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  • Drug-Linker Conjugates for ADC
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2247398-68-9

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Py-MAA-Val-Cit-PAB-MMAE
AAJ8D6-PY-Val-Cit-MMAE
T778762247398-68-9
Py-MAA-Val-Cit-PAB-MMAE (AAJ8D6-PY-Val-Cit-MMAE) serves as an ADC linker for Zapadcine-3a, a broad-spectrum anti-TRAILR2 ADC with antineoplastic properties. Targeting TRAILR2, Zapadcine-3a is internalized into tumor cell lysosomes, releasing a small molecular compound that selectively eradicates TRAILR2-positive tumor cells, potentially leading to tumor remission [1].
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8-10 weeks
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