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arg131

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  • Inhibitors & Agonists
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    TargetMol | Inhibitors_Agonists
PS210
T166701221962-86-2
PS210 is a potent and selective activator of PDK1 (Kd: 3 μM), specifically targeting the PIF-binding pocket of PDK1 without affecting other protein kinases such as S6K, PKB Akt, or GSK3. Its prodrug, PS423, serves as a substrate-selective inhibitor of PDK1 in cells, inhibiting the phosphorylation and activation of S6K.
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(R)-PS210
T126391410101-89-1
(R)-PS210, the R enantiomer of PS210, is a substrate-selective allosteric PDK1 activator with an (AC50 of 1.8 μM).
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6-8 weeks
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