bedoradrine free base is a novel, highly selective β2-adrenoceptor agonist for the treatment of asthma and chronic obstructive pulmonary disease (COPD).
Soquinolol
T28829
Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long durat...
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TargetMol